These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

534 related articles for article (PubMed ID: 18752957)

  • 1. Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents.
    Biava M; Porretta GC; Poce G; Supino S; Manetti F; Forli S; Botta M; Sautebin L; Rossi A; Pergola C; Ghelardini C; Norcini M; Makovec F; Giordani A; Anzellotti P; Cirilli R; Ferretti R; Gallinella B; La Torre F; Anzini M; Patrignani P
    Bioorg Med Chem; 2008 Sep; 16(17):8072-81. PubMed ID: 18752957
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis, biological evaluation, and enzyme docking simulations of 1,5-diarylpyrrole-3-alkoxyethyl ethers as selective cyclooxygenase-2 inhibitors endowed with anti-inflammatory and antinociceptive activity.
    Anzini M; Rovini M; Cappelli A; Vomero S; Manetti F; Botta M; Sautebin L; Rossi A; Pergola C; Ghelardini C; Norcini M; Giordani A; Makovec F; Anzellotti P; Patrignani P; Biava M
    J Med Chem; 2008 Aug; 51(15):4476-81. PubMed ID: 18598017
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Novel ester and acid derivatives of the 1,5-diarylpyrrole scaffold as anti-inflammatory and analgesic agents. Synthesis and in vitro and in vivo biological evaluation.
    Biava M; Porretta GC; Poce G; Battilocchio C; Manetti F; Botta M; Forli S; Sautebin L; Rossi A; Pergola C; Ghelardini C; Galeotti N; Makovec F; Giordani A; Anzellotti P; Patrignani P; Anzini M
    J Med Chem; 2010 Jan; 53(2):723-33. PubMed ID: 19957931
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Cyclooxygenase-2 inhibitors. 1,5-diarylpyrrol-3-acetic esters with enhanced inhibitory activity toward cyclooxygenase-2 and improved cyclooxygenase-2/cyclooxygenase-1 selectivity.
    Biava M; Porretta GC; Poce G; Supino S; Forli S; Rovini M; Cappelli A; Manetti F; Botta M; Sautebin L; Rossi A; Pergola C; Ghelardini C; Vivoli E; Makovec F; Anzellotti P; Patrignani P; Anzini M
    J Med Chem; 2007 Nov; 50(22):5403-11. PubMed ID: 17915854
    [TBL] [Abstract][Full Text] [Related]  

  • 5. In-vivo analgesic and anti-inflammatory activities of newly synthesized benzimidazole derivatives.
    Achar KC; Hosamani KM; Seetharamareddy HR
    Eur J Med Chem; 2010 May; 45(5):2048-54. PubMed ID: 20133024
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and pharmacological evaluation of 2(3H)-furanones and 2(3H)-pyrrolones, combining analgesic and anti-inflammatory properties with reduced gastrointestinal toxicity and lipid peroxidation.
    Alam MM; Husain A; Hasan SM; Suruchi ; Anwer T
    Eur J Med Chem; 2009 Jun; 44(6):2636-42. PubMed ID: 19059680
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Amide derivatives of [5-chloro-6-(2-chloro/fluorobenzoyl)-2-benzoxazolinone-3-yl]acetic acids as potential analgesic and anti-inflammatory compounds.
    Banoglu E; Okçelik B; Kupeli E; Unlü S; Yeşilada E; Amat M; Caturla JF; Sahin MF
    Arch Pharm (Weinheim); 2003 Jul; 336(4-5):251-7. PubMed ID: 12916060
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis of some new pyrimido[2',1':2,3]thiazolo[4,5-b]quinoxaline derivatives as anti-inflammatory and analgesic agents.
    Abu-Hashem AA; Gouda MA; Badria FA
    Eur J Med Chem; 2010 May; 45(5):1976-81. PubMed ID: 20149490
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Novel anti-inflammatory agents based on pyridazinone scaffold; design, synthesis and in vivo activity.
    Abouzid K; Bekhit SA
    Bioorg Med Chem; 2008 May; 16(10):5547-56. PubMed ID: 18430576
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis, analgesic and anti-inflammatory evaluation of some new 3H-quinazolin-4-one derivatives.
    Alafeefy AM; Kadi AA; El-Azab AS; Abdel-Hamide SG; Daba MH
    Arch Pharm (Weinheim); 2008 Jun; 341(6):377-85. PubMed ID: 18535995
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of biologically active N-methyl derivatives of amidines and cyclized five-membered products of amidines with oxalyl chloride.
    Sondhi SM; Dinodia M; Jain S; Kumar A
    Eur J Med Chem; 2008 Dec; 43(12):2824-30. PubMed ID: 18022734
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Aroylpropionic acid based 2,5-disubstituted-1,3,4-oxadiazoles: synthesis and their anti-inflammatory and analgesic activities.
    Akhter M; Husain A; Azad B; Ajmal M
    Eur J Med Chem; 2009 Jun; 44(6):2372-8. PubMed ID: 18977556
    [TBL] [Abstract][Full Text] [Related]  

