BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

211 related articles for article (PubMed ID: 18452016)

  • 21. Indene-based scaffolds. 2. An indole-indene switch: discovery of novel indenylsulfonamides as 5-HT6 serotonin receptor agonists.
    Alcalde E; Mesquida N; López-Pérez S; Frigola J; Mercè R
    J Med Chem; 2009 Feb; 52(3):675-87. PubMed ID: 19159187
    [TBL] [Abstract][Full Text] [Related]  

  • 22. Novel 1-(azacyclyl)-3-arylsulfonyl-1H-pyrrolo[2,3-b]pyridines as 5-HT6 agonists and antagonists.
    Elokdah H; Li D; McFarlane G; Bernotas RC; Robichaud AJ; Magolda RL; Zhang GM; Smith D; Schechter LE
    Bioorg Med Chem; 2007 Sep; 15(18):6208-26. PubMed ID: 17624788
    [TBL] [Abstract][Full Text] [Related]  

  • 23. Discovery of indole-containing tetracycles as a new scaffold for androgen receptor ligands.
    Zhang X; Li X; Allan GF; Musto A; Lundeen SG; Sui Z
    Bioorg Med Chem Lett; 2006 Jun; 16(12):3233-7. PubMed ID: 16603353
    [TBL] [Abstract][Full Text] [Related]  

  • 24. Synthesis of 3-(2'-furoyl)indole derivatives as potential new ligands at the benzodiazepine receptor, structurally more restrained analogues of indoleglyoxylylamides.
    Da Settimo A; Primofiore G; Da Settimo F; Marini AM; Novellino E; Greco G; Martini C; Senatore G; Lucacchini A
    Farmaco; 1995 May; 50(5):311-20. PubMed ID: 7626165
    [TBL] [Abstract][Full Text] [Related]  

  • 25. Indene-based scaffolds. Design and synthesis of novel serotonin 5-HT6 receptor ligands.
    Alcalde E; Mesquida N; Frigola J; López-Pérez S; Mercè R
    Org Biomol Chem; 2008 Oct; 6(20):3795-810. PubMed ID: 18843410
    [TBL] [Abstract][Full Text] [Related]  

  • 26. 1-(1-Naphthyl)piperazine as a novel template for 5-HT6 serotonin receptor ligands.
    Lee M; Rangisetty JB; Pullagurla MR; Dukat M; Setola V; Roth BL; Glennon RA
    Bioorg Med Chem Lett; 2005 Mar; 15(6):1707-11. PubMed ID: 15745826
    [TBL] [Abstract][Full Text] [Related]  

  • 27. Synthesis and structure guided evaluation of estrogen agonist and antagonist activities of some new tetrazolyl indole derivatives.
    Singh US; Shankar R; Yadav GP; Kharkwal G; Dwivedi A; Keshri G; Singh MM; Moulik PR; Hajela K
    Eur J Med Chem; 2008 Oct; 43(10):2149-58. PubMed ID: 18155810
    [TBL] [Abstract][Full Text] [Related]  

  • 28. Novel 3-aminochromans as potential pharmacological tools for the serotonin 5-HT(7) receptor.
    Holmberg P; Tedenborg L; Rosqvist S; Johansson AM
    Bioorg Med Chem Lett; 2005 Feb; 15(3):747-50. PubMed ID: 15664850
    [TBL] [Abstract][Full Text] [Related]  

  • 29. Carbon-11 labeled indolylpropylamine analog as a new potential PET agent for imaging of the serotonin transporter.
    Ben-Daniel R; Deuther-Conrad W; Scheunemann M; Steinbach J; Brust P; Mishani E
    Bioorg Med Chem; 2008 Jun; 16(12):6364-70. PubMed ID: 18487050
    [TBL] [Abstract][Full Text] [Related]  

  • 30. Identification of a series of benzoxazoles as potent 5-HT6 ligands.
    Liu KG; Lo JR; Comery TA; Zhang GM; Zhang JY; Kowal DM; Smith DL; Di L; Kerns EH; Schechter LE; Robichaud AJ
    Bioorg Med Chem Lett; 2009 Feb; 19(4):1115-7. PubMed ID: 19152787
    [TBL] [Abstract][Full Text] [Related]  

