378 related articles for article (PubMed ID: 19422003)
21. In vitro trypanocidal activity of the anti-helminthic drug niclosamide.
Merschjohann K; Steverding D
Exp Parasitol; 2008 Apr; 118(4):637-40. PubMed ID: 18226810
[TBL] [Abstract][Full Text] [Related]
22. Synthesis and biological activity of nitro heterocycles analogous to megazol, a trypanocidal lead.
Chauvière G; Bouteille B; Enanga B; de Albuquerque C; Croft SL; Dumas M; Périé J
J Med Chem; 2003 Jan; 46(3):427-40. PubMed ID: 12540242
[TBL] [Abstract][Full Text] [Related]
23. Discovery of trypanocidal compounds by whole cell HTS of Trypanosoma brucei.
Mackey ZB; Baca AM; Mallari JP; Apsel B; Shelat A; Hansell EJ; Chiang PK; Wolff B; Guy KR; Williams J; McKerrow JH
Chem Biol Drug Des; 2006 May; 67(5):355-63. PubMed ID: 16784460
[TBL] [Abstract][Full Text] [Related]
24. Novel inhibitors of the trypanosome alternative oxidase inhibit Trypanosoma brucei brucei growth and respiration.
Ott R; Chibale K; Anderson S; Chipeleme A; Chaudhuri M; Guerrah A; Colowick N; Hill GC
Acta Trop; 2006 Dec; 100(3):172-84. PubMed ID: 17126803
[TBL] [Abstract][Full Text] [Related]
25. Design, synthesis and cruzain docking of 3-(4-substituted-aryl)-1,2,4-oxadiazole-N-acylhydrazones as anti-Trypanosoma cruzi agents.
dos Santos Filho JM; Leite AC; de Oliveira BG; Moreira DR; Lima MS; Soares MB; Leite LF
Bioorg Med Chem; 2009 Sep; 17(18):6682-91. PubMed ID: 19683450
[TBL] [Abstract][Full Text] [Related]
26. Antitrypanosomal activity of quaternary naphthalimide derivatives.
Muth M; Hoerr V; Glaser M; Ponte-Sucre A; Moll H; Stich A; Holzgrabe U
Bioorg Med Chem Lett; 2007 Mar; 17(6):1590-3. PubMed ID: 17239596
[TBL] [Abstract][Full Text] [Related]
27. 9- and 11-Substituted 4-azapaullones are potent and selective inhibitors of African trypanosoma.
Maiwald F; Benítez D; Charquero D; Dar MA; Erdmann H; Preu L; Koch O; Hölscher C; Loaëc N; Meijer L; Comini MA; Kunick C
Eur J Med Chem; 2014 Aug; 83():274-83. PubMed ID: 24973661
[TBL] [Abstract][Full Text] [Related]
28. In vitro antitrypanosomal activity of five low-MW antibiotics.
Ishiyama A; Otoguro K; Iwatsuki M; Namatame M; Nishihara-Tsukashima A; Takahashi Y; Onodera H; Yamada H; Omura S
J Antibiot (Tokyo); 2012 Feb; 65(2):113-4. PubMed ID: 22167160
[No Abstract] [Full Text] [Related]
29. Synthesis and tripanocidal activity of ferrocenyl and benzyl diamines against Trypanosoma brucei and Trypanosoma cruzi.
Velásquez AM; Francisco AI; Kohatsu AA; Silva FA; Rodrigues DF; Teixeira RG; Chiari BG; de Almeida MG; Isaac VL; Vargas MD; Cicarelli RM
Bioorg Med Chem Lett; 2014 Apr; 24(7):1707-10. PubMed ID: 24630563
[TBL] [Abstract][Full Text] [Related]
30. Identification and development of the 1,4-benzodiazepin-2-one and quinazoline-2,4-dione scaffolds as submicromolar inhibitors of HAT.
