BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

435 related articles for article (PubMed ID: 19275709)

  • 61. Design, synthesis, biological evaluation, and computational studies of novel thiazolo-pyrazole hybrids as promising selective COX-2 inhibitors: Implementation of apoptotic genes expression for ulcerogenic liability assessment.
    Marzouk AA; Taher ES; Shaykoon MSA; Lan P; Abd-Allah WH; Aboregela AM; El-Behairy MF
    Bioorg Chem; 2021 Jun; 111():104883. PubMed ID: 33865053
    [TBL] [Abstract][Full Text] [Related]  

  • 62. Pyrazole-hydrazone derivatives as anti-inflammatory agents: Design, synthesis, biological evaluation, COX-1,2/5-LOX inhibition and docking study.
    Abdelgawad MA; Labib MB; Abdel-Latif M
    Bioorg Chem; 2017 Oct; 74():212-220. PubMed ID: 28865292
    [TBL] [Abstract][Full Text] [Related]  

  • 63. Novel N-substituted 5-aminosalicylamides as dual inhibitors of cyclooxygenase and 5-lipoxygenase enzymes: Synthesis, biological evaluation and docking study.
    El-Nagar MKS; Abdu-Allah HHM; Salem OIA; Kafafy AN; Farghaly HSM
    Bioorg Chem; 2018 Aug; 78():80-93. PubMed ID: 29550533
    [TBL] [Abstract][Full Text] [Related]  

  • 64. Synthesis, biological evaluation and docking study of maleimide derivatives bearing benzenesulfonamide as selective COX-2 inhibitors and anti-inflammatory agents.
    Firke SD; Bari SB
    Bioorg Med Chem; 2015 Sep; 23(17):5273-81. PubMed ID: 26277757
    [TBL] [Abstract][Full Text] [Related]  

  • 65. Synthesis, Cyclooxygenase-2 Inhibition, Anti-inflammatory Evaluation and Docking Study of Substituted-N-(3,4,5-trimethoxyphenyl)-benzo[d]oxazole Derivatives.
    Kaur A; Wakode S; Pathak DP; Sharma V; Shakya AK
    Med Chem; 2018; 14(7):660-673. PubMed ID: 29564981
    [TBL] [Abstract][Full Text] [Related]  

  • 66. A novel COX-2 inhibitor pyrazole derivative proven effective as an anti-inflammatory and analgesic drug.
    Mohy El-Din MM; Senbel AM; Bistawroos AA; El-Mallah A; Nour El-Din NA; Bekhit AA; Abd El Razik HA
    Basic Clin Pharmacol Toxicol; 2011 Apr; 108(4):263-73. PubMed ID: 21138530
    [TBL] [Abstract][Full Text] [Related]  

  • 67. Evaluation of anti-inflammatory, analgesic activities, and side effects of some pyrazole derivatives.
    Domiati S; El-Mallah A; Ghoneim A; Bekhit A; El Razik HA
    Inflammopharmacology; 2016 Aug; 24(4):163-72. PubMed ID: 27342269
    [TBL] [Abstract][Full Text] [Related]  

  • 68. New pyrazole derivatives possessing amino/methanesulphonyl pharmacophore with good gastric safety profile: Design, synthesis, cyclooxygenase inhibition, anti-inflammatory activity and histopathological studies.
    Abdellatif KRA; Abdelall EKA; Lamie PF; Labib MB; El-Nahaas ES; Abdelhakeem MM
    Bioorg Chem; 2020 Jan; 95():103540. PubMed ID: 31911297
    [TBL] [Abstract][Full Text] [Related]  

  • 69. Synthesis and biological evaluation of 4-arylphthalazones bearing benzenesulfonamide as anti-inflammatory and anti-cancer agents.
    Yaseen S; Ovais S; Bashir R; Rathore P; Samim M; Singh S; Nair V; Javed K
    Arch Pharm (Weinheim); 2013 Jun; 346(6):491-8. PubMed ID: 23670888
    [TBL] [Abstract][Full Text] [Related]  

  • 70. Synthesis and evaluation of pyrazolines bearing benzothiazole as anti-inflammatory agents.
    Kharbanda C; Alam MS; Hamid H; Javed K; Bano S; Dhulap A; Ali Y; Nazreen S; Haider S
    Bioorg Med Chem; 2014 Nov; 22(21):5804-12. PubMed ID: 25311566
    [TBL] [Abstract][Full Text] [Related]  

