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4. Highly potent first examples of dual aromatase-steroid sulfatase inhibitors based on a biphenyl template. Woo LW; Jackson T; Putey A; Cozier G; Leonard P; Acharya KR; Chander SK; Purohit A; Reed MJ; Potter BV J Med Chem; 2010 Mar; 53(5):2155-70. PubMed ID: 20148564 [TBL] [Abstract][Full Text] [Related]
5. Chiral aromatase and dual aromatase-steroid sulfatase inhibitors from the letrozole template: synthesis, absolute configuration, and in vitro activity. Wood PM; Woo LW; Labrosse JR; Trusselle MN; Abbate S; Longhi G; Castiglioni E; Lebon F; Purohit A; Reed MJ; Potter BV J Med Chem; 2008 Jul; 51(14):4226-38. PubMed ID: 18590272 [TBL] [Abstract][Full Text] [Related]
6. Dual aromatase-sulfatase inhibitors based on the anastrozole template: synthesis, in vitro SAR, molecular modelling and in vivo activity. Jackson T; Woo LW; Trusselle MN; Chander SK; Purohit A; Reed MJ; Potter BV Org Biomol Chem; 2007 Sep; 5(18):2940-52. PubMed ID: 17728860 [TBL] [Abstract][Full Text] [Related]
7. Aromatase and dual aromatase-steroid sulfatase inhibitors from the letrozole and vorozole templates. Wood PM; Woo LW; Thomas MP; Mahon MF; Purohit A; Potter BV ChemMedChem; 2011 Aug; 6(8):1423-38. PubMed ID: 21608133 [TBL] [Abstract][Full Text] [Related]
8. Synthesis and structure-activity relationship studies of derivatives of the dual aromatase-sulfatase inhibitor 4-{[(4-cyanophenyl)(4H-1,2,4-triazol-4-yl)amino]methyl}phenyl sulfamate. Woo LW; Wood PM; Bubert C; Thomas MP; Purohit A; Potter BV ChemMedChem; 2013 May; 8(5):779-99. PubMed ID: 23495205 [TBL] [Abstract][Full Text] [Related]
9. A letrozole-based dual aromatase-sulphatase inhibitor with in vivo activity. Wood PM; Woo LW; Humphreys A; Chander SK; Purohit A; Reed MJ; Potter BV J Steroid Biochem Mol Biol; 2005 Feb; 94(1-3):123-30. PubMed ID: 15862957 [TBL] [Abstract][Full Text] [Related]
10. First crystal structures of human carbonic anhydrase II in complex with dual aromatase-steroid sulfatase inhibitors. Lloyd MD; Thiyagarajan N; Ho YT; Woo LW; Sutcliffe OB; Purohit A; Reed MJ; Acharya KR; Potter BV Biochemistry; 2005 May; 44(18):6858-66. PubMed ID: 15865431 [TBL] [Abstract][Full Text] [Related]
11. Dual aromatase-sulfatase inhibitors based on the anastrozole template: synthesis, in vitro SAR, molecular modelling and in vivo activity. Jackson T; Woo LW; Trusselle MN; Chander SK; Purohit A; Reed MJ; Potter BV Org Biomol Chem; 2007 Oct; 5(20):2940-52. PubMed ID: 17972413 [TBL] [Abstract][Full Text] [Related]
12. Design and synthesis of carbon-11-labeled dual aromatase-steroid sulfatase inhibitors as new potential PET agents for imaging of aromatase and steroid sulfatase expression in breast cancer. Wang M; Mickens J; Gao M; Miller KD; Sledge GW; Hutchins GD; Zheng QH Steroids; 2009 Nov; 74(12):896-905. PubMed ID: 19559719 [TBL] [Abstract][Full Text] [Related]
13. A new therapeutic strategy against hormone-dependent breast cancer: the preclinical development of a dual aromatase and sulfatase inhibitor. Foster PA; Chander SK; Newman SP; Woo LW; Sutcliffe OB; Bubert C; Zhou D; Chen S; Potter BV; Reed MJ; Purohit A Clin Cancer Res; 2008 Oct; 14(20):6469-77. PubMed ID: 18927286 [TBL] [Abstract][Full Text] [Related]
14. Non-steroidal aromatase inhibitors based on a biphenyl scaffold: synthesis, in vitro SAR, and molecular modelling. Jackson T; Woo LW; Trusselle MN; Purohit A; Reed MJ; Potter BV ChemMedChem; 2008 Apr; 3(4):603-18. PubMed ID: 18236493 [TBL] [Abstract][Full Text] [Related]
15. Synthesis and structure-activity relationship of 1- and 2-substituted-1,2,3-triazole letrozole-based analogues as aromatase inhibitors. Doiron J; Soultan AH; Richard R; Touré MM; Picot N; Richard R; Cuperlović-Culf M; Robichaud GA; Touaibia M Eur J Med Chem; 2011 Sep; 46(9):4010-24. PubMed ID: 21703734 [TBL] [Abstract][Full Text] [Related]
17. Synthesis, in vitro and in vivo activity of benzophenone-based inhibitors of steroid sulfatase. Hejaz HA; Woo LW; Purohit A; Reed MJ; Potter BV Bioorg Med Chem; 2004 May; 12(10):2759-72. PubMed ID: 15110857 [TBL] [Abstract][Full Text] [Related]
18. Steroidal and nonsteroidal sulfamates as potent inhibitors of steroid sulfatase. Woo LW; Howarth NM; Purohit A; Hejaz HA; Reed MJ; Potter BV J Med Chem; 1998 Mar; 41(7):1068-83. PubMed ID: 9544207 [TBL] [Abstract][Full Text] [Related]
19. Solid-phase parallel synthesis of 17alpha-substituted estradiol sulfamate and phenol libraries using the multidetachable sulfamate linker. Ciobanu LC; Poirier D J Comb Chem; 2003; 5(4):429-40. PubMed ID: 12857111 [TBL] [Abstract][Full Text] [Related]
20. Estradiol dimers as a new class of steroid sulfatase reversible inhibitors. Fournier D; Poirier D Bioorg Med Chem Lett; 2009 Feb; 19(3):693-6. PubMed ID: 19128967 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]