These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

201 related articles for article (PubMed ID: 19171802)

  • 1. Synthesis and antimalarial activities of cyclen 4-aminoquinoline analogs.
    Khan MO; Levi MS; Tekwani BL; Khan SI; Kimura E; Borne RF
    Antimicrob Agents Chemother; 2009 Apr; 53(4):1320-4. PubMed ID: 19171802
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Novel 4-aminoquinoline analogs highly active against the blood and sexual stages of Plasmodium in vivo and in vitro.
    Sáenz FE; Mutka T; Udenze K; Oduola AM; Kyle DE
    Antimicrob Agents Chemother; 2012 Sep; 56(9):4685-92. PubMed ID: 22710117
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis, β-hematin inhibition studies and antimalarial evaluation of dehydroxy isotebuquine derivatives against Plasmodium berghei.
    Romero AH; Acosta ME; Gamboa N; Charris JE; Salazar J; López SE
    Bioorg Med Chem; 2015 Aug; 23(15):4755-4762. PubMed ID: 26081761
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Antimalarials with Benzothiophene Moieties as Aminoquinoline Partners.
    Konstantinović J; Videnović M; Srbljanović J; Djurković-Djaković O; Bogojević K; Sciotti R; Šolaja B
    Molecules; 2017 Feb; 22(3):. PubMed ID: 28245583
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and bioevaluation of novel 4-aminoquinoline-tetrazole derivatives as potent antimalarial agents.
    Pandey S; Agarwal P; Srivastava K; Rajakumar S; Puri SK; Verma P; Saxena JK; Sharma A; Lal J; Chauhan PM
    Eur J Med Chem; 2013 Aug; 66():69-81. PubMed ID: 23792317
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and antimalarial activity of side chain modified 4-aminoquinoline derivatives.
    Solomon VR; Haq W; Srivastava K; Puri SK; Katti SB
    J Med Chem; 2007 Jan; 50(2):394-8. PubMed ID: 17228883
    [TBL] [Abstract][Full Text] [Related]  

  • 7. 4-aminoquinoline-triazine-based hybrids with improved in vitro antimalarial activity against CQ-sensitive and CQ-resistant strains of Plasmodium falciparum.
    Manohar S; Khan SI; Rawat DS
    Chem Biol Drug Des; 2013 May; 81(5):625-30. PubMed ID: 23331618
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Antimalarial activity of novel 5-aryl-8-aminoquinoline derivatives.
    Shiraki H; Kozar MP; Melendez V; Hudson TH; Ohrt C; Magill AJ; Lin AJ
    J Med Chem; 2011 Jan; 54(1):131-42. PubMed ID: 21141892
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Antimalarial activity and mechanisms of action of two novel 4-aminoquinolines against chloroquine-resistant parasites.
    Aguiar AC; Santos Rde M; Figueiredo FJ; Cortopassi WA; Pimentel AS; França TC; Meneghetti MR; Krettli AU
    PLoS One; 2012; 7(5):e37259. PubMed ID: 22649514
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Novel conjugated quinoline-indoles compromise Plasmodium falciparum mitochondrial function and show promising antimalarial activity.
    Teguh SC; Klonis N; Duffy S; Lucantoni L; Avery VM; Hutton CA; Baell JB; Tilley L
    J Med Chem; 2013 Aug; 56(15):6200-15. PubMed ID: 23837878
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Bisquinolines. 2. Antimalarial N,N-bis(7-chloroquinolin-4-yl)heteroalkanediamines.
    Vennerstrom JL; Ager AL; Dorn A; Andersen SL; Gerena L; Ridley RG; Milhous WK
    J Med Chem; 1998 Oct; 41(22):4360-4. PubMed ID: 9784111
    [TBL] [Abstract][Full Text] [Related]  

  • 12. 4-Aminoquinoline derivatives: Synthesis, in vitro and in vivo antiplasmodial activity against chloroquine-resistant parasites.
    Singh S; Agarwal D; Sharma K; Sharma M; Nielsen MA; Alifrangis M; Singh AK; Gupta RD; Awasthi SK
    Eur J Med Chem; 2016 Oct; 122():394-407. PubMed ID: 27394399
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Optimization of 4-aminoquinoline/clotrimazole-based hybrid antimalarials: further structure-activity relationships, in vivo studies, and preliminary toxicity profiling.
    Gemma S; Camodeca C; Sanna Coccone S; Joshi BP; Bernetti M; Moretti V; Brogi S; Bonache de Marcos MC; Savini L; Taramelli D; Basilico N; Parapini S; Rottmann M; Brun R; Lamponi S; Caccia S; Guiso G; Summers RL; Martin RE; Saponara S; Gorelli B; Novellino E; Campiani G; Butini S
    J Med Chem; 2012 Aug; 55(15):6948-67. PubMed ID: 22783984
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and antimalarial activity in vitro and in vivo of a new ferrocene-chloroquine analogue.
    Biot C; Glorian G; Maciejewski LA; Brocard JS
    J Med Chem; 1997 Nov; 40(23):3715-8. PubMed ID: 9371235
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis, antimalarial, antileishmanial, antimicrobial, cytotoxicity, and methemoglobin (MetHB) formation activities of new 8-quinolinamines.
    Kaur K; Patel SR; Patil P; Jain M; Khan SI; Jacob MR; Tekwani BL; Jain R
    Bioorg Med Chem; 2007 Jan; 15(2):915-930. PubMed ID: 17084633
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Antiplasmodial activity of new 4-aminoquinoline derivatives against chloroquine resistant strain.
    Sinha M; Dola VR; Agarwal P; Srivastava K; Haq W; Puri SK; Katti SB
    Bioorg Med Chem; 2014 Jul; 22(14):3573-86. PubMed ID: 24906512
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Mapping antimalarial pharmacophores as a useful tool for the rapid discovery of drugs effective in vivo: design, construction, characterization, and pharmacology of metaquine.
    Dascombe MJ; Drew MG; Morris H; Wilairat P; Auparakkitanon S; Moule WA; Alizadeh-Shekalgourabi S; Evans PG; Lloyd M; Dyas AM; Carr P; Ismail FM
    J Med Chem; 2005 Aug; 48(17):5423-36. PubMed ID: 16107142
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis of chiral chloroquine and its analogues as antimalarial agents.
    Sinha M; Dola VR; Soni A; Agarwal P; Srivastava K; Haq W; Puri SK; Katti SB
    Bioorg Med Chem; 2014 Nov; 22(21):5950-60. PubMed ID: 25284252
    [TBL] [Abstract][Full Text] [Related]  

  • 19. 4-Aminoquinoline quinolizidinyl- and quinolizidinylalkyl-derivatives with antimalarial activity.
    Sparatore A; Basilico N; Parapini S; Romeo S; Novelli F; Sparatore F; Taramelli D
    Bioorg Med Chem; 2005 Sep; 13(18):5338-45. PubMed ID: 16054368
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis of ring-substituted 4-aminoquinolines and evaluation of their antimalarial activities.
    Madrid PB; Sherrill J; Liou AP; Weisman JL; Derisi JL; Guy RK
    Bioorg Med Chem Lett; 2005 Feb; 15(4):1015-8. PubMed ID: 15686903
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 11.