These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

131 related articles for article (PubMed ID: 17251015)

  • 1. Opioids and efflux transporters. Part 1: P-glycoprotein substrate activity of N-substituted analogs of meperidine.
    Mercer SL; Hassan HE; Cunningham CW; Eddington ND; Coop A
    Bioorg Med Chem Lett; 2007 Mar; 17(5):1160-2. PubMed ID: 17251015
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Opioids and efflux transporters. Part 3: P-glycoprotein substrate activity of 3-hydroxyl addition to meperidine analogs.
    Mercer SL; Cunningham CW; Eddington ND; Coop A
    Bioorg Med Chem Lett; 2008 Jun; 18(12):3638-40. PubMed ID: 18499452
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Evaluation of the P-glycoprotein (Abcb1) affinity status of a series of morphine analogs: comparative study with meperidine analogs to identify opioids with minimal P-glycoprotein interactions.
    Hassan HE; Mercer SL; Cunningham CW; Coop A; Eddington ND
    Int J Pharm; 2009 Jun; 375(1-2):48-54. PubMed ID: 19481690
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Opioids and efflux transporters. Part 2: P-glycoprotein substrate activity of 3- and 6-substituted morphine analogs.
    Cunningham CW; Mercer SL; Hassan HE; Traynor JR; Eddington ND; Coop A
    J Med Chem; 2008 Apr; 51(7):2316-20. PubMed ID: 18311899
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Opioid analgesics and P-glycoprotein efflux transporters: a potential systems-level contribution to analgesic tolerance.
    Mercer SL; Coop A
    Curr Top Med Chem; 2011; 11(9):1157-64. PubMed ID: 21050174
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Opioids and efflux transporters. Part 4: influence of N-substitution on P-glycoprotein substrate activity of noroxymorphone analogues.
    Metcalf MD; Rosicky AD; Hassan HE; Eddington ND; Coop A; Cunningham CW; Mercer SL
    Bioorg Med Chem Lett; 2014 Aug; 24(15):3592-5. PubMed ID: 24915880
    [TBL] [Abstract][Full Text] [Related]  

  • 7. P-glycoprotein ATPase activating effect of opioid analgesics and their P-glycoprotein-dependent antinociception in mice.
    Hamabe W; Maeda T; Fukazawa Y; Kumamoto K; Shang LQ; Yamamoto A; Yamamoto C; Tokuyama S; Kishioka S
    Pharmacol Biochem Behav; 2006 Nov; 85(3):629-36. PubMed ID: 17134744
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Variable modulation of opioid brain uptake by P-glycoprotein in mice.
    Dagenais C; Graff CL; Pollack GM
    Biochem Pharmacol; 2004 Jan; 67(2):269-76. PubMed ID: 14698039
    [TBL] [Abstract][Full Text] [Related]  

  • 9. The Impact of P-Glycoprotein on Opioid Analgesics: What's the Real Meaning in Pain Management and Palliative Care?
    Coluzzi F; Scerpa MS; Rocco M; Fornasari D
    Int J Mol Sci; 2022 Nov; 23(22):. PubMed ID: 36430602
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Differential involvement of P-glycoprotein (ABCB1) in permeability, tissue distribution, and antinociceptive activity of methadone, buprenorphine, and diprenorphine: in vitro and in vivo evaluation.
    Hassan HE; Myers AL; Coop A; Eddington ND
    J Pharm Sci; 2009 Dec; 98(12):4928-40. PubMed ID: 19370547
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and structure-activity studies of benzyl ester meperidine and normeperidine derivatives as selective serotonin transporter ligands.
    Gu X; Izenwasser S; Wade D; Housman A; Gulasey G; Rhoden JB; Savoie CD; Mobley DL; Lomenzo SA; Trudell ML
    Bioorg Med Chem; 2010 Dec; 18(23):8356-64. PubMed ID: 20980153
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Opioids and the Blood-Brain Barrier: A Dynamic Interaction with Consequences on Drug Disposition in Brain.
    Chaves C; Remiao F; Cisternino S; Decleves X
    Curr Neuropharmacol; 2017 Nov; 15(8):1156-1173. PubMed ID: 28474563
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis and antinociceptive activity of 4-pyridyl and -dihydropyridyl analogues of meperidine and ketobemidone.
    Buolamwini JK; Knaus EE
    Drug Des Deliv; 1990 Dec; 7(1):19-31. PubMed ID: 1982918
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Competitive substrates for P-glycoprotein and organic anion protein transporters differentially reduce blood organ transport of fentanyl and loperamide: pharmacokinetics and pharmacodynamics in Sprague-Dawley rats.
    Elkiweri IA; Zhang YL; Christians U; Ng KY; Tissot van Patot MC; Henthorn TK
    Anesth Analg; 2009 Jan; 108(1):149-59. PubMed ID: 19095843
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Opiate-induced analgesia is increased and prolonged in mice lacking P-glycoprotein.
    Thompson SJ; Koszdin K; Bernards CM
    Anesthesiology; 2000 May; 92(5):1392-9. PubMed ID: 10781286
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Modification of behavioral effects of morphine, meperidine and normeperidine by naloxone and by morphine tolerance.
    Witkin JM; Leander JD; Dykstra LA
    J Pharmacol Exp Ther; 1983 May; 225(2):275-83. PubMed ID: 6842391
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Chronic morphine exposure potentiates p-glycoprotein trafficking from nuclear reservoirs in cortical rat brain microvessels.
    Schaefer CP; Arkwright NB; Jacobs LM; Jarvis CK; Hunn KC; Largent-Milnes TM; Tome ME; Davis TP
    PLoS One; 2018; 13(2):e0192340. PubMed ID: 29414996
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Correlation of opiate receptor affinity with analgetic effects of meperidine homologues.
    Pert CB; Snyder SH
    J Med Chem; 1976 Oct; 19(10):1248-50. PubMed ID: 11345
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Structure-activity studies of 3'-4'-dichloro-meperidine analogues at dopamine and serotonin transporters.
    Rhoden JB; Bouvet M; Izenwasser S; Wade D; Lomenzo SA; Trudell ML
    Bioorg Med Chem; 2005 Oct; 13(19):5623-34. PubMed ID: 15993612
    [TBL] [Abstract][Full Text] [Related]  

  • 20. (18)F-FCWAY, a serotonin 1A receptor radioligand, is a substrate for efflux transport at the human blood-brain barrier.
    Liow JS; Zoghbi SS; Hu S; Hall MD; Hines CS; Shetty HU; Araneta MD; Page EM; Pike VW; Kreisl WC; Herscovitch P; Gottesman MM; Theodore WH; Innis RB
    Neuroimage; 2016 Sep; 138():134-140. PubMed ID: 27211474
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.