These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

343 related articles for article (PubMed ID: 18440098)

  • 1. Substituted benzo[d]oxazol-2(3H)-one derivatives with preference for the sigma1 binding site.
    Zampieri D; Grazia Mamolo M; Laurini E; Zanette C; Florio C; Collina S; Rossi D; Azzolina O; Vio L
    Eur J Med Chem; 2009 Jan; 44(1):124-30. PubMed ID: 18440098
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and quantitative structure-activity relationships of N-(1-benzylpiperidin-4-yl)phenylacetamides and related analogues as potent and selective sigma1 receptor ligands.
    Huang Y; Hammond PS; Whirrett BR; Kuhner RJ; Wu L; Childers SR; Mach RH
    J Med Chem; 1998 Jun; 41(13):2361-70. PubMed ID: 9632369
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Substituted benzylaminoalkylindoles with preference for the sigma2 binding site.
    Mamolo MG; Zampieri D; Zanette C; Florio C; Collina S; Urbano M; Azzolina O; Vio L
    Eur J Med Chem; 2008 Oct; 43(10):2073-81. PubMed ID: 18069094
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis, biological evaluation, and three-dimensional in silico pharmacophore model for sigma(1) receptor ligands based on a series of substituted benzo[d]oxazol-2(3H)-one derivatives.
    Zampieri D; Mamolo MG; Laurini E; Florio C; Zanette C; Fermeglia M; Posocco P; Paneni MS; Pricl S; Vio L
    J Med Chem; 2009 Sep; 52(17):5380-93. PubMed ID: 19673530
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Novel potent sigma 1 ligands: N-[omega-(tetralin-1-yl)alkyl]piperidine derivatives.
    Berardi F; Giudice G; Perrone R; Tortorella V; Govoni S; Lucchi L
    J Med Chem; 1996 Oct; 39(21):4255-60. PubMed ID: 8863803
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Halogenated 4-(phenoxymethyl)piperidines as potential radiolabeled probes for sigma-1 receptors: in vivo evaluation of [123I]-1-(iodopropen-2-yl)-4-[(4-cyanophenoxy)methyl]pip eri dine.
    Waterhouse RN; Mardon K; Giles KM; Collier TL; O'Brien JC
    J Med Chem; 1997 May; 40(11):1657-67. PubMed ID: 9171875
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Design, synthesis, and structure-affinity relationships of regioisomeric N-benzyl alkyl ether piperazine derivatives as sigma-1 receptor ligands.
    Moussa IA; Banister SD; Beinat C; Giboureau N; Reynolds AJ; Kassiou M
    J Med Chem; 2010 Aug; 53(16):6228-39. PubMed ID: 20662542
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and evaluation of aryl-substituted N-(arylethyl)-N-methyl-2-(1-pyrrolidinyl)ethylamines and corresponding arylacetamides for sigma receptor affinity.
    Zhang Y; Williams W; Bowen WD; Rice KC
    J Med Chem; 1996 Aug; 39(18):3564-8. PubMed ID: 8784455
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and structure-activity relationships of 1-aralkyl-4-benzylpiperidine and 1-aralkyl-4-benzylpiperazine derivatives as potent sigma ligands.
    Costantino L; Gandolfi F; Sorbi C; Franchini S; Prezzavento O; Vittorio F; Ronsisvalle G; Leonardi A; Poggesi E; Brasili L
    J Med Chem; 2005 Jan; 48(1):266-73. PubMed ID: 15634021
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Characterization of novel N,N'-disubstituted piperazines as sigma receptor ligands.
    Zhang Y; Williams W; Torrence-Campbell C; Bowen WD; Rice KC
    J Med Chem; 1998 Dec; 41(25):4950-7. PubMed ID: 9836612
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of novel 4- and 5-substituted benzyl ether derivatives of vesamicol and in vitro evaluation of their binding properties to the vesicular acetylcholine transporter site.
    Scheunemann M; Sorger D; Wenzel B; Heinitz K; Schliebs R; Klingner M; Sabri O; Steinbach J
    Bioorg Med Chem; 2004 Mar; 12(6):1459-65. PubMed ID: 15018919
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis and receptor binding studies of some new arylcarboxamide derivatives as sigma-1 ligands.
    Zampieri D; Laurini E; Vio L; Golob S; Fermeglia M; Pricl S; Mamolo MG
    Bioorg Med Chem Lett; 2014 Feb; 24(4):1021-5. PubMed ID: 24486131
    [TBL] [Abstract][Full Text] [Related]  

  • 13. 2(3H)-benzoxazolone and 2(3H)-benzothiazolone derivatives: novel, potent and selective sigma1 receptor ligands.
    Ucar H; Cacciaguerra S; Spampinato S; Van derpoorten K; Isa M; Kanyonyo M; Poupaert JH
    Eur J Pharmacol; 1997 Sep; 335(2-3):267-73. PubMed ID: 9369382
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Divergent Cytotoxic and Metabolically Stimulative Functions of Sigma-2 Receptors: Structure-Activity Relationships of 6-Acetyl-3-(4-(4-(4-fluorophenyl)piperazin-1-yl)butyl)benzo[
    Nicholson HE; Alsharif WF; Comeau AB; Mesangeau C; Intagliata S; Mottinelli M; McCurdy CR; Bowen WD
    J Pharmacol Exp Ther; 2019 Feb; 368(2):272-281. PubMed ID: 30530624
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Thiophene bioisosteres of spirocyclic sigma receptor ligands. 1. N-substituted spiro[piperidine-4,4'-thieno[3,2-c]pyrans].
    Oberdorf C; Schepmann D; Vela JM; Diaz JL; Holenz J; Wünsch B
    J Med Chem; 2008 Oct; 51(20):6531-7. PubMed ID: 18816044
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis, pharmacological activity and structure affinity relationships of spirocyclic σ(1) receptor ligands with a (2-fluoroethyl) residue in 3-position.
    Maestrup EG; Wiese C; Schepmann D; Brust P; Wünsch B
    Bioorg Med Chem; 2011 Jan; 19(1):393-405. PubMed ID: 21126878
    [TBL] [Abstract][Full Text] [Related]  

  • 17. (+)-cis-N-ethyleneamino-N-normetazocine derivatives. Novel and selective sigma ligands with antagonist properties.
    Ronsisvalle G; Marrazzo A; Prezzavento O; Pasquinucci L; Vittorio F; Pittalà V; Pappalardo MS; Cacciaguerra S; Spampinato S
    J Med Chem; 1998 May; 41(10):1574-80. PubMed ID: 9572883
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Chiral, nonracemic (piperazin-2-yl)methanol derivatives with sigma-receptor affinity.
    Bedürftig S; Wünsch B
    Bioorg Med Chem; 2004 Jun; 12(12):3299-311. PubMed ID: 15158798
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and structure-activity relationships of N-(3-phenylpropyl)-N'-benzylpiperazines: Potent ligands for sigma1 and sigma2 receptors.
    Nahas RI; Lever JR; Lever SZ
    Bioorg Med Chem; 2008 Jan; 16(2):755-61. PubMed ID: 18029187
    [TBL] [Abstract][Full Text] [Related]  

  • 20. N-[omega-(Tetralin-1-yl)alkyl] derivatives of 3,3-dimethylpiperidine are highly potent and selective sigma1 or sigma2 ligands.
    Berardi F; Santoro S; Perrone R; Tortorella V; Govoni S; Lucchi L
    J Med Chem; 1998 Oct; 41(21):3940-7. PubMed ID: 9767631
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 18.