BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

229 related articles for article (PubMed ID: 18262419)

  • 1. Individual stereoisomers of phosphinic dipeptide inhibitor of leucine aminopeptidase.
    Mucha A; Lämmerhofer M; Lindner W; Pawełczak M; Kafarski P
    Bioorg Med Chem Lett; 2008 Mar; 18(5):1550-4. PubMed ID: 18262419
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Stereoselective separations of chiral phosphinic acid pseudodipeptides by CEC using silica monoliths modified with an anion-exchange-type chiral selector.
    Preinerstorfer B; Lubda D; Mucha A; Kafarski P; Lindner W; Lämmerhofer M
    Electrophoresis; 2006 Nov; 27(21):4312-20. PubMed ID: 17006883
    [TBL] [Abstract][Full Text] [Related]  

  • 3. A synthetic method for diversification of the P1' substituent in phosphinic dipeptides as a tool for exploration of the specificity of the S1' binding pockets of leucine aminopeptidases.
    Vassiliou S; Xeilari M; Yiotakis A; Grembecka J; Pawełczak M; Kafarski P; Mucha A
    Bioorg Med Chem; 2007 May; 15(9):3187-200. PubMed ID: 17337192
    [TBL] [Abstract][Full Text] [Related]  

  • 4. The most potent organophosphorus inhibitors of leucine aminopeptidase. Structure-based design, chemistry, and activity.
    Grembecka J; Mucha A; Cierpicki T; Kafarski P
    J Med Chem; 2003 Jun; 46(13):2641-55. PubMed ID: 12801228
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Identification of phosphinate dipeptide analog inhibitors directed against the Plasmodium falciparum M17 leucine aminopeptidase as lead antimalarial compounds.
    Skinner-Adams TS; Lowther J; Teuscher F; Stack CM; Grembecka J; Mucha A; Kafarski P; Trenholme KR; Dalton JP; Gardiner DL
    J Med Chem; 2007 Nov; 50(24):6024-31. PubMed ID: 17960925
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Design, synthesis, and metal binding of novel Pseudo- oligopeptides containing two phosphinic acid groups.
    Ye Y; Liu M; Kao JL; Marshall GR
    Biopolymers; 2008 Jan; 89(1):72-85. PubMed ID: 17910046
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Efficient synthesis of Fmoc-protected phosphinic pseudodipeptides: Building blocks for the synthesis of matrix metalloproteinase inhibitors.
    Bhowmick M; Sappidi RR; Fields GB; Lepore SD
    Biopolymers; 2011; 96(1):1-3. PubMed ID: 20225219
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis of α-carboxyphosphinopeptides derived from norleucine.
    Pícha J; Buděšínský M; Fiedler P; Sanda M; Jiráček J
    Amino Acids; 2010 Nov; 39(5):1265-80. PubMed ID: 20349321
    [TBL] [Abstract][Full Text] [Related]  

  • 9. [Affinity labeling of leucine aminopeptidase with new substrate analog inhibitors].
    Fittkau S; Schunck WH; Mootsi S
    Acta Biol Med Ger; 1976; 35(3-4):365-78. PubMed ID: 970045
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Conformational and solvation studies via computer simulation of the novel large scale diastereoselectively synthesized phosphinic MMP inhibitor RXP03 diluted in selected solvents.
    Matziari M; Dellis D; Dive V; Yiotakis A; Samios J
    J Phys Chem B; 2010 Jan; 114(1):421-8. PubMed ID: 20014753
    [TBL] [Abstract][Full Text] [Related]  

  • 11. A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases.
    Węglarz-Tomczak E; Berlicki Ł; Pawełczak M; Nocek B; Joachimiak A; Mucha A
    Eur J Med Chem; 2016 Jul; 117():187-96. PubMed ID: 27100031
    [TBL] [Abstract][Full Text] [Related]  

  • 12. A phosphinic acid dipeptide analogue to stabilize peptide drugs during their intranasal absorption.
    Hussain MA; Lim MS; Raghavan KS; Rogers NJ; Hidalgo R; Kettner CA
    Pharm Res; 1992 May; 9(5):626-8. PubMed ID: 1608893
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Phosphorus amino acid analogues as inhibitors of leucine aminopeptidase.
    Giannousis PP; Bartlett PA
    J Med Chem; 1987 Sep; 30(9):1603-9. PubMed ID: 3625708
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Diastereoselective synthesis of alpha,beta'-disubstituted aminomethyl(2-carboxyethyl)phosphinates as phosphinyl dipeptide isosteres.
    Yamagishi T; Ichikawa H; Haruki T; Yokomatsu T
    Org Lett; 2008 Oct; 10(19):4347-50. PubMed ID: 18781768
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Unusual activity pattern of leucine aminopeptidase inhibitors based on phosphorus containing derivatives of methionine and norleucine.
    Pícha J; Liboska R; Buděšínský M; Jiráček J; Pawełczak M; Mucha A
    J Enzyme Inhib Med Chem; 2011 Apr; 26(2):155-61. PubMed ID: 20578976
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Phosphinate, sulfonate, and sulfonamidate dipeptides as potential inhibitors of Escherichia coli aminopeptidase N.
    Yang KW; Golich FC; Sigdel TK; Crowder MW
    Bioorg Med Chem Lett; 2005 Dec; 15(23):5150-3. PubMed ID: 16168644
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Stereoselective synthesis of 1-aminoalkanephosphonic acids with two chiral centers and their activity towards leucine aminopeptidase.
    Drag M; Pawelczak M; Kafarski P
    Chirality; 2003; 15 Suppl():S104-7. PubMed ID: 12884381
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis and structure-activity relationships of bestatin analogues, inhibitors of aminopeptidase B.
    Nishizawa R; Saino T; Takita T; Suda H; Aoyagi T
    J Med Chem; 1977 Apr; 20(4):510-5. PubMed ID: 850237
    [TBL] [Abstract][Full Text] [Related]  

  • 19. A novel method for the separation of bis(alpha-hydroxyalkyl)phosphinic acid diastereoisomers via formation of novel cyclic phosphinic acids.
    Kaboudin B; Haghighat H; Yokomatsu T
    J Org Chem; 2006 Aug; 71(17):6604-6. PubMed ID: 16901151
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis and modifications of phosphinic dipeptide analogues.
    Mucha A
    Molecules; 2012 Nov; 17(11):13530-68. PubMed ID: 23154272
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 12.