BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

169 related articles for article (PubMed ID: 18674899)

  • 1. Synthesis and antiviral properties of some polyphenols related to Salvia genus.
    Queffélec C; Bailly F; Mbemba G; Mouscadet JF; Hayes S; Debyser Z; Witvrouw M; Cotelle P
    Bioorg Med Chem Lett; 2008 Aug; 18(16):4736-40. PubMed ID: 18674899
    [TBL] [Abstract][Full Text] [Related]  

  • 2. A potent anti-HIV polyphenol from Salvia yunnanensis.
    Zhang ZF; Chen HS; Peng ZG; Li ZR; Jiang JD
    J Asian Nat Prod Res; 2008; 10(3-4):273-7. PubMed ID: 18335344
    [TBL] [Abstract][Full Text] [Related]  

  • 3. N-(4-Fluorobenzyl)-3-hydroxy-9,9-dimethyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrazino[1,2-a]pyrimidine-2-carboxamides a novel class of potent HIV-1 integrase inhibitors.
    Petrocchi A; Jones P; Rowley M; Fiore F; Summa V
    Bioorg Med Chem Lett; 2009 Aug; 19(15):4245-9. PubMed ID: 19523819
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Efficient synthesis and utilization of phenyl-substituted heteroaromatic carboxylic acids as aryl diketo acid isosteres in the design of novel HIV-1 integrase inhibitors.
    Zeng LF; Zhang HS; Wang YH; Sanchez T; Zheng YT; Neamati N; Long YQ
    Bioorg Med Chem Lett; 2008 Aug; 18(16):4521-4. PubMed ID: 18662877
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis of trans-caffeate analogues and their bioactivities against HIV-1 integrase and cancer cell lines.
    Xia CN; Li HB; Liu F; Hu WX
    Bioorg Med Chem Lett; 2008 Dec; 18(24):6553-7. PubMed ID: 18952420
    [TBL] [Abstract][Full Text] [Related]  

  • 6. 4-Hydroxy-5-pyrrolinone-3-carboxamide HIV-1 integrase inhibitors.
    Pace P; Spieser SA; Summa V
    Bioorg Med Chem Lett; 2008 Jul; 18(14):3865-9. PubMed ID: 18595690
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Naphthoxazepine inhibitors of HIV-1 integrase: synthesis and biological evaluation.
    Garofalo A; Grande F; Brizzi A; Aiello F; Dayam R; Neamati N
    ChemMedChem; 2008 Jun; 3(6):986-90. PubMed ID: 18383063
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis of potent antitumor and antiviral benzofuran derivatives.
    Galal SA; Abd El-All AS; Abdallah MM; El-Diwani HI
    Bioorg Med Chem Lett; 2009 May; 19(9):2420-8. PubMed ID: 19345581
    [TBL] [Abstract][Full Text] [Related]  

  • 9. The use of oxadiazole and triazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 1: Establishing the pharmacophore.
    Johns BA; Weatherhead JG; Allen SH; Thompson JB; Garvey EP; Foster SA; Jeffrey JL; Miller WH
    Bioorg Med Chem Lett; 2009 Mar; 19(6):1802-6. PubMed ID: 19217781
    [TBL] [Abstract][Full Text] [Related]  

  • 10. The total synthesis of fukiic acid, an HIV-1 integrase inhibitor.
    Queffélec C; Bailly F; Mbemba G; Mouscadet JF; Debyser Z; Witvrouw M; Cotelle P
    Eur J Med Chem; 2008 Oct; 43(10):2268-71. PubMed ID: 18243421
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Anti-HBV agents. Part 1: Synthesis of alisol A derivatives: a new class of hepatitis B virus inhibitors.
    Zhang Q; Jiang ZY; Luo J; Cheng P; Ma YB; Zhang XM; Zhang FX; Zhou J; Chen JJ
    Bioorg Med Chem Lett; 2008 Aug; 18(16):4647-50. PubMed ID: 18644720
    [TBL] [Abstract][Full Text] [Related]  

