756 related articles for article (PubMed ID: 17570124)
1. Contribution of specific binding to the central benzodiazepine site to the brain concentrations of two novel benzodiazepine site ligands.
Pike A; Cook SM; Watt AP; Scott-Stevens P; Rosahl TW; McKernan RM; Pym LJ; Guiblin A; Moyes C; Sohal B; Atack JR
Biopharm Drug Dispos; 2007 Sep; 28(6):275-82. PubMed ID: 17570124
[TBL] [Abstract][Full Text] [Related]
2. Comparison of in vivo and ex vivo [3H]flumazenil binding assays to determine occupancy at the benzodiazepine binding site of rat brain GABAA receptors.
Li J; Fish RL; Cook SM; Tattersall FD; Atack JR
Neuropharmacology; 2006 Jul; 51(1):168-72. PubMed ID: 16697018
[TBL] [Abstract][Full Text] [Related]
3. Down-regulation of benzodiazepine binding to alpha 5 subunit-containing gamma-aminobutyric Acid(A) receptors in tolerant rat brain indicates particular involvement of the hippocampal CA1 region.
Li M; Szabo A; Rosenberg HC
J Pharmacol Exp Ther; 2000 Nov; 295(2):689-96. PubMed ID: 11046107
[TBL] [Abstract][Full Text] [Related]
4. Native gamma-aminobutyric acid type A receptors from rat hippocampus, containing both alpha 1 and alpha 5 subunits, exhibit a single benzodiazepine binding site with alpha 5 pharmacological properties.
Araujo F; Ruano D; Vitorica J
J Pharmacol Exp Ther; 1999 Sep; 290(3):989-97. PubMed ID: 10454469
[TBL] [Abstract][Full Text] [Related]
5. Differential effects of ammonia on the benzodiazepine modulatory site on the GABA-A receptor complex of human brain.
Ahboucha S; Araqi F; Layrargues GP; Butterworth RF
Neurochem Int; 2005 Jul; 47(1-2):58-63. PubMed ID: 15913842
[TBL] [Abstract][Full Text] [Related]
6. Rodent pharmacokinetics and receptor occupancy of the GABAA receptor subtype selective benzodiazepine site ligand L-838417.
Scott-Stevens P; Atack JR; Sohal B; Worboys P
Biopharm Drug Dispos; 2005 Jan; 26(1):13-20. PubMed ID: 15578749
[TBL] [Abstract][Full Text] [Related]
7. In vivo labelling of alpha5 subunit-containing GABA(A) receptors using the selective radioligand [(3)H]L-655,708.
Atack JR; Alder L; Cook SM; Smith AJ; McKernan RM
Neuropharmacology; 2005 Aug; 49(2):220-9. PubMed ID: 15996568
[TBL] [Abstract][Full Text] [Related]
8. Selective labelling of diazepam-insensitive GABAA receptors in vivo using [3H]Ro 15-4513.
Pym LJ; Cook SM; Rosahl T; McKernan RM; Atack JR
Br J Pharmacol; 2005 Nov; 146(6):817-25. PubMed ID: 16184188
[TBL] [Abstract][Full Text] [Related]
9. In vivo saturation binding of GABA-A receptor ligands to estimate receptor occupancy using liquid chromatography/tandem mass spectrometry.
Hopkins SC; Brian Nofsinger J; Allen MS; Koch P; Varney MA
Biopharm Drug Dispos; 2009 Jan; 30(1):9-20. PubMed ID: 19152227
[TBL] [Abstract][Full Text] [Related]
10. [11C-Ro15-1788 and 11C-flunitrazepam, two coordinates for the study by positron emission tomography of benzodiazepine binding sites].
