BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

129 related articles for article (PubMed ID: 19359182)

  • 1. Synthesis and evaluation of aryl-substituted diarylpropionitriles, selective ligands for estrogen receptor beta, as positron-emission tomographic imaging agents.
    Moon BS; Carlson KE; Katzenellenbogen JA; Choi TH; Chi DY; Kim JY; Cheon GJ; Koh HY; Lee KC; An G
    Bioorg Med Chem; 2009 May; 17(9):3479-88. PubMed ID: 19359182
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Estrogen receptor-beta potency-selective ligands: structure-activity relationship studies of diarylpropionitriles and their acetylene and polar analogues.
    Meyers MJ; Sun J; Carlson KE; Marriner GA; Katzenellenbogen BS; Katzenellenbogen JA
    J Med Chem; 2001 Nov; 44(24):4230-51. PubMed ID: 11708925
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Diarylpropionitrile (DPN) enantiomers: synthesis and evaluation of estrogen receptor β-selective ligands.
    Carroll VM; Jeyakumar M; Carlson KE; Katzenellenbogen JA
    J Med Chem; 2012 Jan; 55(1):528-37. PubMed ID: 22122563
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and biological evaluation of two agents for imaging estrogen receptor β by positron emission tomography: challenges in PET imaging of a low abundance target.
    Lee JH; Peters O; Lehmann L; Dence CS; Sharp TL; Carlson KE; Zhou D; Jeyakumar M; Welch MJ; Katzenellenbogen JA
    Nucl Med Biol; 2012 Nov; 39(8):1105-16. PubMed ID: 22749433
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis of an estrogen receptor beta-selective radioligand: 5-[18F]fluoro-(2R,3S)-2,3-bis(4-hydroxyphenyl)pentanenitrile and comparison of in vivo distribution with 16alpha-[18F]fluoro-17beta-estradiol.
    Yoo J; Dence CS; Sharp TL; Katzenellenbogen JA; Welch MJ
    J Med Chem; 2005 Oct; 48(20):6366-78. PubMed ID: 16190762
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Functional characterization of estrogen receptor subtypes, ERalpha and ERbeta, mediating vitellogenin production in the liver of rainbow trout.
    Leaños-Castañeda O; Van Der Kraak G
    Toxicol Appl Pharmacol; 2007 Oct; 224(2):116-25. PubMed ID: 17662327
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Computational Study of the Binding Modes of Diverse DPN Analogues on Estrogen Receptors (ER) and the Biological Evaluation of a New Potential Antiestrogenic Ligand.
    Martinez-Archundia M; García-Vázquez JB; Colin-Astudillo B; Bello M; Prestegui-Martel B; Chavez-Blanco A; Dueñas-González A; Fragoso-Vázquez MJ; Mendieta-Wejebe J; Abarca-Rojano E; Ordaz-Rosado D; García-Becerra R; Castillo-Bautista D; Correa Basurto J
    Anticancer Agents Med Chem; 2018; 18(11):1508-1520. PubMed ID: 29189179
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Evaluating the correlation of binding affinities between isothermal titration calorimetry and fragment molecular orbital method of estrogen receptor beta with diarylpropionitrile (DPN) or DPN derivatives.
    Handa C; Yamazaki Y; Yonekubo S; Furuya N; Momose T; Ozawa T; Furuishi T; Fukuzawa K; Yonemochi E
    J Steroid Biochem Mol Biol; 2022 Sep; 222():106152. PubMed ID: 35810932
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Estrogen receptor-beta agonist diarylpropionitrile: biological activities of R- and S-enantiomers on behavior and hormonal response to stress.
    Weiser MJ; Wu TJ; Handa RJ
    Endocrinology; 2009 Apr; 150(4):1817-25. PubMed ID: 19074580
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Molecular basis for the subtype discrimination of the estrogen receptor-beta-selective ligand, diarylpropionitrile.
    Sun J; Baudry J; Katzenellenbogen JA; Katzenellenbogen BS
    Mol Endocrinol; 2003 Feb; 17(2):247-58. PubMed ID: 12554752
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and characterization of hydrogen peroxide activated estrogen receptor beta ligands.
    Park H; McEachon JD; Pollock JA
    Bioorg Med Chem; 2019 May; 27(10):2075-2082. PubMed ID: 30967304
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Indazole estrogens: highly selective ligands for the estrogen receptor beta.
    De Angelis M; Stossi F; Carlson KA; Katzenellenbogen BS; Katzenellenbogen JA
    J Med Chem; 2005 Feb; 48(4):1132-44. PubMed ID: 15715479
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Fluorine-substituted cyclofenil derivatives as estrogen receptor ligands: synthesis and structure-affinity relationship study of potential positron emission tomography agents for imaging estrogen receptors in breast cancer.
    Seo JW; Comninos JS; Chi DY; Kim DW; Carlson KE; Katzenellenbogen JA
    J Med Chem; 2006 Apr; 49(8):2496-511. PubMed ID: 16610793
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Evaluation of ligand selectivity using reporter cell lines stably expressing estrogen receptor alpha or beta.
    Escande A; Pillon A; Servant N; Cravedi JP; Larrea F; Muhn P; Nicolas JC; Cavaillès V; Balaguer P
    Biochem Pharmacol; 2006 May; 71(10):1459-69. PubMed ID: 16554039
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Activities of estrogen receptor alpha- and beta-selective ligands at diverse estrogen responsive gene sites mediating transactivation or transrepression.
    Harrington WR; Sheng S; Barnett DH; Petz LN; Katzenellenbogen JA; Katzenellenbogen BS
    Mol Cell Endocrinol; 2003 Aug; 206(1-2):13-22. PubMed ID: 12943986
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Novel actions of estrogen receptor-beta on anxiety-related behaviors.
    Lund TD; Rovis T; Chung WC; Handa RJ
    Endocrinology; 2005 Feb; 146(2):797-807. PubMed ID: 15514081
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Structure-based design of estrogen receptor-beta selective ligands.
    Manas ES; Unwalla RJ; Xu ZB; Malamas MS; Miller CP; Harris HA; Hsiao C; Akopian T; Hum WT; Malakian K; Wolfrom S; Bapat A; Bhat RA; Stahl ML; Somers WS; Alvarez JC
    J Am Chem Soc; 2004 Nov; 126(46):15106-19. PubMed ID: 15548008
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Estradiol-induced desensitization of 5-HT1A receptor signaling in the paraventricular nucleus of the hypothalamus is independent of estrogen receptor-beta.
    Rossi DV; Dai Y; Thomas P; Carrasco GA; DonCarlos LL; Muma NA; Li Q
    Psychoneuroendocrinology; 2010 Aug; 35(7):1023-33. PubMed ID: 20138435
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Identification of ligands with bicyclic scaffolds provides insights into mechanisms of estrogen receptor subtype selectivity.
    Hsieh RW; Rajan SS; Sharma SK; Guo Y; DeSombre ER; Mrksich M; Greene GL
    J Biol Chem; 2006 Jun; 281(26):17909-19. PubMed ID: 16648639
    [TBL] [Abstract][Full Text] [Related]  

  • 20. A high-affinity subtype-selective fluorescent probe for estrogen receptor β imaging in living cells.
    Hu Z; Yang L; Ning W; Tang C; Meng Q; Zheng J; Dong C; Zhou HB
    Chem Commun (Camb); 2018 Apr; 54(31):3887-3890. PubMed ID: 29610818
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.