186 related articles for article (PubMed ID: 19053748)
21. Cocaine and 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid ester and amide analogues. New high-affinity and selective compounds for the dopamine transporter.
Carroll FI; Kotian P; Dehghani A; Gray JL; Kuzemko MA; Parham KA; Abraham P; Lewin AH; Boja JW; Kuhar MJ
J Med Chem; 1995 Jan; 38(2):379-88. PubMed ID: 7830281
[TBL] [Abstract][Full Text] [Related]
22. Structure-activity relationship comparison of (S)-2beta-substituted 3alpha-(bis[4-fluorophenyl]methoxy)tropanes and (R)-2beta-substituted 3beta-(3,4-dichlorophenyl)tropanes at the dopamine transporter.
Zou MF; Kopajtic T; Katz JL; Newman AH
J Med Chem; 2003 Jul; 46(14):2908-16. PubMed ID: 12825932
[TBL] [Abstract][Full Text] [Related]
23. Synthesis and ligand binding of nortropane derivatives: N-substituted 2beta-carbomethoxy-3beta-(4'-iodophenyl)nortropane and N-(3-iodoprop-(2E)-enyl)-2beta-carbomethoxy-3beta-(3',4'-disubstituted phenyl)nortropane. New high-affinity and selective compounds for the dopamine transporter.
Emond P; Garreau L; Chalon S; Boazi M; Caillet M; Bricard J; Frangin Y; Mauclaire L; Besnard JC; Guilloteau D
J Med Chem; 1997 Apr; 40(9):1366-72. PubMed ID: 9135033
[TBL] [Abstract][Full Text] [Related]
24. Synthesis and transporter binding properties of 2,3-diphenyltropane stereoisomers. Comparison to 3beta-phenyltropane-2beta-carboxylic acid esters.
Chang AC; Burgess JP; Mascarella SW; Abraham P; Kuhar MJ; Carroll FI
J Med Chem; 1997 Apr; 40(8):1247-51. PubMed ID: 9111298
[TBL] [Abstract][Full Text] [Related]
25. Synthesis and biological evaluation of 6/7-exo-methyl-3beta-(4-iodo)phenyltropane-2beta-carboxylic acid methyl esters.
Airaksinen AJ; Huotari M; Shvetsov A; Vainiotalo P; Männisto PT; Tuomisto L; Bergström KA; Vepsäläinen J
Eur J Med Chem; 2005 Mar; 40(3):299-304. PubMed ID: 15725499
[TBL] [Abstract][Full Text] [Related]
26. Synthesis, monoamine transporter binding, properties, and functional monoamine uptake activity of 3beta-[4-methylphenyl and 4-chlorophenyl]-2 beta-[5-(substituted phenyl)thiazol-2-yl]tropanes.
Gong PK; Blough BE; Brieaddy LE; Huang X; Kuhar MJ; Navarro HA; Carroll FI
J Med Chem; 2007 Jul; 50(15):3686-95. PubMed ID: 17602602
[TBL] [Abstract][Full Text] [Related]
27. Rhodamine-labeled 2beta-carbomethoxy-3beta-(3,4-dichlorophenyl)tropane analogues as high-affinity fluorescent probes for the dopamine transporter.
Cha JH; Zou MF; Adkins EM; Rasmussen SG; Loland CJ; Schoenenberger B; Gether U; Newman AH
J Med Chem; 2005 Dec; 48(24):7513-6. PubMed ID: 16302792
[TBL] [Abstract][Full Text] [Related]
28. Structure-activity relationships at monoamine transporters for a series of N-substituted 3alpha-(bis[4-fluorophenyl]methoxy)tropanes: comparative molecular field analysis, synthesis, and pharmacological evaluation.
Kulkarni SS; Grundt P; Kopajtic T; Katz JL; Newman AH
J Med Chem; 2004 Jun; 47(13):3388-98. PubMed ID: 15189035
[TBL] [Abstract][Full Text] [Related]
29. Biaryl analogues of conformationally constrained tricyclic tropanes as potent and selective norepinephrine reuptake inhibitors: synthesis and evaluation of their uptake inhibition at monoamine transporter sites.
Zhou J; Zhang A; Kläss T; Johnson KM; Wang CZ; Ye YP; Kozikowski AP
J Med Chem; 2003 May; 46(10):1997-2007. PubMed ID: 12723962
[TBL] [Abstract][Full Text] [Related]
30. N-substituted analogs of 2 beta-carbomethoxy-3 beta- (4'-iodophenyl)tropane (beta-CIT) with selective affinity to dopamine or serotonin transporters in rat forebrain.
