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4. Analogs of the antituberculous agent pyrazinamide are competitive inhibitors of NADPH binding to M. tuberculosis fatty acid synthase I. Sayahi H; Pugliese KM; Zimhony O; Jacobs WR; Shekhtman A; Welch JT Chem Biodivers; 2012 Nov; 9(11):2582-96. PubMed ID: 23161636 [TBL] [Abstract][Full Text] [Related]
5. Pyrazinoic acid and its n-propyl ester inhibit fatty acid synthase type I in replicating tubercle bacilli. Zimhony O; Vilchèze C; Arai M; Welch JT; Jacobs WR Antimicrob Agents Chemother; 2007 Feb; 51(2):752-4. PubMed ID: 17101678 [TBL] [Abstract][Full Text] [Related]
6. Pyrazinamide, but not pyrazinoic acid, is a competitive inhibitor of NADPH binding to Mycobacterium tuberculosis fatty acid synthase I. Sayahi H; Zimhony O; Jacobs WR; Shekhtman A; Welch JT Bioorg Med Chem Lett; 2011 Aug; 21(16):4804-7. PubMed ID: 21775138 [TBL] [Abstract][Full Text] [Related]
7. Mutually exclusive genotypes for pyrazinamide and 5-chloropyrazinamide resistance reveal a potential resistance-proofing strategy. Baughn AD; Deng J; Vilchèze C; Riestra A; Welch JT; Jacobs WR; Zimhony O Antimicrob Agents Chemother; 2010 Dec; 54(12):5323-8. PubMed ID: 20876380 [TBL] [Abstract][Full Text] [Related]
8. Effects of pyrazinamide on fatty acid synthesis by whole mycobacterial cells and purified fatty acid synthase I. Boshoff HI; Mizrahi V; Barry CE J Bacteriol; 2002 Apr; 184(8):2167-72. PubMed ID: 11914348 [TBL] [Abstract][Full Text] [Related]
9. Activity of n-propyl pyrazinoate against pyrazinamide-resistant Mycobacterium tuberculosis: investigations into mechanism of action of and mechanism of resistance to pyrazinamide. Speirs RJ; Welch JT; Cynamon MH Antimicrob Agents Chemother; 1995 Jun; 39(6):1269-71. PubMed ID: 7574514 [TBL] [Abstract][Full Text] [Related]
10. Pyrazinamide and Pyrazinoic Acid Derivatives Directed to Mycobacterial Enzymes Against Tuberculosis. Corrêa MF; Fernandes JP Curr Protein Pept Sci; 2016; 17(3):213-9. PubMed ID: 26427385 [TBL] [Abstract][Full Text] [Related]
11. Lipophilic pyrazinoic acid amide and ester prodrugs stability, activation and activity against M. tuberculosis. Simões MF; Valente E; Gómez MJ; Anes E; Constantino L Eur J Pharm Sci; 2009 Jun; 37(3-4):257-63. PubMed ID: 19491013 [TBL] [Abstract][Full Text] [Related]
12. Structural basis for targeting the ribosomal protein S1 of Mycobacterium tuberculosis by pyrazinamide. Yang J; Liu Y; Bi J; Cai Q; Liao X; Li W; Guo C; Zhang Q; Lin T; Zhao Y; Wang H; Liu J; Zhang X; Lin D Mol Microbiol; 2015 Mar; 95(5):791-803. PubMed ID: 25430994 [TBL] [Abstract][Full Text] [Related]
13. [Nutrient starved incubation conditions enhance pyrazinamide activity against Mycobacterium tuberculosis]. Chen ZF; Huang Q; Li YY; Zhang Y; Ren Y; Li KS; Fu ZJ; Xu SQ Zhonghua Jie He He Hu Xi Za Zhi; 2007 May; 30(5):359-62. PubMed ID: 17651643 [TBL] [Abstract][Full Text] [Related]
14. The paradox of pyrazinamide: an update on the molecular mechanisms of pyrazinamide resistance in Mycobacteria. Singh P; Mishra AK; Malonia SK; Chauhan DS; Sharma VD; Venkatesan K; Katoch VM J Commun Dis; 2006 Mar; 38(3):288-98. PubMed ID: 17373362 [TBL] [Abstract][Full Text] [Related]
15. Mycobacterium tuberculosis isolates from Rio de Janeiro reveal unusually low correlation between pyrazinamide resistance and mutations in the pncA gene. Bhuju S; Fonseca Lde S; Marsico AG; de Oliveira Vieira GB; Sobral LF; Stehr M; Singh M; Saad MH Infect Genet Evol; 2013 Oct; 19():1-6. PubMed ID: 23770140 [TBL] [Abstract][Full Text] [Related]
16. Does pyrazinoic acid as an active moiety of pyrazinamide have specific activity against Mycobacterium tuberculosis? Heifets LB; Flory MA; Lindholm-Levy PJ Antimicrob Agents Chemother; 1989 Aug; 33(8):1252-4. PubMed ID: 2508544 [TBL] [Abstract][Full Text] [Related]
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20. [A study of the bacteriophage-based assay for the detection of pyrazinamide resistance in Mycobacterium tuberculosis]. Ao JP; Chen JW; Hu ZY; Li JN; Wang J; Wang Q; Cui ZL; Zhang WH; Wong XH Zhonghua Jie He He Hu Xi Za Zhi; 2006 Sep; 29(9):625-8. PubMed ID: 17129472 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]