These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

125 related articles for article (PubMed ID: 17303428)

  • 1. Novel chiral isoxazole derivatives: synthesis and pharmacological characterization at human beta-adrenergic receptor subtypes.
    Dallanoce C; Frigerio F; De Amici M; Dorsch S; Klotz KN; De Micheli C
    Bioorg Med Chem; 2007 Apr; 15(7):2533-43. PubMed ID: 17303428
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis of enantiopure Delta2-isoxazoline derivatives and evaluation of their affinity and efficacy profiles at human beta-adrenergic receptor subtypes.
    Dallanoce C; Meroni G; De Amici M; Hoffmann C; Klotz KN; De Micheli C
    Bioorg Med Chem; 2006 Jul; 14(13):4393-401. PubMed ID: 16530417
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Isomeric-activity ratios of trimetoquinol enantiomers on beta-adrenergic receptor subtypes: functional and biochemical studies.
    Fraundorfer PF; Lezama EJ; Salazar-Bookaman MM; Fertel RH; Miller DD; Feller DR
    Chirality; 1994; 6(2):76-85. PubMed ID: 7911313
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Biochemical and pharmacological characterization of high-affinity trimetoquinol analogs on guinea pig and human beta adrenergic receptor subtypes: evidence for partial agonism.
    Fraundorfer PF; Fertel RH; Miller DD; Feller DR
    J Pharmacol Exp Ther; 1994 Aug; 270(2):665-74. PubMed ID: 7915318
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Comparison of the binding affinity of some newly synthesized phenylethanolamine and phenoxypropanolamine compounds at recombinant human beta- and alpha1-adrenoceptor subtypes.
    Ahmed M; Hanaoka Y; Kiso T; Kakita T; Ohtsubo Y; Muramatsu I; Nagatomo T
    J Pharm Pharmacol; 2005 Jan; 57(1):75-81. PubMed ID: 15638996
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Characterization of a new, highly specific, beta 3-adrenergic receptor radioligand, [3H]SB 206606.
    Muzzin P; Boss O; Mathis N; Revelli JP; Giacobino JP; Willcocks K; Badman GT; Cantello BC; Hindley RM; Cawthorne MA
    Mol Pharmacol; 1994 Aug; 46(2):357-63. PubMed ID: 8078497
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Novel isoxazole carboxamides as growth hormone secretagogue receptor (GHS-R) antagonists.
    Liu B; Liu G; Xin Z; Serby MD; Zhao H; Schaefer VG; Falls HD; Kaszubska W; Collins CA; Sham HL
    Bioorg Med Chem Lett; 2004 Oct; 14(20):5223-6. PubMed ID: 15380232
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis, binding affinity at glutamic acid receptors, neuroprotective effects, and molecular modeling investigation of novel dihydroisoxazole amino acids.
    Conti P; De Amici M; Grazioso G; Roda G; Pinto A; Hansen KB; Nielsen B; Madsen U; Bräuner-Osborne H; Egebjerg J; Vestri V; Pellegrini-Giampietro DE; Sibille P; Acher FC; De Micheli C
    J Med Chem; 2005 Oct; 48(20):6315-25. PubMed ID: 16190758
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Structure-activity relationship studies of phenoxypropanolamine derivatives for beta 3-adrenergic activity.
    Ahmed M; Hanaoka Y; Nagatomo T
    Nihon Yakurigaku Zasshi; 2002 Nov; 120(1):112P-113P. PubMed ID: 12491799
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis and pharmacological characterization at glutamate receptors of the four enantiopure isomers of tricholomic acid.
    Pinto A; Conti P; De Amici M; Tamborini L; Madsen U; Nielsen B; Christesen T; Bräuner-Osborne H; De Micheli C
    J Med Chem; 2008 Apr; 51(7):2311-5. PubMed ID: 18338843
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Novel diastereomeric opioid tetrapeptides exhibit differing pharmacological activity profiles.
    Ioja E; Tourwé D; Kertész I; Tóth G; Borsodi A; Benyhe S
    Brain Res Bull; 2007 Sep; 74(1-3):119-29. PubMed ID: 17683797
    [TBL] [Abstract][Full Text] [Related]  

