BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

442 related articles for article (PubMed ID: 18538567)

  • 1. Antimalarial activity of novel pyrrolizidinyl derivatives of 4-aminoquinoline.
    Sparatore A; Basilico N; Casagrande M; Parapini S; Taramelli D; Brun R; Wittlin S; Sparatore F
    Bioorg Med Chem Lett; 2008 Jul; 18(13):3737-40. PubMed ID: 18538567
    [TBL] [Abstract][Full Text] [Related]  

  • 2. 4-Aminoquinoline quinolizidinyl- and quinolizidinylalkyl-derivatives with antimalarial activity.
    Sparatore A; Basilico N; Parapini S; Romeo S; Novelli F; Sparatore F; Taramelli D
    Bioorg Med Chem; 2005 Sep; 13(18):5338-45. PubMed ID: 16054368
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis, antimalarial activity, and cellular toxicity of new arylpyrrolylaminoquinolines.
    Casagrande M; Basilico N; Rusconi C; Taramelli D; Sparatore A
    Bioorg Med Chem; 2010 Sep; 18(18):6625-33. PubMed ID: 20797868
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Antimalarial activity of novel 5-aryl-8-aminoquinoline derivatives.
    Shiraki H; Kozar MP; Melendez V; Hudson TH; Ohrt C; Magill AJ; Lin AJ
    J Med Chem; 2011 Jan; 54(1):131-42. PubMed ID: 21141892
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and bioevaluation of hybrid 4-aminoquinoline triazines as a new class of antimalarial agents.
    Kumar A; Srivastava K; Raja Kumar S; Puri SK; Chauhan PM
    Bioorg Med Chem Lett; 2008 Dec; 18(24):6530-3. PubMed ID: 18951791
    [TBL] [Abstract][Full Text] [Related]  

  • 6. 4-aminoquinoline-triazine-based hybrids with improved in vitro antimalarial activity against CQ-sensitive and CQ-resistant strains of Plasmodium falciparum.
    Manohar S; Khan SI; Rawat DS
    Chem Biol Drug Des; 2013 May; 81(5):625-30. PubMed ID: 23331618
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Toward a novel metal-based chemotherapy against tropical diseases. 2. Synthesis and antimalarial activity in vitro and in vivo of new ruthenium- and rhodium-chloroquine complexes.
    Sánchez-Delgado RA; Navarro M; Pérez H; Urbina JA
    J Med Chem; 1996 Mar; 39(5):1095-99. PubMed ID: 8676344
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis, antimalarial activity and cytotoxicity of 4-aminoquinoline-triazine conjugates.
    Manohar S; Khan SI; Rawat DS
    Bioorg Med Chem Lett; 2010 Jan; 20(1):322-5. PubMed ID: 19910192
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and antimalarial activity in vitro and in vivo of a new ferrocene-chloroquine analogue.
    Biot C; Glorian G; Maciejewski LA; Brocard JS
    J Med Chem; 1997 Nov; 40(23):3715-8. PubMed ID: 9371235
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis, antimalarial activity, and preclinical pharmacology of a novel series of 4'-fluoro and 4'-chloro analogues of amodiaquine. Identification of a suitable "back-up" compound for N-tert-butyl isoquine.
    O'Neill PM; Shone AE; Stanford D; Nixon G; Asadollahy E; Park BK; Maggs JL; Roberts P; Stocks PA; Biagini G; Bray PG; Davies J; Berry N; Hall C; Rimmer K; Winstanley PA; Hindley S; Bambal RB; Davis CB; Bates M; Gresham SL; Brigandi RA; Gomez-de-Las-Heras FM; Gargallo DV; Parapini S; Vivas L; Lander H; Taramelli D; Ward SA
    J Med Chem; 2009 Apr; 52(7):1828-44. PubMed ID: 19284751
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Optimization of 4-aminoquinoline/clotrimazole-based hybrid antimalarials: further structure-activity relationships, in vivo studies, and preliminary toxicity profiling.
    Gemma S; Camodeca C; Sanna Coccone S; Joshi BP; Bernetti M; Moretti V; Brogi S; Bonache de Marcos MC; Savini L; Taramelli D; Basilico N; Parapini S; Rottmann M; Brun R; Lamponi S; Caccia S; Guiso G; Summers RL; Martin RE; Saponara S; Gorelli B; Novellino E; Campiani G; Butini S
    J Med Chem; 2012 Aug; 55(15):6948-67. PubMed ID: 22783984
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Candidate selection and preclinical evaluation of N-tert-butyl isoquine (GSK369796), an affordable and effective 4-aminoquinoline antimalarial for the 21st century.
    O'Neill PM; Park BK; Shone AE; Maggs JL; Roberts P; Stocks PA; Biagini GA; Bray PG; Gibbons P; Berry N; Winstanley PA; Mukhtar A; Bonar-Law R; Hindley S; Bambal RB; Davis CB; Bates M; Hart TK; Gresham SL; Lawrence RM; Brigandi RA; Gomez-delas-Heras FM; Gargallo DV; Ward SA
    J Med Chem; 2009 Mar; 52(5):1408-15. PubMed ID: 19222165
    [TBL] [Abstract][Full Text] [Related]  

