201 related articles for article (PubMed ID: 17582659)
1. Synthesis and cannabinoid activity of 1-substituted-indole-3-oxadiazole derivatives: novel agonists for the CB1 receptor.
Moloney GP; Angus JA; Robertson AD; Stoermer MJ; Robinson M; Wright CE; McRae K; Christopoulos A
Eur J Med Chem; 2008 Mar; 43(3):513-39. PubMed ID: 17582659
[TBL] [Abstract][Full Text] [Related]
2. Low brain penetrant CB1 receptor agonists for the treatment of neuropathic pain.
Adam JM; Clark JK; Davies K; Everett K; Fields R; Francis S; Jeremiah F; Kiyoi T; Maidment M; Morrison A; Ratcliffe P; Prosser A; Schulz J; Wishart G; Baker J; Boyce S; Campbell R; Cottney JE; Deehan M; Martin I
Bioorg Med Chem Lett; 2012 Apr; 22(8):2932-7. PubMed ID: 22421020
[TBL] [Abstract][Full Text] [Related]
3. 1-Pentyl-3-phenylacetylindoles, a new class of cannabimimetic indoles.
Huffman JW; Szklennik PV; Almond A; Bushell K; Selley DE; He H; Cassidy MP; Wiley JL; Martin BR
Bioorg Med Chem Lett; 2005 Sep; 15(18):4110-3. PubMed ID: 16005223
[TBL] [Abstract][Full Text] [Related]
4. Indol-3-ylcycloalkyl ketones: effects of N1 substituted indole side chain variations on CB(2) cannabinoid receptor activity.
Frost JM; Dart MJ; Tietje KR; Garrison TR; Grayson GK; Daza AV; El-Kouhen OF; Yao BB; Hsieh GC; Pai M; Zhu CZ; Chandran P; Meyer MD
J Med Chem; 2010 Jan; 53(1):295-315. PubMed ID: 19921781
[TBL] [Abstract][Full Text] [Related]
5. Diarylimidazolyl oxadiazole and thiadiazole derivatives as cannabinoid CB1 receptor antagonists.
Kim JY; Seo HJ; Lee SH; Jung ME; Ahn K; Kim J; Lee J
Bioorg Med Chem Lett; 2009 Jan; 19(1):142-5. PubMed ID: 19022666
[TBL] [Abstract][Full Text] [Related]
6. Oxadiazole-diarylpyrazole 4-carboxamides as cannabinoid CB1 receptor ligands.
Lee SH; Seo HJ; Kim MJ; Kang SY; Song KS; Lee SH; Jung ME; Kim J; Lee J
Bioorg Med Chem Lett; 2009 Apr; 19(7):1899-902. PubMed ID: 19269817
[TBL] [Abstract][Full Text] [Related]
7. Design, synthesis, and structure-activity relationships of indole-3-heterocycles as agonists of the CB1 receptor.
Morrison AJ; Adam JM; Baker JA; Campbell RA; Clark JK; Cottney JE; Deehan M; Easson AM; Fields R; Francis S; Jeremiah F; Keddie N; Kiyoi T; McArthur DR; Meyer K; Ratcliffe PD; Schulz J; Wishart G; Yoshiizumi K
Bioorg Med Chem Lett; 2011 Jan; 21(1):506-9. PubMed ID: 21075630
[TBL] [Abstract][Full Text] [Related]
8. Design, synthesis, and structure-activity relationship study of conformationally constrained analogs of indole-3-carboxamides as novel CB1 cannabinoid receptor agonists.
Kiyoi T; York M; Francis S; Edwards D; Walker G; Houghton AK; Cottney JE; Baker J; Adam JM
Bioorg Med Chem Lett; 2010 Aug; 20(16):4918-21. PubMed ID: 20634067
[TBL] [Abstract][Full Text] [Related]
9. Biarylpyrazolyl oxadiazole as potent, selective, orally bioavailable cannabinoid-1 receptor antagonists for the treatment of obesity.