  • 71. Design, synthesis and biological evaluation of novel pyrazole sulfonamide derivatives as dual COX-2/5-LOX inhibitors.
    Gedawy EM; Kassab AE; El Kerdawy AM
    Eur J Med Chem; 2020 Mar; 189():112066. PubMed ID: 31982653
    [TBL] [Abstract][Full Text] [Related]  

  • 72. New
    Szczukowski Ł; Krzyżak E; Wiatrak B; Jawień P; Marciniak A; Kotynia A; Świątek P
    Int J Mol Sci; 2021 Oct; 22(20):. PubMed ID: 34681894
    [TBL] [Abstract][Full Text] [Related]  

  • 73. Synthesis, biological evaluation, docking study and ulcerogenicity profiling of some novel quinoline-2-carboxamides as dual COXs/LOX inhibitors endowed with anti-inflammatory activity.
    Abdelrahman MH; Youssif BGM; Abdelgawad MA; Abdelazeem AH; Ibrahim HM; Moustafa AEGA; Treamblu L; Bukhari SNA
    Eur J Med Chem; 2017 Feb; 127():972-985. PubMed ID: 27837994
    [TBL] [Abstract][Full Text] [Related]  

  • 74. New pyrazole derivatives: Synthesis, anti-inflammatory activity, cycloxygenase inhibition assay and evaluation of mPGES.
    Hassan GS; Abdel Rahman DE; Abdelmajeed EA; Refaey RH; Alaraby Salem M; Nissan YM
    Eur J Med Chem; 2019 Jun; 171():332-342. PubMed ID: 30928706
    [TBL] [Abstract][Full Text] [Related]  

  • 75. Design, synthesis, modeling studies and biological evaluation of thiazolidine derivatives containing pyrazole core as potential anti-diabetic PPAR-γ agonists and anti-inflammatory COX-2 selective inhibitors.
    Abdellatif KRA; Fadaly WAA; Kamel GM; Elshaier YAMM; El-Magd MA
    Bioorg Chem; 2019 Feb; 82():86-99. PubMed ID: 30278282
    [TBL] [Abstract][Full Text] [Related]  

  • 76. Non-acidic 1,3,4-trisubstituted-pyrazole derivatives as lonazolac analogs with promising COX-2 selectivity, anti-inflammatory activity and gastric safety profile.
    Abdellatif KRA; Fadaly WAA; Elshaier YAMM; Ali WAM; Kamel GM
    Bioorg Chem; 2018 Apr; 77():568-578. PubMed ID: 29475165
    [TBL] [Abstract][Full Text] [Related]  

  • 77. Synthesis and biological evaluation of some new 2-pyrazolines bearing benzene sulfonamide moiety as potential anti-inflammatory and anti-cancer agents.
    Bano S; Javed K; Ahmad S; Rathish IG; Singh S; Alam MS
    Eur J Med Chem; 2011 Dec; 46(12):5763-8. PubMed ID: 22019186
    [TBL] [Abstract][Full Text] [Related]  

  • 78. Design, synthesis, and anti-inflammatory evaluation of a series of novel amino acid-binding 1,5-diarylpyrazole derivatives.
    Li MH; Yin LL; Cai MJ; Zhang WY; Huang Y; Wang X; Zhu XZ; Shen JK
    Acta Pharmacol Sin; 2005 Jul; 26(7):865-72. PubMed ID: 15960895
    [TBL] [Abstract][Full Text] [Related]  

  • 79. Synthesis, molecular docking and anti-inflammatory screening of novel quinoline incorporated pyrazole derivatives using the Pfitzinger reaction II.
    El-Feky SA; Abd El-Samii ZK; Osman NA; Lashine J; Kamel MA; Thabet HKh
    Bioorg Chem; 2015 Feb; 58():104-16. PubMed ID: 25590381
    [TBL] [Abstract][Full Text] [Related]  

  • 80. Celecoxib analogs bearing benzofuran moiety as cyclooxygenase-2 inhibitors: design, synthesis and evaluation as potential anti-inflammatory agents.
    Hassan GS; Abou-Seri SM; Kamel G; Ali MM
    Eur J Med Chem; 2014 Apr; 76():482-93. PubMed ID: 24607877
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 22.