  • 12. The beta3-adrenoceptor agonist 4-[[(Hexylamino)carbonyl]amino]-N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]-phenyl]-benzenesulfonamide (L755507) and antagonist (S)-N-[4-[2-[[3-[3-(acetamidomethyl)phenoxy]-2-hydroxypropyl]amino]-ethyl]phenyl]benzenesulfonamide (L748337) activate different signaling pathways in Chinese hamster ovary-K1 cells stably expressing the human beta3-adrenoceptor.
    Sato M; Hutchinson DS; Evans BA; Summers RJ
    Mol Pharmacol; 2008 Nov; 74(5):1417-28. PubMed ID: 18684840
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Are so many adrenergic receptor subtypes really present in domestic animal tissues? A pharmacological perspective.
    Badino P; Odore R; Re G
    Vet J; 2005 Sep; 170(2):163-74. PubMed ID: 16129337
    [TBL] [Abstract][Full Text] [Related]  

  • 14. High-throughput screening with a miniaturized radioligand competition assay identifies new modulators of human α2-adrenoceptors.
    Fallarero A; Pohjanoksa K; Wissel G; Parkkisenniemi-Kinnunen UM; Xhaard H; Scheinin M; Vuorela P
    Eur J Pharm Sci; 2012 Dec; 47(5):941-51. PubMed ID: 22982401
    [TBL] [Abstract][Full Text] [Related]  

  • 15. New isoxazole derivatives with a potent and selective beta 2-adrenergic activity.
    Chiarino D; Fantucci M; Carenzi A; Della Bella D; Frigeni V; Sala R
    Farmaco Sci; 1986 Jun; 41(6):440-53. PubMed ID: 2874994
    [TBL] [Abstract][Full Text] [Related]  

  • 16. N6-Cycloalkyl- and N6-bicycloalkyl-C5'(C2')-modified adenosine derivatives as high-affinity and selective agonists at the human A1 adenosine receptor with antinociceptive effects in mice.
    Franchetti P; Cappellacci L; Vita P; Petrelli R; Lavecchia A; Kachler S; Klotz KN; Marabese I; Luongo L; Maione S; Grifantini M
    J Med Chem; 2009 Apr; 52(8):2393-406. PubMed ID: 19317449
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Pharmacological properties of Chinese hamster ovary cells coexpressing two vasoactive intestinal peptide receptors (hVPAC1 and hVPAC2).
    Langer I; Gaspard N; Robberecht P
    Br J Pharmacol; 2006 Aug; 148(8):1051-9. PubMed ID: 16783404
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Stereospecific synthesis and bio-activity of novel beta(3)-adrenoceptor agonists and inverse agonists.
    Perrone MG; Santandrea E; Bleve L; Vitale P; Colabufo NA; Jockers R; Milazzo FM; Sciarroni AF; Scilimati A
    Bioorg Med Chem; 2008 Mar; 16(5):2473-88. PubMed ID: 18083578
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Tethered yohimbine analogs as selective human alpha2C-adrenergic receptor ligands.
    Bavadekar SA; Ma G; Mustafa SM; Moore BM; Miller DD; Feller DR
    J Pharmacol Exp Ther; 2006 Nov; 319(2):739-48. PubMed ID: 16873606
    [TBL] [Abstract][Full Text] [Related]  

  • 20. GW427353 (solabegron), a novel, selective beta3-adrenergic receptor agonist, evokes bladder relaxation and increases micturition reflex threshold in the dog.
    Hicks A; McCafferty GP; Riedel E; Aiyar N; Pullen M; Evans C; Luce TD; Coatney RW; Rivera GC; Westfall TD; Hieble JP
    J Pharmacol Exp Ther; 2007 Oct; 323(1):202-9. PubMed ID: 17626794
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.