BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

135 related articles for article (PubMed ID: 18640043)

  • 1. Muscarinic receptor 1 agonist activity of novel N-arylthioureas substituted 3-morpholino arecoline derivatives in Alzheimer's presenile dementia models.
    Malviya M; Kumar YC; Asha D; Chandra JN; Subhash MN; Rangappa KS
    Bioorg Med Chem; 2008 Aug; 16(15):7095-101. PubMed ID: 18640043
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Muscarinic receptor 1 agonist activity of novel N-aryl carboxamide substituted 3-morpholino arecoline derivatives in Alzheimer's presenile dementia models.
    Malviya M; Kumar YC; Mythri RB; Venkateshappa C; Subhash MN; Rangappa KS
    Bioorg Med Chem; 2009 Aug; 17(15):5526-34. PubMed ID: 19595599
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Effect of novel N-aryl sulfonamide substituted 3-morpholino arecoline derivatives as muscarinic receptor 1 agonists in Alzheimer's dementia models.
    Kumar YC; Malviya M; Chandra JN; Sadashiva CT; Kumar CS; Prasad SB; Prasanna DS; Subhash MN; Rangappa KS
    Bioorg Med Chem; 2008 May; 16(9):5157-63. PubMed ID: 18359231
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Effect of novel arecoline thiazolidinones as muscarinic receptor 1 agonist in Alzheimer's dementia models.
    Chandra JN; Malviya M; Sadashiva CT; Subhash MN; Rangappa KS
    Neurochem Int; 2008 Feb; 52(3):376-83. PubMed ID: 17719699
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and pharmacological evaluation of novel N-alkyl/aryl substituted thiazolidinone arecoline analogues as muscarinic receptor 1 agonist in Alzheimer's dementia models.
    Sadashiva CT; Chandra JN; Kavitha CV; Thimmegowda A; Subhash MN; Rangappa KS
    Eur J Med Chem; 2009 Dec; 44(12):4848-54. PubMed ID: 19717214
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and biological characterization of 1,4,5,6-tetrahydropyrimidine and 2-amino-3,4,5,6-tetrahydropyridine derivatives as selective m1 agonists.
    Messer WS; Abuh YF; Liu Y; Periyasamy S; Ngur DO; Edgar MA; El-Assadi AA; Sbeih S; Dunbar PG; Roknich S; Rho T; Fang Z; Ojo B; Zhang H; Huzl JJ; Nagy PI
    J Med Chem; 1997 Apr; 40(8):1230-46. PubMed ID: 9111297
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Bioisosteres of arecoline: 1,2,3,6-tetrahydro-5-pyridyl-substituted and 3-piperidyl-substituted derivatives of tetrazoles and 1,2,3-triazoles. Synthesis and muscarinic activity.
    Moltzen EK; Pedersen H; Bøgesø KP; Meier E; Frederiksen K; Sánchez C; Løve Lembøl H
    J Med Chem; 1994 Nov; 37(24):4085-99. PubMed ID: 7990109
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Quantitative structure-selectivity relationship for M2 selectivity between M1 and M2 of piperidinyl piperidine derivatives as muscarinic antagonists.
    Niu YY; Yang LM; Deng KM; Yao JH; Zhu L; Chen CY; Zhang M; Zhou JE; Shen TX; Chen HZ; Lu Y
    Bioorg Med Chem Lett; 2007 Apr; 17(8):2260-6. PubMed ID: 17289384
    [TBL] [Abstract][Full Text] [Related]  

