297 related articles for article (PubMed ID: 18789686)
1. Synthesis and biological activity of anticoccidial agents: 5,6-diarylimidazo[2,1-b][1,3]thiazoles.
Scribner A; Meitz S; Fisher M; Wyvratt M; Leavitt P; Liberator P; Gurnett A; Brown C; Mathew J; Thompson D; Schmatz D; Biftu T
Bioorg Med Chem Lett; 2008 Oct; 18(19):5263-7. PubMed ID: 18789686
[TBL] [Abstract][Full Text] [Related]
2. Synthesis and biological activity of anticoccidial agents: 2,3-diarylindoles.
Scribner A; Moore JA; Ouvry G; Fisher M; Wyvratt M; Leavitt P; Liberator P; Gurnett A; Brown C; Mathew J; Thompson D; Schmatz D; Biftu T
Bioorg Med Chem Lett; 2009 Mar; 19(5):1517-21. PubMed ID: 19195883
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and biological activity of imidazopyridine anticoccidial agents: part I.
Scribner A; Dennis R; Hong J; Lee S; McIntyre D; Perrey D; Feng D; Fisher M; Wyvratt M; Leavitt P; Liberator P; Gurnett A; Brown C; Mathew J; Thompson D; Schmatz D; Biftu T
Eur J Med Chem; 2007; 42(11-12):1334-57. PubMed ID: 17433505
[TBL] [Abstract][Full Text] [Related]
4. N-alkyl-4-piperidinyl-2,3-diarylpyrrole derivatives with heterocyclic substitutions as potent and broad spectrum anticoccidial agents.
Liang GB; Qian X; Feng D; Fisher M; Crumley T; Darkin-Rattray SJ; Dulski PM; Gurnett A; Leavitt PS; Liberator PA; Misura AS; Samaras S; Tamas T; Schmatz DM; Wyvratt M; Biftu T
Bioorg Med Chem Lett; 2008 Mar; 18(6):2019-22. PubMed ID: 18276140
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and biological activity of imidazopyridine anticoccidial agents: Part II.
Scribner A; Dennis R; Lee S; Ouvry G; Perrey D; Fisher M; Wyvratt M; Leavitt P; Liberator P; Gurnett A; Brown C; Mathew J; Thompson D; Schmatz D; Biftu T
Eur J Med Chem; 2008 Jun; 43(6):1123-51. PubMed ID: 17981367
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and SAR of 2-(4-fluorophenyl)-3-pyrimidin-4-ylimidazo[1,2-a]pyridine derivatives as anticoccidial agents.
Feng D; Fisher M; Liang GB; Qian X; Brown C; Gurnett A; Leavitt PS; Liberator PA; Mathew J; Misura A; Samaras S; Tamas T; Schmatz DM; Wyvratt M; Biftu T
Bioorg Med Chem Lett; 2006 Dec; 16(23):5978-81. PubMed ID: 17000105
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and SAR studies of potent imidazopyridine anticoccidial agents.
Liang GB; Qian X; Feng D; Fisher M; Brown CM; Gurnett A; Leavitt PS; Liberator PA; Misura AS; Tamas T; Schmatz DM; Wyvratt M; Biftu T
Bioorg Med Chem Lett; 2007 Jul; 17(13):3558-61. PubMed ID: 17475489
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and SAR of 2,3-diarylpyrrole inhibitors of parasite cGMP-dependent protein kinase as novel anticoccidial agents.
Biftu T; Feng D; Ponpipom M; Girotra N; Liang GB; Qian X; Bugianesi R; Simeone J; Chang L; Gurnett A; Liberator P; Dulski P; Leavitt PS; Crumley T; Misura A; Murphy T; Rattray S; Samaras S; Tamas T; Mathew J; Brown C; Thompson D; Schmatz D; Fisher M; Wyvratt M
Bioorg Med Chem Lett; 2005 Jul; 15(13):3296-301. PubMed ID: 15922595
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and SAR studies of diarylpyrrole anticoccidial agents.
Qian X; Liang GB; Feng D; Fisher M; Crumley T; Rattray S; Dulski PM; Gurnett A; Leavitt PS; Liberator PA; Misura AS; Samaras S; Tamas T; Schmatz DM; Wyvratt M; Biftu T
Bioorg Med Chem Lett; 2006 May; 16(10):2817-21. PubMed ID: 16517161
[TBL] [Abstract][Full Text] [Related]
10. Hydroxylated N-alkyl-4-piperidinyl-2,3-diarylpyrrole derivatives as potent broad-spectrum anticoccidial agents.
Liang GB; Qian X; Biftu T; Feng D; Fisher M; Crumley T; Darkin-Rattray SJ; Dulski PM; Gurnett A; Leavitt PS; Liberator PA; Misura AS; Samaras S; Tamas T; Schmatz DM; Wyvratt M
Bioorg Med Chem Lett; 2005 Oct; 15(20):4570-3. PubMed ID: 16087336
[TBL] [Abstract][Full Text] [Related]
11. Anticoccidial kinase inhibitors: identification of protein kinase targets secondary to cGMP-dependent protein kinase.
