BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

191 related articles for article (PubMed ID: 17489570)

  • 1. The potential of transient receptor potential vanilloid type 1 channel modulators for the treatment of pain.
    Westaway SM
    J Med Chem; 2007 May; 50(11):2589-96. PubMed ID: 17489570
    [No Abstract]   [Full Text] [Related]  

  • 2. Therapeutic potential of vanilloid receptor TRPV1 agonists and antagonists as analgesics: Recent advances and setbacks.
    Wong GY; Gavva NR
    Brain Res Rev; 2009 Apr; 60(1):267-77. PubMed ID: 19150372
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Transient receptor potential vanilloid-1 antagonists: a survey of recent patent literature.
    Voight EA; Kort ME
    Expert Opin Ther Pat; 2010 Sep; 20(9):1107-22. PubMed ID: 20586701
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Discovery of novel 6,6-heterocycles as transient receptor potential vanilloid (TRPV1) antagonists.
    Blum CA; Caldwell T; Zheng X; Bakthavatchalam R; Capitosti S; Brielmann H; De Lombaert S; Kershaw MT; Matson D; Krause JE; Cortright D; Crandall M; Martin WJ; Murphy BA; Boyce S; Jones AB; Mason G; Rycroft W; Perrett H; Conley R; Burnaby-Davies N; Chenard BL; Hodgetts KJ
    J Med Chem; 2010 Apr; 53(8):3330-48. PubMed ID: 20307063
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Answering the burning question of how transient receptor potential vanilloid-1 channel antagonists cause unwanted hyperthermia.
    Ayoub SS; Hunter JC; Simmons DL
    Pharmacol Rev; 2009 Sep; 61(3):225-7. PubMed ID: 19805475
    [TBL] [Abstract][Full Text] [Related]  

  • 6. The vanilloid receptor TRPV1: 10 years from channel cloning to antagonist proof-of-concept.
    Szallasi A; Cortright DN; Blum CA; Eid SR
    Nat Rev Drug Discov; 2007 May; 6(5):357-72. PubMed ID: 17464295
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Clinical development of TRPV1 antagonists: targeting a pivotal point in the pain pathway.
    Gunthorpe MJ; Chizh BA
    Drug Discov Today; 2009 Jan; 14(1-2):56-67. PubMed ID: 19063991
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Adlea (ALGRX-4975), an injectable capsaicin (TRPV1 receptor agonist) formulation for longlasting pain relief.
    Remadevi R; Szallisi A
    IDrugs; 2008 Feb; 11(2):120-32. PubMed ID: 18240098
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Repeated administration of vanilloid receptor TRPV1 antagonists attenuates hyperthermia elicited by TRPV1 blockade.
    Gavva NR; Bannon AW; Hovland DN; Lehto SG; Klionsky L; Surapaneni S; Immke DC; Henley C; Arik L; Bak A; Davis J; Ernst N; Hever G; Kuang R; Shi L; Tamir R; Wang J; Wang W; Zajic G; Zhu D; Norman MH; Louis JC; Magal E; Treanor JJ
    J Pharmacol Exp Ther; 2007 Oct; 323(1):128-37. PubMed ID: 17652633
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Modulation of intracellular calcium influences capsaicin-induced currents of TRPV-1 and voltage-activated channel currents in nociceptive neurones.
    Hagenacker T; Büsselberg D
    J Peripher Nerv Syst; 2007 Dec; 12(4):277-84. PubMed ID: 18042138
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Estrogen amplifies pain responses to uterine cervical distension in rats by altering transient receptor potential-1 function.
    Yan T; Liu B; Du D; Eisenach JC; Tong C
    Anesth Analg; 2007 May; 104(5):1246-50, tables of contents. PubMed ID: 17456681
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Pharmacology of vanilloid transient receptor potential cation channels.
    Vriens J; Appendino G; Nilius B
    Mol Pharmacol; 2009 Jun; 75(6):1262-79. PubMed ID: 19297520
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Antihyperalgesic effects of (R,E)-N-(2-hydroxy-2,3-dihydro-1H-inden-4-yl)-3-(2-(piperidin-1-yl)-4-(trifluoromethyl)phenyl)-acrylamide (AMG8562), a novel transient receptor potential vanilloid type 1 modulator that does not cause hyperthermia in rats.
    Lehto SG; Tamir R; Deng H; Klionsky L; Kuang R; Le A; Lee D; Louis JC; Magal E; Manning BH; Rubino J; Surapaneni S; Tamayo N; Wang T; Wang J; Wang J; Wang W; Youngblood B; Zhang M; Zhu D; Norman MH; Gavva NR
    J Pharmacol Exp Ther; 2008 Jul; 326(1):218-29. PubMed ID: 18420600
    [TBL] [Abstract][Full Text] [Related]  

  • 14. QX-314 produces long-lasting local anesthesia modulated by transient receptor potential vanilloid receptors in mice.
    Ries CR; Pillai R; Chung CC; Wang JT; MacLeod BA; Schwarz SK
    Anesthesiology; 2009 Jul; 111(1):122-6. PubMed ID: 19512885
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Inhibitory effect of cochinchinenin B on capsaicin-activated responses in rat dorsal root ganglion neurons.
    Wang ST; Chen S; Guo M; Liu XM
    Brain Res; 2008 Mar; 1201():34-40. PubMed ID: 18294619
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Transient receptor potential channels on sensory nerves.
    Eid SR; Cortright DN
    Handb Exp Pharmacol; 2009; (194):261-81. PubMed ID: 19655110
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Capsaicin (TRPV1 Agonist) therapy for pain relief: farewell or revival?
    Knotkova H; Pappagallo M; Szallasi A
    Clin J Pain; 2008 Feb; 24(2):142-54. PubMed ID: 18209521
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Hot receptors in the brain.
    Steenland HW; Ko SW; Wu LJ; Zhuo M
    Mol Pain; 2006 Nov; 2():34. PubMed ID: 17092351
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Design and synthesis of indole-based peptoids as potent noncompetitive antagonists of transient receptor potential vanilloid 1.
    Quintanar-Audelo M; Fernández-Carvajal A; Van Den Nest W; Carreño C; Ferrer-Montiel A; Albericio F
    J Med Chem; 2007 Nov; 50(24):6133-43. PubMed ID: 17985859
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Activation of the transient receptor potential vanilloid-1 (TRPV1) channel opens the gate for pain relief.
    Jancsó G; Dux M; Oszlács O; Sántha P
    Br J Pharmacol; 2008 Dec; 155(8):1139-41. PubMed ID: 18997813
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.