  • 9. 1,2,5-Thiadiazole derivatives of arecoline stimulate M1 receptors coupled to phosphoinositide turnover.
    Periyasamy S; Messer WS; Roknich S; Sauerberg P; Hoss W
    Brain Res; 1995 Sep; 693(1-2):118-23. PubMed ID: 8653399
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Cognitive effects of muscarinic M1 functional agonists in non-human primates and clinical trials.
    McArthur RA; Gray J; Schreiber R
    Curr Opin Investig Drugs; 2010 Jul; 11(7):740-60. PubMed ID: 20571970
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Inhibitory effect of curcuminoids on acetylcholinesterase activity and attenuation of scopolamine-induced amnesia may explain medicinal use of turmeric in Alzheimer's disease.
    Ahmed T; Gilani AH
    Pharmacol Biochem Behav; 2009 Feb; 91(4):554-9. PubMed ID: 18930076
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Active site directed docking studies: synthesis and pharmacological evaluation of cis-2,6-dimethyl piperidine sulfonamides as inhibitors of acetylcholinesterase.
    Girisha HR; Narendra Sharath Chandra JN; Boppana S; Malviya M; Sadashiva CT; Rangappa KS
    Eur J Med Chem; 2009 Oct; 44(10):4057-62. PubMed ID: 19493592
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Discovery of N-substituted 7-azaindoline derivatives as potent, orally available M1 and M4 muscarinic acetylcholine receptors selective agonists.
    Takai K; Inoue Y; Konishi Y; Suwa A; Uruno Y; Matsuda H; Nakako T; Sakai M; Nishikawa H; Hashimoto G; Enomoto T; Kitamura A; Uematsu Y; Kiyoshi A; Sumiyoshi T
    Bioorg Med Chem Lett; 2014 Jul; 24(14):3189-93. PubMed ID: 24856064
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Discovery of N-{1-[3-(3-oxo-2,3-dihydrobenzo[1,4]oxazin-4-yl)propyl]piperidin-4-yl}-2-phenylacetamide (Lu AE51090): an allosteric muscarinic M1 receptor agonist with unprecedented selectivity and procognitive potential.
    Sams AG; Hentzer M; Mikkelsen GK; Larsen K; Bundgaard C; Plath N; Christoffersen CT; Bang-Andersen B
    J Med Chem; 2010 Sep; 53(17):6386-97. PubMed ID: 20684563
    [TBL] [Abstract][Full Text] [Related]  

  • 15. The profile of sabcomeline (SB-202026), a functionally selective M1 receptor partial agonist, in the marmoset.
    Harries MH; Samson NA; Cilia J; Hunter AJ
    Br J Pharmacol; 1998 May; 124(2):409-15. PubMed ID: 9641560
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis and biological evaluation of isoxazoline derivatives as potent M₁ muscarinic acetylcholine receptor agonists.
    Huang M; Suk DH; Cho NC; Bhattarai D; Kang SB; Kim Y; Pae AN; Rhim H; Keum G
    Bioorg Med Chem Lett; 2015 Apr; 25(7):1546-51. PubMed ID: 25765911
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Alzheimer's disease.
    Pomara N; Sidtis JJ
    N Engl J Med; 2010 May; 362(19):1844; author reply 1844-5. PubMed ID: 20463348
    [No Abstract]   [Full Text] [Related]  

  • 18. [Synthesis and vascular relaxing activity of arecoline derivatives coupled with nitric oxide donors].
    Huang ST; Huang WL; Zhang HB
    Yao Xue Xue Bao; 2006 Jan; 41(1):71-5. PubMed ID: 16683531
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Enhanced arecoline derivatives as muscarinic acetylcholine receptor M1 ligands for potential application as PET radiotracers.
    Ozenil M; Pacher K; Balber T; Vraka C; Roller A; Holzer W; Spreitzer H; Mitterhauser M; Wadsak W; Hacker M; Pichler V
    Eur J Med Chem; 2020 Oct; 204():112623. PubMed ID: 32717485
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Ex vivo study of 5-HT(1A) and 5-HT(7) receptor agonists and antagonists on cAMP accumulation during memory formation and amnesia.
    Perez-García G; Meneses A
    Behav Brain Res; 2008 Dec; 195(1):139-46. PubMed ID: 18723050
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.