  • 12. 1,3,4-Oxadiazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 2: SAR of the C5 position.
    Johns BA; Weatherhead JG; Allen SH; Thompson JB; Garvey EP; Foster SA; Jeffrey JL; Miller WH
    Bioorg Med Chem Lett; 2009 Mar; 19(6):1807-10. PubMed ID: 19217284
    [TBL] [Abstract][Full Text] [Related]  

  • 13. 10-Hydroxy-7,8-dihydropyrazino[1',2':1,5]pyrrolo[2,3-d]pyridazine-1,9(2H,6H)-diones: potent, orally bioavailable HIV-1 integrase strand-transfer inhibitors with activity against integrase mutants.
    Wiscount CM; Williams PD; Tran LO; Embrey MW; Fisher TE; Sherman V; Homnick CF; Donnette Staas D; Lyle TA; Wai JS; Vacca JP; Wang Z; Felock PJ; Stillmock KA; Witmer MV; Miller MD; Hazuda DJ; Day AM; Gabryelski LJ; Ecto LT; Schleif WA; DiStefano DJ; Kochansky CJ; Anari MR
    Bioorg Med Chem Lett; 2008 Aug; 18(16):4581-3. PubMed ID: 18657970
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Phosphorous acid analogs of novel P2-P4 macrocycles as inhibitors of HCV-NS3 protease.
    Pompei M; Francesco ME; Koch U; Liverton NJ; Summa V
    Bioorg Med Chem Lett; 2009 May; 19(9):2574-8. PubMed ID: 19328685
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and HIV-1 integrase inhibitory activities of caffeic acid dimers derived from Salvia officinalis.
    Bailly F; Queffelec C; Mbemba G; Mouscadet JF; Cotelle P
    Bioorg Med Chem Lett; 2005 Nov; 15(22):5053-6. PubMed ID: 16183277
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Biologically-validated HIV integrase inhibitors with nucleobase scaffolds: structure, synthesis, chemical biology, molecular modeling, and antiviral activity.
    Nair V; Uchil V; Chi G; Dams I; Cox A; Seo B
    Nucleosides Nucleotides Nucleic Acids; 2007; 26(6-7):665-8. PubMed ID: 18066876
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis of 4-oxo-4,7-dihydrofuro[2,3-b]pyridine-5-carboxamides with broad-spectrum human herpesvirus polymerase inhibition.
    Schnute ME; Brideau RJ; Collier SA; Cudahy MM; Hopkins TA; Knechtel ML; Oien NL; Sackett RS; Scott A; Stephan ML; Wathen MW; Wieber JL
    Bioorg Med Chem Lett; 2008 Jul; 18(14):3856-9. PubMed ID: 18595689
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Radical-scavenging polyphenols: new strategies for their synthesis.
    Bovicelli P
    J Pharm Pharmacol; 2007 Dec; 59(12):1703-10. PubMed ID: 18053333
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Design, synthesis, and biological evaluation of a series of 2-hydroxyisoquinoline-1,3(2H,4H)-diones as dual inhibitors of human immunodeficiency virus type 1 integrase and the reverse transcriptase RNase H domain.
    Billamboz M; Bailly F; Barreca ML; De Luca L; Mouscadet JF; Calmels C; Andréola ML; Witvrouw M; Christ F; Debyser Z; Cotelle P
    J Med Chem; 2008 Dec; 51(24):7717-30. PubMed ID: 19053754
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design, synthesis, and SAR studies of novel and highly active tri-cyclic HIV integrase inhibitors.
    Jin H; Cai RZ; Schacherer L; Jabri S; Tsiang M; Fardis M; Chen X; Chen JM; Kim CU
    Bioorg Med Chem Lett; 2006 Aug; 16(15):3989-92. PubMed ID: 16723225
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 9.