  • 13. 1,2-Diarylpyrroles as potent and selective inhibitors of cyclooxygenase-2.
    Khanna IK; Weier RM; Yu Y; Collins PW; Miyashiro JM; Koboldt CM; Veenhuizen AW; Currie JL; Seibert K; Isakson PC
    J Med Chem; 1997 May; 40(11):1619-33. PubMed ID: 9171872
    [TBL] [Abstract][Full Text] [Related]  

  • 14. New cyclooxygenase-2/5-lipoxygenase inhibitors. 3. 7-tert-butyl-2, 3-dihydro-3,3-dimethylbenzofuran derivatives as gastrointestinal safe antiinflammatory and analgesic agents: variations at the 5 position.
    Janusz JM; Young PA; Ridgeway JM; Scherz MW; Enzweiler K; Wu LI; Gan L; Chen J; Kellstein DE; Green SA; Tulich JL; Rosario-Jansen T; Magrisso IJ; Wehmeyer KR; Kuhlenbeck DL; Eichhold TH; Dobson RL
    J Med Chem; 1998 Aug; 41(18):3515-29. PubMed ID: 9719605
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis, characterization, evaluation and molecular dynamics studies of 5, 6-diphenyl-1,2,4-triazin-3(2H)-one derivatives bearing 5-substituted 1,3,4-oxadiazole as potential anti-inflammatory and analgesic agents.
    Banerjee AG; Das N; Shengule SA; Srivastava RS; Shrivastava SK
    Eur J Med Chem; 2015 Aug; 101():81-95. PubMed ID: 26117820
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Design, synthesis and analgesic/anti-inflammatory evaluation of novel diarylthiazole and diarylimidazole derivatives towards selective COX-1 inhibitors with better gastric profile.
    Abdelazeem AH; El-Saadi MT; Safi El-Din AG; Omar HA; El-Moghazy SM
    Bioorg Med Chem; 2017 Jan; 25(2):665-676. PubMed ID: 27916468
    [TBL] [Abstract][Full Text] [Related]  

  • 17. 1,3,4-Oxadiazole/thiadiazole and 1,2,4-triazole derivatives of biphenyl-4-yloxy acetic acid: synthesis and preliminary evaluation of biological properties.
    Kumar H; Javed SA; Khan SA; Amir M
    Eur J Med Chem; 2008 Dec; 43(12):2688-98. PubMed ID: 18395299
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Investigations of new pyridazinone derivatives for the synthesis of potent analgesic and anti-inflammatory compounds with cyclooxygenase inhibitory activity.
    Okçelik B; Unlü S; Banoglu E; Küpeli E; Yeşilada E; Sahin MF
    Arch Pharm (Weinheim); 2003 Sep; 336(9):406-12. PubMed ID: 14528488
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and structure-activity relationship of a new series of COX-2 selective inhibitors: 1,5-diarylimidazoles.
    Almansa C; Alfón J; de Arriba AF; Cavalcanti FL; Escamilla I; Gómez LA; Miralles A; Soliva R; Bartrolí J; Carceller E; Merlos M; García-Rafanell J
    J Med Chem; 2003 Jul; 46(16):3463-75. PubMed ID: 12877584
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design and synthesis of 2-phenoxynicotinic acid hydrazides as anti-inflammatory and analgesic agents.
    Moradi A; Navidpour L; Amini M; Sadeghian H; Shadnia H; Firouzi O; Miri R; Ebrahimi SE; Abdollahi M; Zahmatkesh MH; Shafiee A
    Arch Pharm (Weinheim); 2010 Sep; 343(9):509-18. PubMed ID: 20806271
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 27.