152 related articles for article (PubMed ID: 1826744)
1. Kynurenic acid derivatives. Structure-activity relationships for excitatory amino acid antagonism and identification of potent and selective antagonists at the glycine site on the N-methyl-D-aspartate receptor.
Leeson PD; Baker R; Carling RW; Curtis NR; Moore KW; Williams BJ; Foster AC; Donald AE; Kemp JA; Marshall GR
J Med Chem; 1991 Apr; 34(4):1243-52. PubMed ID: 1826744
[TBL] [Abstract][Full Text] [Related]
2. Kynurenic acid analogues with improved affinity and selectivity for the glycine site on the N-methyl-D-aspartate receptor from rat brain.
Foster AC; Kemp JA; Leeson PD; Grimwood S; Donald AE; Marshall GR; Priestley T; Smith JD; Carling RW
Mol Pharmacol; 1992 May; 41(5):914-22. PubMed ID: 1375317
[TBL] [Abstract][Full Text] [Related]
3. Thiokynurenates: a new group of antagonists of the glycine modulatory site of the NMDA receptor.
Moroni F; Alesiani M; Galli A; Mori F; Pecorari R; Carlà V; Cherici G; Pellicciari R
Eur J Pharmacol; 1991 Jun; 199(2):227-32. PubMed ID: 1720099
[TBL] [Abstract][Full Text] [Related]
4. Structure-activity relationships of alkyl- and alkoxy-substituted 1,4-dihydroquinoxaline-2,3-diones: potent and systemically active antagonists for the glycine site of the NMDA receptor.
Cai SX; Kher SM; Zhou ZL; Ilyin V; Espitia SA; Tran M; Hawkinson JE; Woodward RM; Weber E; Keana JF
J Med Chem; 1997 Feb; 40(5):730-8. PubMed ID: 9057859
[TBL] [Abstract][Full Text] [Related]
5. Novel class of amino acid antagonists at non-N-methyl-D-aspartic acid excitatory amino acid receptors. Synthesis, in vitro and in vivo pharmacology, and neuroprotection.
Krogsgaard-Larsen P; Ferkany JW; Nielsen EO; Madsen U; Ebert B; Johansen JS; Diemer NH; Bruhn T; Beattie DT; Curtis DR
J Med Chem; 1991 Jan; 34(1):123-30. PubMed ID: 1825114
[TBL] [Abstract][Full Text] [Related]
6. 3-Nitro-3,4-dihydro-2(1H)-quinolones. Excitatory amino acid antagonists acting at glycine-site NMDA and (RS)-alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptors.
Carling RW; Leeson PD; Moore KW; Smith JD; Moyes CR; Mawer IM; Thomas S; Chan T; Baker R; Foster AC
J Med Chem; 1993 Oct; 36(22):3397-408. PubMed ID: 8230130
[TBL] [Abstract][Full Text] [Related]
7. Selectivity of quinoxalines and kynurenines as antagonists of the glycine site on N-methyl-D-aspartate receptors.
Kleckner NW; Dingledine R
Mol Pharmacol; 1989 Sep; 36(3):430-6. PubMed ID: 2550776
[TBL] [Abstract][Full Text] [Related]
8. Analogs of 3-hydroxy-1H-1-benzazepine-2,5-dione: structure-activity relationship at N-methyl-D-aspartate receptor glycine sites.
Guzikowski AP; Cai SX; Espitia SA; Hawkinson JE; Huettner JE; Nogales DF; Tran M; Woodward RM; Weber E; Keana JF
J Med Chem; 1996 Nov; 39(23):4643-53. PubMed ID: 8917653
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and structure-activity relationships of 1,2,3,4-tetrahydroquinoline-2,3,4-trione 3-oximes: novel and highly potent antagonists for NMDA receptor glycine site.
Cai SX; Zhou ZL; Huang JC; Whittemore ER; Egbuwoku ZO; Lü Y; Hawkinson JE; Woodward RM; Weber E; Keana JF
J Med Chem; 1996 Aug; 39(17):3248-55. PubMed ID: 8765507
[TBL] [Abstract][Full Text] [Related]
10. Structure-activity analysis of binding kinetics for NMDA receptor competitive antagonists: the influence of conformational restriction.