Lee SH; Seo HJ; Lee SH; Jung ME; Park JH; Park HJ; Yoo J; Yun H; Na J; Kang SY; Song KS; Kim MA; Chang CH; Kim J; Lee J
J Med Chem; 2008 Nov; 51(22):7216-33. PubMed ID: 18954042
[TBL] [Abstract][Full Text] [Related]
10. The discovery of novel indole-2-carboxamides as cannabinoid CB(1) receptor antagonists.
Cowley PM; Baker J; Barn DR; Buchanan KI; Carlyle I; Clark JK; Clarkson TR; Deehan M; Edwards D; Goodwin RR; Jaap D; Kiyoi Y; Mort C; Palin R; Prosser A; Walker G; Ward N; Wishart G; Young T
Bioorg Med Chem Lett; 2011 Jan; 21(1):497-501. PubMed ID: 21075628
[TBL] [Abstract][Full Text] [Related]
11. Potent cannabinergic indole analogues as radioiodinatable brain imaging agents for the CB1 cannabinoid receptor.
Deng H; Gifford AN; Zvonok AM; Cui G; Li X; Fan P; Deschamps JR; Flippen-Anderson JL; Gatley SJ; Makriyannis A
J Med Chem; 2005 Oct; 48(20):6386-92. PubMed ID: 16190764
[TBL] [Abstract][Full Text] [Related]
12. Design and synthesis of indole-based peptoids as potent noncompetitive antagonists of transient receptor potential vanilloid 1.
Quintanar-Audelo M; Fernández-Carvajal A; Van Den Nest W; Carreño C; Ferrer-Montiel A; Albericio F
J Med Chem; 2007 Nov; 50(24):6133-43. PubMed ID: 17985859
[TBL] [Abstract][Full Text] [Related]
13. Design, synthesis and pro-apoptotic antitumour properties of indole-based 3,5-disubstituted oxadiazoles.
Ziedan NI; Stefanelli F; Fogli S; Westwell AD
Eur J Med Chem; 2010 Oct; 45(10):4523-30. PubMed ID: 20705365
[TBL] [Abstract][Full Text] [Related]
14. Indol-3-yl-tetramethylcyclopropyl ketones: effects of indole ring substitution on CB2 cannabinoid receptor activity.
Frost JM; Dart MJ; Tietje KR; Garrison TR; Grayson GK; Daza AV; El-Kouhen OF; Miller LN; Li L; Yao BB; Hsieh GC; Pai M; Zhu CZ; Chandran P; Meyer MD
J Med Chem; 2008 Mar; 51(6):1904-12. PubMed ID: 18311894
[TBL] [Abstract][Full Text] [Related]
15. Synthesis of novel 1,3,4-oxadiazole derivatives and their biological properties.
Husain A; Ajmal M
Acta Pharm; 2009 Jun; 59(2):223-33. PubMed ID: 19564146
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and pharmacological evaluation of coumarin derivatives as cannabinoid receptor antagonists and inverse agonists.
Behrenswerth A; Volz N; Toräng J; Hinz S; Bräse S; Müller CE
Bioorg Med Chem; 2009 Apr; 17(7):2842-51. PubMed ID: 19278853
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and biological evaluation of new 3-substituted indole derivatives as potential anti-inflammatory and analgesic agents.
Radwan MA; Ragab EA; Sabry NM; El-Shenawy SM
Bioorg Med Chem; 2007 Jun; 15(11):3832-41. PubMed ID: 17395469
[TBL] [Abstract][Full Text] [Related]
18. 2-[3-(4-chloro/ethyl phenyl)propan-3-one]-5-(substituted phenyl)-1,3,4-oxadiazoles: synthesis and biological evaluation.
Husain A; Sarafroz M; Ahuja P
Acta Pol Pharm; 2008; 65(5):527-34. PubMed ID: 19051598
[TBL] [Abstract][Full Text] [Related]
19. Aroylpropionic acid based 2,5-disubstituted-1,3,4-oxadiazoles: synthesis and their anti-inflammatory and analgesic activities.
Akhter M; Husain A; Azad B; Ajmal M
Eur J Med Chem; 2009 Jun; 44(6):2372-8. PubMed ID: 18977556
[TBL] [Abstract][Full Text] [Related]
20. An efficient synthesis and biological study of novel indolyl-1,3,4-oxadiazoles as potent anticancer agents.
Kumar D; Sundaree S; Johnson EO; Shah K
Bioorg Med Chem Lett; 2009 Aug; 19(15):4492-4. PubMed ID: 19559607
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
