136 related articles for article (PubMed ID: 17533127)
21. Effects of mitemcinal (GM-611), an acid-resistant nonpeptide motilin receptor agonist, on the gastrointestinal contractile activity in conscious dogs.
Ozaki K; Yogo K; Sudo H; Onoma M; Kamei K; Akima M; Koga H; Itoh Z; Omura S; Takanashi H
Pharmacology; 2007; 79(4):223-35. PubMed ID: 17426410
[TBL] [Abstract][Full Text] [Related]
22. Desensitization and internalization of the human motilin receptor is independent of the C-terminal tail.
Mitselos A; Peeters TL; Depoortere I
Peptides; 2008 Jul; 29(7):1167-75. PubMed ID: 18420306
[TBL] [Abstract][Full Text] [Related]
23. Design and synthesis of motilin antagonists derived from the [1-4] fragment of porcine motilin.
Haramura M; Okamachi A; Tsuzuki K; Yogo K; Ikuta M; Kozono T; Takanashi H; Murayama E
J Med Chem; 2002 Jan; 45(3):670-5. PubMed ID: 11806718
[TBL] [Abstract][Full Text] [Related]
24. Motilin and erythromycin-A share a common binding site in the third transmembrane segment of the motilin receptor.
Xu L; Depoortere I; Vertongen P; Waelbroeck M; Robberecht P; Peeters TL
Biochem Pharmacol; 2005 Sep; 70(6):879-87. PubMed ID: 16076462
[TBL] [Abstract][Full Text] [Related]
25. Amino-acid templated assembly of sucrose-derived macrocycles.
Lewandowski B; Jarosz S
Org Lett; 2010 Jun; 12(11):2532-5. PubMed ID: 20441188
[TBL] [Abstract][Full Text] [Related]
26. Novel potent macrocyclic inhibitors of the hepatitis C virus NS3 protease: use of cyclopentane and cyclopentene P2-motifs.
Bäck M; Johansson PO; Wångsell F; Thorstensson F; Kvarnström I; Ayesa S; Wähling H; Pelcman M; Jansson K; Lindström S; Wallberg H; Classon B; Rydergård C; Vrang L; Hamelink E; Hallberg A; Rosenquist S; Samuelsson B
Bioorg Med Chem; 2007 Nov; 15(22):7184-202. PubMed ID: 17845856
[TBL] [Abstract][Full Text] [Related]
27. The identification of and rationale for drugs which act at the motilin receptor.
Westaway SM; Sanger GJ
Prog Med Chem; 2009; 48():31-80. PubMed ID: 21544957
[No Abstract] [Full Text] [Related]
28. Distribution and electrophysiological effects of motilin in Purkinje cells.
Chen H; Chen L; Wang JJ; Wei HJ; Yung WH
Neuroreport; 2007 Aug; 18(13):1345-9. PubMed ID: 17762710
[TBL] [Abstract][Full Text] [Related]
29. Characterization of the motilin receptor, a member of a new receptor family.
Miller LJ; Coulie B
Dig Liver Dis; 2000 Dec; 32 Suppl 3():S223-4. PubMed ID: 11245302
[No Abstract] [Full Text] [Related]
30. GSK962040: a small molecule, selective motilin receptor agonist, effective as a stimulant of human and rabbit gastrointestinal motility.
Sanger GJ; Westaway SM; Barnes AA; Macpherson DT; Muir AI; Jarvie EM; Bolton VN; Cellek S; Näslund E; Hellström PM; Borman RA; Unsworth WP; Matthews KL; Lee K
Neurogastroenterol Motil; 2009 Jun; 21(6):657-64, e30-1. PubMed ID: 19374732
[TBL] [Abstract][Full Text] [Related]
31. Molecular identification and characterization of the dog motilin receptor.
Ohshiro H; Nonaka M; Ichikawa K
Regul Pept; 2008 Feb; 146(1-3):80-7. PubMed ID: 17870192
[TBL] [Abstract][Full Text] [Related]
32. Identification of genes for the ghrelin and motilin receptors and a novel related gene in fish, and stimulation of intestinal motility in zebrafish (Danio rerio) by ghrelin and motilin.
Olsson C; Holbrook JD; Bompadre G; Jönsson E; Hoyle CH; Sanger GJ; Holmgren S; Andrews PL
Gen Comp Endocrinol; 2008 Jan; 155(1):217-26. PubMed ID: 17582410
[TBL] [Abstract][Full Text] [Related]
33. Protein and cellular engineering with unnatural amino acids.
Liao J
Biotechnol Prog; 2007; 23(1):28-31. PubMed ID: 17269666
[TBL] [Abstract][Full Text] [Related]
34. Macrocycles are great cycles: applications, opportunities, and challenges of synthetic macrocycles in drug discovery.
Marsault E; Peterson ML
J Med Chem; 2011 Apr; 54(7):1961-2004. PubMed ID: 21381769
[No Abstract] [Full Text] [Related]
35. Discovery of N-(3-fluorophenyl)-1-[(4-([(3S)-3-methyl-1-piperazinyl]methyl)phenyl)acetyl]-4-piperidinamine (GSK962040), the first small molecule motilin receptor agonist clinical candidate.
Westaway SM; Brown SL; Fell SC; Johnson CN; MacPherson DT; Mitchell DJ; Myatt JW; Stanway SJ; Seal JT; Stemp G; Thompson M; Lawless K; McKay F; Muir AI; Barford JM; Cluff C; Mahmood SR; Matthews KL; Mohamed S; Smith B; Stevens AJ; Bolton VJ; Jarvie EM; Sanger GJ
J Med Chem; 2009 Feb; 52(4):1180-9. PubMed ID: 19191554
[TBL] [Abstract][Full Text] [Related]
36. Identification of the motilide pharmacophores using quantitative structure activity relationships.
Khiat A; Boulanger Y
J Pept Res; 1998 Oct; 52(4):321-8. PubMed ID: 9832311
[TBL] [Abstract][Full Text] [Related]
37. Amino acid derived macrocycles--an area driven by synthesis or application?
Gibson SE; Lecci C
Angew Chem Int Ed Engl; 2006 Feb; 45(9):1364-77. PubMed ID: 16444788
[TBL] [Abstract][Full Text] [Related]
38. Conformational analysis of N,N-disubstituted-1,4-diazepane orexin receptor antagonists and implications for receptor binding.
Cox CD; McGaughey GB; Bogusky MJ; Whitman DB; Ball RG; Winrow CJ; Renger JJ; Coleman PJ
Bioorg Med Chem Lett; 2009 Jun; 19(11):2997-3001. PubMed ID: 19406641
[TBL] [Abstract][Full Text] [Related]
39. Ribosomal synthesis of backbone-macrocyclic peptides containing γ-amino acids.
Ohshiro Y; Nakajima E; Goto Y; Fuse S; Takahashi T; Doi T; Suga H
Chembiochem; 2011 May; 12(8):1183-7. PubMed ID: 21506233
[No Abstract] [Full Text] [Related]
40. Rapid generation of macrocycles with natural-product-like side chains by multiple multicomponent macrocyclizations (MiBs).
Rivera DG; Vercillo OE; Wessjohann LA
Org Biomol Chem; 2008 May; 6(10):1787-95. PubMed ID: 18452014
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