Neumeyer JL; Tamagnan G; Wang S; Gao Y; Milius RA; Kula NS; Baldessarini RJ
J Med Chem; 1996 Jan; 39(2):543-8. PubMed ID: 8558525
[TBL] [Abstract][Full Text] [Related]
31. Synthesis and monoamine transporter affinity of new 2beta-carbomethoxy-3beta-[4-(substituted thiophenyl)]phenyltropanes: discovery of a selective SERT antagonist with picomolar potency.
Tamagnan G; Alagille D; Fu X; Kula NS; Baldessarini RJ; Innis RB; Baldwin RM
Bioorg Med Chem Lett; 2005 Feb; 15(4):1131-3. PubMed ID: 15686927
[TBL] [Abstract][Full Text] [Related]
32. Secondary amine analogues of 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid esters and N-norcocaine exhibit enhanced affinity for serotonin and norepinephrine transporters.
Boja JW; Kuhar MJ; Kopajtic T; Yang E; Abraham P; Lewin AH; Carroll FI
J Med Chem; 1994 Apr; 37(8):1220-3. PubMed ID: 8164265
[TBL] [Abstract][Full Text] [Related]
33. Structure-activity relationships at monoamine transporters and muscarinic receptors for N-substituted-3alpha-(3'-chloro-, 4'-chloro-, and 4',4''-dichloro-substituted-diphenyl)methoxytropanes.
Newman AH; Robarge MJ; Howard IM; Wittkopp SL; George C; Kopajtic T; Izenwasser S; Katz JL
J Med Chem; 2001 Feb; 44(4):633-40. PubMed ID: 11170654
[TBL] [Abstract][Full Text] [Related]
34. Effects of combined dopamine and serotonin transporter inhibitors on cocaine self-administration in rhesus monkeys.
Howell LL; Carroll FI; Votaw JR; Goodman MM; Kimmel HL
J Pharmacol Exp Ther; 2007 Feb; 320(2):757-65. PubMed ID: 17105829
[TBL] [Abstract][Full Text] [Related]
35. Synthesis of 6- and 7- hydroxy-8-azabicyclo[3.2.1]octanes and their binding affinity for the dopamine and serotonin transporters.
Meltzer PC; Wang B; Chen Z; Blundell P; Jayaraman M; Gonzalez MD; George C; Madras BK
J Med Chem; 2001 Aug; 44(16):2619-35. PubMed ID: 11472216
[TBL] [Abstract][Full Text] [Related]
36. Inhibitor mechanisms in the S1 binding site of the dopamine transporter defined by multi-site molecular tethering of photoactive cocaine analogs.
Krout D; Pramod AB; Dahal RA; Tomlinson MJ; Sharma B; Foster JD; Zou MF; Boatang C; Newman AH; Lever JR; Vaughan RA; Henry LK
Biochem Pharmacol; 2017 Oct; 142():204-215. PubMed ID: 28734777
[TBL] [Abstract][Full Text] [Related]
37. An extended study of dimeric phenyl tropanes.
Nielsen S; Pedersen CM; Hansen SG; Petersen MD; Sinning S; Wiborg O; Jensen HH; Bols M
Bioorg Med Chem; 2009 Jul; 17(14):4900-9. PubMed ID: 19560930
[TBL] [Abstract][Full Text] [Related]
38. 3alpha-(4-Substituted phenyl)nortropane-2beta-carboxylic acid methyl esters show selective binding at the norepinephrine transporter.
Blough BE; Holmquist CR; Abraham P; Kuhar MJ; Carroll FI
Bioorg Med Chem Lett; 2000 Nov; 10(21):2445-7. PubMed ID: 11078197
[TBL] [Abstract][Full Text] [Related]
39. Synthesis and monoamine uptake inhibition of conformationally constrained 2beta-carbomethoxy-3beta-phenyl tropanes.
Riss PJ; Hummerich R; Schloss P
Org Biomol Chem; 2009 Jul; 7(13):2688-98. PubMed ID: 19532984
[TBL] [Abstract][Full Text] [Related]
40. 3'-Chloro-3 alpha-(diphenylmethoxy)tropane but not 4'-chloro-3 alpha-(diphenylmethoxy)tropane produces a cocaine-like behavioral profile.
Kline RH; Izenwasser S; Katz JL; Joseph DB; Bowen WD; Newman AH
J Med Chem; 1997 Mar; 40(6):851-7. PubMed ID: 9083473
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]