These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

128 related articles for article (PubMed ID: 17379515)

  • 1. Synthesis, characterization, and estrogen receptor binding affinity of flavone-, indole-, and furan-estradiol conjugates.
    Ahmed N; Dubuc C; Rousseau J; Bénard F; van Lier JE
    Bioorg Med Chem Lett; 2007 Jun; 17(11):3212-6. PubMed ID: 17379515
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and biological activities of nucleoside-estradiol conjugates.
    Ali H; Ahmed N; Tessier G; van Lier JE
    Bioorg Med Chem Lett; 2006 Jan; 16(2):317-9. PubMed ID: 16275069
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Selective estrogen receptor modulators with conformationally restricted side chains. Synthesis and structure-activity relationship of ERalpha-selective tetrahydroisoquinoline ligands.
    Renaud J; Bischoff SF; Buhl T; Floersheim P; Fournier B; Geiser M; Halleux C; Kallen J; Keller H; Ramage P
    J Med Chem; 2005 Jan; 48(2):364-79. PubMed ID: 15658851
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and evaluation of 17alpha-20E-21-(4-substituted phenyl)-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diols as probes for the estrogen receptor alpha hormone binding domain.
    Hanson RN; Lee CY; Friel CJ; Dilis R; Hughes A; DeSombre ER
    J Med Chem; 2003 Jul; 46(14):2865-76. PubMed ID: 12825929
    [TBL] [Abstract][Full Text] [Related]  

  • 5. New scaffolds for the design of selective estrogen receptor modulators.
    Martín-Santamaría S; Rodríguez JJ; de Pascual-Teresa S; Gordon S; Bengtsson M; Garrido-Laguna I; Rubio-Viqueira B; López-Casas PP; Hidalgo M; de Pascual-Teresa B; Ramos A
    Org Biomol Chem; 2008 Oct; 6(19):3486-96. PubMed ID: 19082149
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Discovery of novel quinoline-based estrogen receptor ligands using peptide interaction profiling.
    Hoekstra WJ; Patel HS; Liang X; Blanc JB; Heyer DO; Willson TM; Iannone MA; Kadwell SH; Miller LA; Pearce KH; Simmons CA; Shearin J
    J Med Chem; 2005 Mar; 48(6):2243-7. PubMed ID: 15771467
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Improved synthesis of unique estradiol-linked platinum(II) complexes showing potent cytocidal activity and affinity for the estrogen receptor alpha and beta.
    Descôteaux C; Leblanc V; Bélanger G; Parent S; Asselin E; Bérubé G
    Steroids; 2008 Oct; 73(11):1077-89. PubMed ID: 18572212
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Benzopyrans are selective estrogen receptor beta agonists with novel activity in models of benign prostatic hyperplasia.
    Norman BH; Dodge JA; Richardson TI; Borromeo PS; Lugar CW; Jones SA; Chen K; Wang Y; Durst GL; Barr RJ; Montrose-Rafizadeh C; Osborne HE; Amos RM; Guo S; Boodhoo A; Krishnan V
    J Med Chem; 2006 Oct; 49(21):6155-7. PubMed ID: 17034120
    [TBL] [Abstract][Full Text] [Related]  

  • 9. QSAR of estrogen receptor modulators: exploring selectivity requirements for ER(alpha) versus ER(beta) binding of tetrahydroisoquinoline derivatives using E-state and physicochemical parameters.
    Mukherjee S; Saha A; Roy K
    Bioorg Med Chem Lett; 2005 Feb; 15(4):957-61. PubMed ID: 15686893
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Novel estradiol derivatives labeled with Ru, W, and Co complexes. Influence on hormone-receptor affinity of several organometallic groups at the 17 alpha position.
    Top S; el Hafa H; Vessiéres A; Huché M; Vaissermann J; Jaouen G
    Chemistry; 2002 Nov; 8(22):5241-9. PubMed ID: 12613043
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Benzothieno[3,2-b]indole derivatives as potent selective estrogen receptor modulators.
    Ji Q; Gao J; Wang J; Yang C; Hui X; Yan X; Wu X; Xie Y; Wang MW
    Bioorg Med Chem Lett; 2005 Jun; 15(11):2891-3. PubMed ID: 15911274
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Rapid synthesis of 4-benzylidene and 4-[bis-(4-methoxyphenyl)-methylene-2-substituted phenyl-benzopyrans as potential selective estrogen receptor modulators (SERMs) using McMurry coupling reaction.
    Gupta A; Dwivedy A; Keshri G; Sharma R; Balapure AK; Singh MM; Ray S
    Bioorg Med Chem Lett; 2006 Dec; 16(23):6006-12. PubMed ID: 16979337
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis, receptor binding, molecular modeling, and proliferative assays of a series of 17alpha-arylestradiols.
    Foy N; Stéphan E; Vessières A; Salomon E; Heldt JM; Huché M; Jaouen G
    Chembiochem; 2003 Jun; 4(6):494-503. PubMed ID: 12794859
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Fluorous tolerance of the estrogen receptor alpha as probed by 11-polyfluoroalkylestradiol derivatives.
    Agouridas V; Blazejewski JC; Cleeren A; Laïos I; Leclercq G; Magnier E
    Steroids; 2008 Mar; 73(3):320-7. PubMed ID: 18177682
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Lead identification of a potent benzopyranone selective estrogen receptor modulator.
    McKie JA; Bhagwat SS; Brady H; Doubleday M; Gayo L; Hickman M; Jalluri RK; Khammungkhune S; Kois A; Mortensen D; Richard N; Sapienza J; Shevlin G; Stein B; Sutherland M
    Bioorg Med Chem Lett; 2004 Jul; 14(13):3407-10. PubMed ID: 15177442
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Estradiol derivatives bearing sulfur-containing substituents at the 11beta or 7alpha positions: versatile reagents for the preparation of estrogen conjugates.
    Spera D; Cabrera G; Fiaschi R; Carlson KE; Katzenellenbogen JA; Napolitano E
    Bioorg Med Chem; 2004 Aug; 12(16):4393-401. PubMed ID: 15265491
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and biological activities of phthalocyanine-estradiol conjugates.
    Khan EH; Ali H; Tian H; Rousseau J; Tessier G; Shafiullah ; van Lier JE
    Bioorg Med Chem Lett; 2003 Apr; 13(7):1287-90. PubMed ID: 12657265
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Benzothiophenes containing a piperazine side chain as selective ligands for the estrogen receptor alpha and their bioactivities in vivo.
    Yang C; Xu G; Li J; Wu X; Liu B; Yan X; Wang M; Xie Y
    Bioorg Med Chem Lett; 2005 Mar; 15(5):1505-7. PubMed ID: 15713417
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and evaluation of (17alpha,20Z)-21-(4-substituted-phenyl)-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diols as ligands for the estrogen receptor-alpha hormone binding domain: comparison with 20E-isomers.
    Hanson RN; Friel CJ; Dilis R; Hughes A; DeSombre ER
    J Med Chem; 2005 Jun; 48(13):4300-11. PubMed ID: 15974584
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Novel 7α-alkoxy-17α-(4'-halophenylethynyl)estradiols as potential SPECT/PET imaging agents for estrogen receptor expressing tumours: synthesis and binding affinity evaluation.
    Neto C; Oliveira MC; Gano L; Marques F; Yasuda T; Thiemann T; Kniess T; Santos I
    Steroids; 2012 Sep; 77(11):1123-32. PubMed ID: 22633985
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.