  • 31. Synthesis and antioxidant properties of some indole ethylamine derivatives as melatonin analogs.
    Ates-Alagoz Z; Buyukbingol Z; Buyukbingol E
    Pharmazie; 2005 Sep; 60(9):643-7. PubMed ID: 16222860
    [TBL] [Abstract][Full Text] [Related]  

  • 32. Novel antagonists of serotonin-4 receptors: synthesis and biological evaluation of pyrrolothienopyrazines.
    Lemaître S; Lepailleur A; Bureau R; Butt-Gueulle S; Lelong-Boulouard V; Duchatelle P; Boulouard M; Dumuis A; Daveu C; Lezoualc'h F; Pfeiffer B; Dauphin F; Rault S
    Bioorg Med Chem; 2009 Mar; 17(6):2607-22. PubMed ID: 19261477
    [TBL] [Abstract][Full Text] [Related]  

  • 33. N2-benzyl-N1-(1-(1-naphthyl)ethyl)-3-phenylpropane-1,2-diamines and conformationally restrained indole analogues: development of calindol as a new calcimimetic acting at the calcium sensing receptor.
    Kessler A; Faure H; Petrel C; Ruat M; Dauban P; Dodd RH
    Bioorg Med Chem Lett; 2004 Jun; 14(12):3345-9. PubMed ID: 15149704
    [TBL] [Abstract][Full Text] [Related]  

  • 34. Stereoselective synthesis of both enantiomers of N-aryl indoles with axially chiral N-C bonds.
    Kamikawa K; Kinoshita S; Furusyo M; Takemoto S; Matsuzaka H; Uemura M
    J Org Chem; 2007 Apr; 72(9):3394-402. PubMed ID: 17394356
    [TBL] [Abstract][Full Text] [Related]  

  • 35. N-arylsulfonyl-2-vinyltryptamines as new 5-HT6 serotonin receptor ligands.
    Raoul M; Patigny D; Fabis F; Dauphin F; Rault S; Sapi J; Laronze JY
    J Enzyme Inhib Med Chem; 2006 Jun; 21(3):251-60. PubMed ID: 16918072
    [TBL] [Abstract][Full Text] [Related]  

  • 36. A new entry to polycyclic indole derivatives via intramolecular imino Diels-Alder reaction: observation of unexpected reaction.
    Gaddam V; Nagarajan R
    J Org Chem; 2007 Apr; 72(9):3573-6. PubMed ID: 17408284
    [TBL] [Abstract][Full Text] [Related]  

  • 37. Synthesis and biological evaluation of novel gamma-carboline analogues of Dimebon as potent 5-HT6 receptor antagonists.
    Ivachtchenko AV; Frolov EB; Mitkin OD; Kysil VM; Khvat AV; Okun IM; Tkachenko SE
    Bioorg Med Chem Lett; 2009 Jun; 19(12):3183-7. PubMed ID: 19443217
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Tetrahydrothienopyridylbutyl-tetrahydrobenzindoles: new selective ligands of the 5-HT(7) receptor.
    Kikuchi C; Hiranuma T; Koyama M
    Bioorg Med Chem Lett; 2002 Sep; 12(18):2549-52. PubMed ID: 12182857
    [TBL] [Abstract][Full Text] [Related]  

  • 39. Influence of amine substituents on 5-HT2A versus 5-HT2C binding of phenylalkyl- and indolylalkylamines.
    Glennon RA; Dukat M; el-Bermawy M; Law H; De los Angeles J; Teitler M; King A; Herrick-Davis K
    J Med Chem; 1994 Jun; 37(13):1929-35. PubMed ID: 8027974
    [TBL] [Abstract][Full Text] [Related]  

  • 40. Binding of methoxy-substituted N1-benzenesulfonylindole analogs at human 5-HT6 serotonin receptors.
    Siripurapu U; Kolanos R; Dukat M; Roth BL; Glennon RA
    Bioorg Med Chem Lett; 2006 Jul; 16(14):3793-6. PubMed ID: 16709453
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 11.