Mazière M; Prenant C; Sastre J; Crouzel M; Comar D; Hantraye P; Kaïsima M; Guibert B; Naquet R
C R Seances Acad Sci III; 1983; 296(18):871-6. PubMed ID: 6136317
[TBL] [Abstract][Full Text] [Related]
11. Sedative but not anxiolytic properties of benzodiazepines are mediated by the GABA(A) receptor alpha1 subtype.
McKernan RM; Rosahl TW; Reynolds DS; Sur C; Wafford KA; Atack JR; Farrar S; Myers J; Cook G; Ferris P; Garrett L; Bristow L; Marshall G; Macaulay A; Brown N; Howell O; Moore KW; Carling RW; Street LJ; Castro JL; Ragan CI; Dawson GR; Whiting PJ
Nat Neurosci; 2000 Jun; 3(6):587-92. PubMed ID: 10816315
[TBL] [Abstract][Full Text] [Related]
12. Postnatal development and kinetics of [3H]gaboxadol binding in rat brain: in vitro homogenate binding and quantitative autoradiography.
Friemel A; Ebert B; Hutson PH; Brust P; Nieber K; Deuther-Conrad W
Brain Res; 2007 Sep; 1170():39-47. PubMed ID: 17692833
[TBL] [Abstract][Full Text] [Related]
13. Acute pentylenetetrazol injection reduces rat GABAA receptor mRNA levels and GABA stimulation of benzodiazepine binding with No effect on benzodiazepine binding site density.
Walsh LA; Li M; Zhao TJ; Chiu TH; Rosenberg HC
J Pharmacol Exp Ther; 1999 Jun; 289(3):1626-33. PubMed ID: 10336561
[TBL] [Abstract][Full Text] [Related]
14. The plasma-occupancy relationship of the novel GABAA receptor benzodiazepine site ligand, alpha5IA, is similar in rats and primates.
Atack JR; Eng WS; Gibson RE; Ryan C; Francis B; Sohal B; Dawson GR; Hargreaves RJ; Burns HD
Br J Pharmacol; 2009 Jul; 157(5):796-803. PubMed ID: 19422390
[TBL] [Abstract][Full Text] [Related]
15. Receptor subtype-dependent positive and negative modulation of GABA(A) receptor function by niflumic acid, a nonsteroidal anti-inflammatory drug.
Sinkkonen ST; Mansikkamäki S; Möykkynen T; Lüddens H; Uusi-Oukari M; Korpi ER
Mol Pharmacol; 2003 Sep; 64(3):753-63. PubMed ID: 12920213
[TBL] [Abstract][Full Text] [Related]
16. N,N'-dicyclohexylsulfamide and N,N'-diphenethylsulfamide are anticonvulsant sulfamides with affinity for the benzodiazepine binding site of the GABA(A) receptor and anxiolytic activity in mice.
Wasowski C; Gavernet L; Barrios IA; Villalba ML; Pastore V; Samaja G; Enrique A; Bruno-Blanch LE; Marder M
Biochem Pharmacol; 2012 Jan; 83(2):253-9. PubMed ID: 22056620
[TBL] [Abstract][Full Text] [Related]
17. Modulation of ligand binding to components of the GABAA receptor complex by ammonia: implications for the pathogenesis of hyperammonemic syndromes.
Ha JH; Basile AS
Brain Res; 1996 May; 720(1-2):35-44. PubMed ID: 8782894
[TBL] [Abstract][Full Text] [Related]
18. Effect of ergot alkaloids on 3H-flunitrazepam binding to mouse brain GABAA receptors.
Tvrdeić A; Pericić D
Coll Antropol; 2003; 27 Suppl 1():175-82. PubMed ID: 12955907
[TBL] [Abstract][Full Text] [Related]
19. Differential contribution of GABA(A) receptor subtypes to the anticonvulsant efficacy of benzodiazepine site ligands.
Fradley RL; Guscott MR; Bull S; Hallett DJ; Goodacre SC; Wafford KA; Garrett EM; Newman RJ; O'Meara GF; Whiting PJ; Rosahl TW; Dawson GR; Reynolds DS; Atack JR
J Psychopharmacol; 2007 Jun; 21(4):384-91. PubMed ID: 17092983
[TBL] [Abstract][Full Text] [Related]
20. CNS 7056: a novel ultra-short-acting Benzodiazepine.
Kilpatrick GJ; McIntyre MS; Cox RF; Stafford JA; Pacofsky GJ; Lovell GG; Wiard RP; Feldman PL; Collins H; Waszczak BL; Tilbrook GS
Anesthesiology; 2007 Jul; 107(1):60-6. PubMed ID: 17585216
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]