  • 13. The chemotherapy of rodent malaria, XXXVIII. Studies on the activity of three new antimalarials (WR 194,965, WR 228,258 and WR 225,448) against rodent and human malaria parasites (Plasmodium berghei and P. falciparum).
    Peters W; Irare SG; Ellis DS; Warhurst DC; Robinson BL
    Ann Trop Med Parasitol; 1984 Dec; 78(6):567-79. PubMed ID: 6398032
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and antimalarial activity of side chain modified 4-aminoquinoline derivatives.
    Solomon VR; Haq W; Srivastava K; Puri SK; Katti SB
    J Med Chem; 2007 Jan; 50(2):394-8. PubMed ID: 17228883
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Imidazolidin-4-one peptidomimetic derivatives of primaquine: synthesis and antimalarial activity.
    Vale N; Matos J; Gut J; Nogueira F; do Rosário V; Rosenthal PJ; Moreira R; Gomes P
    Bioorg Med Chem Lett; 2008 Jul; 18(14):4150-3. PubMed ID: 18539459
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Design and synthesis of new antimalarial agents from 4-aminoquinoline.
    Solomon VR; Puri SK; Srivastava K; Katti SB
    Bioorg Med Chem; 2005 Mar; 13(6):2157-65. PubMed ID: 15727868
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Antimalarial activity of 4-(5-trifluoromethyl-1H-pyrazol-1-yl)-chloroquine analogues.
    Cunico W; Cechinel CA; Bonacorso HG; Martins MA; Zanatta N; de Souza MV; Freitas IO; Soares RP; Krettli AU
    Bioorg Med Chem Lett; 2006 Feb; 16(3):649-53. PubMed ID: 16257205
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synergistic interaction of a chloroquine metabolite with chloroquine against drug-resistant malaria parasites.
    Kalkanidis M; Klonis N; Tschan S; Deady LW; Tilley L
    Biochem Pharmacol; 2004 Apr; 67(7):1347-53. PubMed ID: 15013850
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and evaluation of sulfonylurea derivatives as novel antimalarials.
    León C; Rodrigues J; Gamboa de Domínguez N; Charris J; Gut J; Rosenthal PJ; Domínguez JN
    Eur J Med Chem; 2007 Jun; 42(6):735-42. PubMed ID: 17321641
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Evaluation of the antimalarial activity of new compounds against Plasmodium falciparum in vitro, and Plasmodium berghei in vivo.
    Tedlaouti F; Gasquet M; Delmas F; Timon-David P; Madadi NE; Vanelle P; Maldonado J
    J Pharm Belg; 1990; 45(5):306-10. PubMed ID: 2086754
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 23.