136 related articles for article (PubMed ID: 17644772)
1. A fluorescence lifetime based binding assay to characterize kinase inhibitors.
Lebakken CS; Hee Chol Kang ; Vogel KW
J Biomol Screen; 2007 Sep; 12(6):828-41. PubMed ID: 17644772
[TBL] [Abstract][Full Text] [Related]
2. Development and applications of a broad-coverage, TR-FRET-based kinase binding assay platform.
Lebakken CS; Riddle SM; Singh U; Frazee WJ; Eliason HC; Gao Y; Reichling LJ; Marks BD; Vogel KW
J Biomol Screen; 2009 Sep; 14(8):924-35. PubMed ID: 19564447
[TBL] [Abstract][Full Text] [Related]
3. A high-throughput, nonisotopic, competitive binding assay for kinases using nonselective inhibitor probes (ED-NSIP).
Vainshtein I; Silveria S; Kaul P; Rouhani R; Eglen RM; Wang J
J Biomol Screen; 2002 Dec; 7(6):507-14. PubMed ID: 14599348
[TBL] [Abstract][Full Text] [Related]
4. Development of a fluorescent-tagged kinase assay system for the detection and characterization of allosteric kinase inhibitors.
Simard JR; Getlik M; Grütter C; Pawar V; Wulfert S; Rabiller M; Rauh D
J Am Chem Soc; 2009 Sep; 131(37):13286-96. PubMed ID: 19572644
[TBL] [Abstract][Full Text] [Related]
5. Staurosporine-based binding assay for testing the affinity of compounds to protein kinases.
Iyer GH; Taslimi P; Pazhanisamy S
Anal Biochem; 2008 Feb; 373(2):197-206. PubMed ID: 18047825
[TBL] [Abstract][Full Text] [Related]
6. Three mechanistically distinct kinase assays compared: Measurement of intrinsic ATPase activity identified the most comprehensive set of ITK inhibitors.
Kashem MA; Nelson RM; Yingling JD; Pullen SS; Prokopowicz AS; Jones JW; Wolak JP; Rogers GR; Morelock MM; Snow RJ; Homon CA; Jakes S
J Biomol Screen; 2007 Feb; 12(1):70-83. PubMed ID: 17166826
[TBL] [Abstract][Full Text] [Related]
7. Fluorescence labels in kinases: a high-throughput kinase binding assay for the identification of DFG-out binding ligands.
Simard JR; Rauh D
Methods Mol Biol; 2012; 800():95-117. PubMed ID: 21964785
[TBL] [Abstract][Full Text] [Related]
8. Multiplexing terbium- and europium-based TR-FRET readouts to increase kinase assay capacity.
Horton RA; Vogel KW
J Biomol Screen; 2010 Sep; 15(8):1008-15. PubMed ID: 20460248
[TBL] [Abstract][Full Text] [Related]
9. Duplexed, bead-based competitive assay for inhibitors of protein kinases.
Simons PC; Young SM; Gibaja V; Lee WC; Josiah S; Edwards BS; Sklar LA
Cytometry A; 2007 Jul; 71(7):451-9. PubMed ID: 17542028
[TBL] [Abstract][Full Text] [Related]
10. Detection of allosteric kinase inhibitors by displacement of active site probes.
Lebakken CS; Reichling LJ; Ellefson JM; Riddle SM
J Biomol Screen; 2012 Jul; 17(6):813-21. PubMed ID: 22453235
[TBL] [Abstract][Full Text] [Related]
11. A general technique to rank protein-ligand binding affinities and determine allosteric versus direct binding site competition in compound mixtures.
Annis DA; Nazef N; Chuang CC; Scott MP; Nash HM
J Am Chem Soc; 2004 Dec; 126(47):15495-503. PubMed ID: 15563178
[TBL] [Abstract][Full Text] [Related]
12. A fluorescence resonance energy transfer-based binding assay for characterizing kinase inhibitors: important role for C-terminal biotin tagging of the kinase.
Kwan J; Ling A; Papp E; Shaw D; Bradshaw JM
Anal Biochem; 2009 Dec; 395(2):256-62. PubMed ID: 19716360
[TBL] [Abstract][Full Text] [Related]
13. High-affinity bisubstrate probe for fluorescence anisotropy binding/displacement assays with protein kinases PKA and ROCK.
Vaasa A; Viil I; Enkvist E; Viht K; Raidaru G; Lavogina D; Uri A
Anal Biochem; 2009 Feb; 385(1):85-93. PubMed ID: 19017524
[TBL] [Abstract][Full Text] [Related]
14. Development of a novel fluorescent probe for fluorescence correlation spectroscopic detection of kinase inhibitors.
Kawaguchi M; Terai T; Utata R; Kato M; Tsuganezawa K; Tanaka A; Kojima H; Okabe T; Nagano T
Bioorg Med Chem Lett; 2008 Jul; 18(13):3752-5. PubMed ID: 18524589
[TBL] [Abstract][Full Text] [Related]
15. Screening kinase inhibitors with a microarray-based fluorescent and resonance light scattering assay.
Li T; Liu D; Wang Z
Anal Chem; 2010 Apr; 82(7):3067-72. PubMed ID: 20201592
[TBL] [Abstract][Full Text] [Related]
16. Development of a Transcreener kinase assay for protein kinase A and demonstration of concordance of data with a filter-binding assay format.
Huss KL; Blonigen PE; Campbell RM
J Biomol Screen; 2007 Jun; 12(4):578-84. PubMed ID: 17409274
[TBL] [Abstract][Full Text] [Related]
17. Functional characterization of peanut serine/threonine/tyrosine protein kinase: molecular docking and inhibition kinetics with tyrosine kinase inhibitors.
Rudrabhatla P; Rajasekharan R
Biochemistry; 2004 Sep; 43(38):12123-32. PubMed ID: 15379551
[TBL] [Abstract][Full Text] [Related]
18. Fluorescence polarization competition immunoassay for tyrosine kinases.
Seethala R
Methods; 2000 Sep; 22(1):61-70. PubMed ID: 11020319
[TBL] [Abstract][Full Text] [Related]
19. Utilization of fluorescence polarization and time resolved fluorescence resonance energy transfer assay formats for SAR studies: Src kinase as a model system.
Newman M; Josiah S
J Biomol Screen; 2004 Sep; 9(6):525-32. PubMed ID: 15452339
[TBL] [Abstract][Full Text] [Related]
20. A liquid chromatography/mass spectrometry-based method for the selection of ATP competitive kinase inhibitors.
Khandekar SS; Feng B; Yi T; Chen S; Laping N; Bramson N
J Biomol Screen; 2005 Aug; 10(5):447-55. PubMed ID: 16093554
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]