Donald RG; Zhong T; Wiersma H; Nare B; Yao D; Lee A; Allocco J; Liberator PA
Mol Biochem Parasitol; 2006 Sep; 149(1):86-98. PubMed ID: 16765465
[TBL] [Abstract][Full Text] [Related]
12. Novel thienopyrimidine and thiazolopyrimidine kinase inhibitors with activity against Tie-2 in vitro and in vivo.
Luke RW; Ballard P; Buttar D; Campbell L; Curwen J; Emery SC; Griffen AM; Hassall L; Hayter BR; Jones CD; McCoull W; Mellor M; Swain ML; Tucker JA
Bioorg Med Chem Lett; 2009 Dec; 19(23):6670-4. PubMed ID: 19854647
[TBL] [Abstract][Full Text] [Related]
13. New antitumor imidazo[2,1-b]thiazole guanylhydrazones and analogues.
Andreani A; Burnelli S; Granaiola M; Leoni A; Locatelli A; Morigi R; Rambaldi M; Varoli L; Calonghi N; Cappadone C; Farruggia G; Zini M; Stefanelli C; Masotti L; Radin NS; Shoemaker RH
J Med Chem; 2008 Feb; 51(4):809-16. PubMed ID: 18251494
[TBL] [Abstract][Full Text] [Related]
14. Synthesis and chemiluminescent high throughput screening for inhibition of acetylcholinesterase activity by imidazo[2,1-b]thiazole derivatives.
Andreani A; Granaiola M; Guardigli M; Leoni A; Locatelli A; Morigi R; Rambaldi M; Roda A
Eur J Med Chem; 2005 Dec; 40(12):1331-4. PubMed ID: 16129518
[TBL] [Abstract][Full Text] [Related]
15. Synthesis, initial SAR and biological evaluation of 1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-4-amine derived inhibitors of IkappaB kinase.
Kempson J; Guo J; Das J; Moquin RV; Spergel SH; Watterson SH; Langevine CM; Dyckman AJ; Pattoli M; Burke JR; Yang X; Gillooly KM; McIntyre KW; Chen L; Dodd JH; McKinnon M; Barrish JC; Pitts WJ
Bioorg Med Chem Lett; 2009 May; 19(10):2646-9. PubMed ID: 19376699
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and SAR studies of very potent imidazopyridine antiprotozoal agents.
Biftu T; Feng D; Fisher M; Liang GB; Qian X; Scribner A; Dennis R; Lee S; Liberator PA; Brown C; Gurnett A; Leavitt PS; Thompson D; Mathew J; Misura A; Samaras S; Tamas T; Sina JF; McNulty KA; McKnight CG; Schmatz DM; Wyvratt M
Bioorg Med Chem Lett; 2006 May; 16(9):2479-83. PubMed ID: 16464591
[TBL] [Abstract][Full Text] [Related]
17. Potent 2-[(pyrimidin-4-yl)amine}-1,3-thiazole-5-carbonitrile-based inhibitors of VEGFR-2 (KDR) kinase.
Sisko JT; Tucker TJ; Bilodeau MT; Buser CA; Ciecko PA; Coll KE; Fernandes C; Gibbs JB; Koester TJ; Kohl N; Lynch JJ; Mao X; McLoughlin D; Miller-Stein CM; Rodman LD; Rickert KW; Sepp-Lorenzino L; Shipman JM; Thomas KA; Wong BK; Hartman GD
Bioorg Med Chem Lett; 2006 Mar; 16(5):1146-50. PubMed ID: 16368234
[TBL] [Abstract][Full Text] [Related]
18. Isolation, structure, and coccidiostat activity of coccidiostatin A.
Jayasuriya H; Guan Z; Dombrowski AW; Bills GF; Polishook JD; Jenkins RG; Koch L; Crumley T; Tamas T; Dubois M; Misura A; Darkin-Rattray SJ; Gregory L; Singh SB
J Nat Prod; 2007 Aug; 70(8):1364-7. PubMed ID: 17636951
[TBL] [Abstract][Full Text] [Related]
19. Isothiazolidinone inhibitors of PTP1B containing imidazoles and imidazolines.
Douty B; Wayland B; Ala PJ; Bower MJ; Pruitt J; Bostrom L; Wei M; Klabe R; Gonneville L; Wynn R; Burn TC; Liu PC; Combs AP; Yue EW
Bioorg Med Chem Lett; 2008 Jan; 18(1):66-71. PubMed ID: 18037290
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and antihypertensive activity of imidazo[2,1-b]-thiazoles bearing a 2,6-dichlorophenyl group.
Andreani A; Rambaldi M; Locatelli A; Cristoni A; Malandrino S; Pifferi G
Acta Pharm Nord; 1992; 4(2):93-6. PubMed ID: 1388775
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]