Benveniste M; Mayer ML
Br J Pharmacol; 1991 Sep; 104(1):207-21. PubMed ID: 1686203
[TBL] [Abstract][Full Text] [Related]
11. 5,7-Dichlorokynurenic acid, a potent and selective competitive antagonist of the glycine site on NMDA receptors.
McNamara D; Smith EC; Calligaro DO; O'Malley PJ; McQuaid LA; Dingledine R
Neurosci Lett; 1990 Nov; 120(1):17-20. PubMed ID: 2149877
[TBL] [Abstract][Full Text] [Related]
12. Support for radiolabeling of a glycine recognition domain on the N-methyl-D-aspartate receptor ionophore complex by 5,7-[3H]dichlorokynurenate in rat brain.
Yoneda Y; Suzuki T; Ogita K; Han D
J Neurochem; 1993 Feb; 60(2):634-45. PubMed ID: 8419541
[TBL] [Abstract][Full Text] [Related]
13. 4-Amido-2-carboxytetrahydroquinolines. Structure-activity relationships for antagonism at the glycine site of the NMDA receptor.
Leeson PD; Carling RW; Moore KW; Moseley AM; Smith JD; Stevenson G; Chan T; Baker R; Foster AC; Grimwood S
J Med Chem; 1992 May; 35(11):1954-68. PubMed ID: 1534584
[TBL] [Abstract][Full Text] [Related]
14. Synthesis of 1,4,7,8,9,10-hexahydro-9-methyl-6-nitropyrido[3,4-f]- quinoxaline-2,3-dione and related quinoxalinediones: characterization of alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (and N-methyl-D-aspartate) receptor and anticonvulsant activity.
Bigge CF; Malone TC; Boxer PA; Nelson CB; Ortwine DF; Schelkun RM; Retz DM; Lescosky LJ; Borosky SA; Vartanian MG
J Med Chem; 1995 Sep; 38(19):3720-40. PubMed ID: 7562904
[TBL] [Abstract][Full Text] [Related]
15. Quinoxaline derivatives: structure-activity relationships and physiological implications of inhibition of N-methyl-D-aspartate and non-N-methyl-D-aspartate receptor-mediated currents and synaptic potentials.
Randle JC; Guet T; Bobichon C; Moreau C; Curutchet P; Lambolez B; de Carvalho LP; Cordi A; Lepagnol JM
Mol Pharmacol; 1992 Feb; 41(2):337-45. PubMed ID: 1371583
[TBL] [Abstract][Full Text] [Related]
16. Characterization of indole-2-carboxylate derivatives as antagonists of N-methyl-D-aspartate receptor activity at the associated glycine recognition site.
Hood WF; Gray NM; Dappen MS; Watson GB; Compton RP; Cordi AA; Lanthorn TH; Monahan JB
J Pharmacol Exp Ther; 1992 Aug; 262(2):654-60. PubMed ID: 1386886
[TBL] [Abstract][Full Text] [Related]
17. Evidence for heterogenous glycine domains but conserved multiple states of the excitatory amino acid recognition site of the NMDA receptor: regional binding studies with [3H]glycine and [3H]L-glutamate.
O'Shea RD; Manallack DT; Conway EL; Mercer LD; Beart PM
Exp Brain Res; 1991; 86(3):652-62. PubMed ID: 1684753
[TBL] [Abstract][Full Text] [Related]
18. NMDA receptor coagonist glycine site: evidence for a role in lateral hypothalamic stimulation of feeding.
Stanley BG; Butterfield BS; Grewal RS
Am J Physiol; 1997 Aug; 273(2 Pt 2):R790-6. PubMed ID: 9277570
[TBL] [Abstract][Full Text] [Related]
19. Gp120 can revert antagonism at the glycine site of NMDA receptors mediating GABA release from cultured hippocampal neurons.
Fontana G; Valenti L; Raiteri M
J Neurosci Res; 1997 Sep; 49(6):732-8. PubMed ID: 9335260
[TBL] [Abstract][Full Text] [Related]
20. Activity of 5,7-dichlorokynurenic acid, a potent antagonist at the N-methyl-D-aspartate receptor-associated glycine binding site.
Baron BM; Harrison BL; Miller FP; McDonald IA; Salituro FG; Schmidt CJ; Sorensen SM; White HS; Palfreyman MG
Mol Pharmacol; 1990 Oct; 38(4):554-61. PubMed ID: 2172769
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