Clark RL; Clements CJ; Barrett MP; Mackay SP; Rathnam RP; Owusu-Dapaah G; Spencer J; Huggan JK
Bioorg Med Chem; 2012 Oct; 20(20):6019-33. PubMed ID: 22985960
[TBL] [Abstract][Full Text] [Related]
31. Chemical validation of GPI biosynthesis as a drug target against African sleeping sickness.
Smith TK; Crossman A; Brimacombe JS; Ferguson MA
EMBO J; 2004 Nov; 23(23):4701-8. PubMed ID: 15526036
[TBL] [Abstract][Full Text] [Related]
32. New oxapolycyclic cage amines with NMDA receptor antagonist and trypanocidal activities.
Duque MD; Camps P; Torres E; Valverde E; Sureda FX; López-Querol M; Camins A; Prathalingam SR; Kelly JM; Vázquez S
Bioorg Med Chem; 2010 Jan; 18(1):46-57. PubMed ID: 19954985
[TBL] [Abstract][Full Text] [Related]
33. Novel functionalized melamine-based nitroheterocycles: synthesis and activity against trypanosomatid parasites.
Baliani A; Peal V; Gros L; Brun R; Kaiser M; Barrett MP; Gilbert IH
Org Biomol Chem; 2009 Mar; 7(6):1154-66. PubMed ID: 19262935
[TBL] [Abstract][Full Text] [Related]
34. Evaluation of azasterols as anti-parasitics.
Gros L; Lorente SO; Jimenez CJ; Yardley V; Rattray L; Wharton H; Little S; Croft SL; Ruiz-Perez LM; Gonzalez-Pacanowska D; Gilbert IH
J Med Chem; 2006 Oct; 49(20):6094-103. PubMed ID: 17004723
[TBL] [Abstract][Full Text] [Related]
35. Antitrypanosomal structure-activity-relationship study of synthetic cynaropicrin derivatives.
Usuki T; Sato M; Hara S; Yoshimoto Y; Kondo R; Zimmermann S; Kaiser M; Brun R; Hamburger M; Adams M
Bioorg Med Chem Lett; 2014 Feb; 24(3):794-8. PubMed ID: 24433861
[TBL] [Abstract][Full Text] [Related]
36. Isothiocoumarin-3-carboxylic acid derivatives: synthesis, anticancer and antitrypanosomal activity evaluation.
Kaminskyy D; Kryshchyshyn A; Nektegayev I; Vasylenko O; Grellier P; Lesyk R
Eur J Med Chem; 2014 Mar; 75():57-66. PubMed ID: 24530491
[TBL] [Abstract][Full Text] [Related]
37. SAR of 2-amino and 2,4-diamino pyrimidines with in vivo efficacy against Trypanosoma brucei.
Perales JB; Freeman J; Bacchi CJ; Bowling T; Don R; Gaukel E; Mercer L; Moore JA; Nare B; Nguyen TM; Noe RA; Randolph R; Rewerts C; Wring SA; Yarlett N; Jacobs RT
Bioorg Med Chem Lett; 2011 May; 21(10):2816-9. PubMed ID: 21507639
[TBL] [Abstract][Full Text] [Related]
38. Novel 1,2-dihydroquinazolin-2-ones: Design, synthesis, and biological evaluation against Trypanosoma brucei.
Pham T; Walden M; Butler C; Diaz-Gonzalez R; Pérez-Moreno G; Ceballos-Pérez G; Gomez-Pérez V; García-Hernández R; Zecca H; Krakoff E; Kopec B; Ichire O; Mackenzie C; Pitot M; Ruiz LM; Gamarro F; González-Pacanowska D; Navarro M; Dounay AB
Bioorg Med Chem Lett; 2017 Aug; 27(16):3629-3635. PubMed ID: 28729055
[TBL] [Abstract][Full Text] [Related]
39. Structure-activity relationships of synthetic cordycepin analogues as experimental therapeutics for African trypanosomiasis.
Vodnala SK; Lundbäck T; Yeheskieli E; Sjöberg B; Gustavsson AL; Svensson R; Olivera GC; Eze AA; de Koning HP; Hammarström LG; Rottenberg ME
J Med Chem; 2013 Dec; 56(24):9861-73. PubMed ID: 24283924
[TBL] [Abstract][Full Text] [Related]
40. Design and synthesis of α-phenoxy-N-sulfonylphenyl acetamides as Trypanosoma brucei Leucyl-tRNA synthetase inhibitors.
Xin W; Li Z; Wang Q; Du J; Zhu M; Zhou H
Eur J Med Chem; 2020 Jan; 185():111827. PubMed ID: 31732256
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
