208 related articles for article (PubMed ID: 19402665)
1. Rhodamine inhibitors of P-glycoprotein: an amide/thioamide "switch" for ATPase activity.
Gannon MK; Holt JJ; Bennett SM; Wetzel BR; Loo TW; Bartlett MC; Clarke DM; Sawada GA; Higgins JW; Tombline G; Raub TJ; Detty MR
J Med Chem; 2009 May; 52(10):3328-41. PubMed ID: 19402665
[TBL] [Abstract][Full Text] [Related]
2. Thiorhodamines containing amide and thioamide functionality as inhibitors of the ATP-binding cassette drug transporter P-glycoprotein (ABCB1).
Orchard A; Schamerhorn GA; Calitree BD; Sawada GA; Loo TW; Claire Bartlett M; Clarke DM; Detty MR
Bioorg Med Chem; 2012 Jul; 20(14):4290-302. PubMed ID: 22727780
[TBL] [Abstract][Full Text] [Related]
3. Chalcogenopyrylium compounds as modulators of the ATP-binding cassette transporters P-glycoprotein (P-gp/ABCB1) and multidrug resistance protein 1 (MRP1/ABCC1).
Ebert SP; Wetzel B; Myette RL; Conseil G; Cole SP; Sawada GA; Loo TW; Bartlett MC; Clarke DM; Detty MR
J Med Chem; 2012 May; 55(10):4683-99. PubMed ID: 22533905
[TBL] [Abstract][Full Text] [Related]
4. Methanethiosulfonate derivatives of rhodamine and verapamil activate human P-glycoprotein at different sites.
Loo TW; Bartlett MC; Clarke DM
J Biol Chem; 2003 Dec; 278(50):50136-41. PubMed ID: 14522974
[TBL] [Abstract][Full Text] [Related]
5. Chalcogenopyrylium dyes as inhibitors/modulators of P-glycoprotein in multidrug-resistant cells.
Sawada GA; Raub TJ; William Higgins J; Brennan NK; Moore TM; Tombline G; Detty MR
Bioorg Med Chem; 2008 Nov; 16(22):9745-56. PubMed ID: 18849167
[TBL] [Abstract][Full Text] [Related]
6. Phosphorylation site mutations in the human multidrug transporter modulate its drug-stimulated ATPase activity.
Szabó K; Bakos E; Welker E; Müller M; Goodfellow HR; Higgins CF; Váradi A; Sarkadi B
J Biol Chem; 1997 Sep; 272(37):23165-71. PubMed ID: 9287320
[TBL] [Abstract][Full Text] [Related]
7. Efficiency of P-glycoprotein-mediated exclusion of rhodamine dyes from multidrug-resistant cells is determined by their passive transmembrane movement rate.
Eytan GD; Regev R; Oren G; Hurwitz CD; Assaraf YG
Eur J Biochem; 1997 Aug; 248(1):104-12. PubMed ID: 9310367
[TBL] [Abstract][Full Text] [Related]
8. Interaction of the P-glycoprotein multidrug transporter (MDR1) with high affinity peptide chemosensitizers in isolated membranes, reconstituted systems, and intact cells.
Sharom FJ; Yu X; Lu P; Liu R; Chu JW; Szabó K; Müller M; Hose CD; Monks A; Váradi A; Seprôdi J; Sarkadi B
Biochem Pharmacol; 1999 Aug; 58(4):571-86. PubMed ID: 10413294
[TBL] [Abstract][Full Text] [Related]
9. Phorbol 12-myristate 13-acetate inhibits P-glycoprotein-mediated efflux of digoxin in MDCKII-MDR1 and Caco-2 cell monolayer models.
Li YH; Bi HC; Huang L; Jin J; Zhong GP; Zhou XN; Huang M
Acta Pharmacol Sin; 2014 Feb; 35(2):283-91. PubMed ID: 24362330
[TBL] [Abstract][Full Text] [Related]
10. Competitive and non-competitive inhibition of the multidrug-resistance-associated P-glycoprotein ATPase--further experimental evidence for a multisite model.
Garrigos M; Mir LM; Orlowski S
Eur J Biochem; 1997 Mar; 244(2):664-73. PubMed ID: 9119038
[TBL] [Abstract][Full Text] [Related]
11. Delineating the contribution of secretory transporters in the efflux of etoposide using Madin-Darby canine kidney (MDCK) cells overexpressing P-glycoprotein (Pgp), multidrug resistance-associated protein (MRP1), and canalicular multispecific organic anion transporter (cMOAT).
Guo A; Marinaro W; Hu P; Sinko PJ
Drug Metab Dispos; 2002 Apr; 30(4):457-63. PubMed ID: 11901101
[TBL] [Abstract][Full Text] [Related]
12. Celastraceae sesquiterpenes as a new class of modulators that bind specifically to human P-glycoprotein and reverse cellular multidrug resistance.
Muñoz-Martínez F; Lu P; Cortés-Selva F; Pérez-Victoria JM; Jiménez IA; Ravelo AG; Sharom FJ; Gamarro F; Castanys S
Cancer Res; 2004 Oct; 64(19):7130-8. PubMed ID: 15466210
[TBL] [Abstract][Full Text] [Related]
13. P-glycoprotein substrates and antagonists cluster into two distinct groups.
Scala S; Akhmed N; Rao US; Paull K; Lan LB; Dickstein B; Lee JS; Elgemeie GH; Stein WD; Bates SE
Mol Pharmacol; 1997 Jun; 51(6):1024-33. PubMed ID: 9187269
[TBL] [Abstract][Full Text] [Related]
14. Caffeic Acid Attenuates Multi-Drug Resistance in Cancer Cells by Inhibiting Efflux Function of Human P-glycoprotein.
Teng YN; Wang CCN; Liao WC; Lan YH; Hung CC
Molecules; 2020 Jan; 25(2):. PubMed ID: 31936160
[No Abstract] [Full Text] [Related]
15. Role of P-glycoprotein in the intestinal absorption of tanshinone IIA, a major active ingredient in the root of Salvia miltiorrhiza Bunge.
Yu XY; Lin SG; Zhou ZW; Chen X; Liang J; Liu PQ; Duan W; Chowbay B; Wen JY; Li CG; Zhou SF
Curr Drug Metab; 2007 May; 8(4):325-40. PubMed ID: 17504222
[TBL] [Abstract][Full Text] [Related]
16. Nonionic surfactants increase digoxin absorption in Caco-2 and MDCKII MDR1 cells: Impact on P-glycoprotein inhibition, barrier function, and repeated cellular exposure.
Al-Ali AAA; Steffansen B; Holm R; Nielsen CU
Int J Pharm; 2018 Nov; 551(1-2):270-280. PubMed ID: 30240828
[TBL] [Abstract][Full Text] [Related]
17. Selenorhodamine photosensitizers for photodynamic therapy of P-glycoprotein-expressing cancer cells.
Hill JE; Linder MK; Davies KS; Sawada GA; Morgan J; Ohulchanskyy TY; Detty MR
J Med Chem; 2014 Oct; 57(20):8622-34. PubMed ID: 25250825
[TBL] [Abstract][Full Text] [Related]
18. Cloning and expression of murine sister of P-glycoprotein reveals a more discriminating transporter than MDR1/P-glycoprotein.
Lecureur V; Sun D; Hargrove P; Schuetz EG; Kim RB; Lan LB; Schuetz JD
Mol Pharmacol; 2000 Jan; 57(1):24-35. PubMed ID: 10617675
[TBL] [Abstract][Full Text] [Related]
19. Modulation of function of three ABC drug transporters, P-glycoprotein (ABCB1), mitoxantrone resistance protein (ABCG2) and multidrug resistance protein 1 (ABCC1) by tetrahydrocurcumin, a major metabolite of curcumin.
Limtrakul P; Chearwae W; Shukla S; Phisalphong C; Ambudkar SV
Mol Cell Biochem; 2007 Feb; 296(1-2):85-95. PubMed ID: 16960658
[TBL] [Abstract][Full Text] [Related]
20. Functional detection of MDR1/P170 and MRP/P190-mediated multidrug resistance in tumour cells by flow cytometry.
Feller N; Kuiper CM; Lankelma J; Ruhdal JK; Scheper RJ; Pinedo HM; Broxterman HJ
Br J Cancer; 1995 Sep; 72(3):543-9. PubMed ID: 7669559
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
