301 related articles for article (PubMed ID: 19463002)
1. Synthesis of novel 2-alkoxy-3-amino-3-arylpropan-1-ols and 5-alkoxy-4-aryl-1,3-oxazinanes with antimalarial activity.
D'hooghe M; Dekeukeleire S; Mollet K; Lategan C; Smith PJ; Chibale K; De Kimpe N
J Med Chem; 2009 Jul; 52(13):4058-62. PubMed ID: 19463002
[TBL] [Abstract][Full Text] [Related]
2. Microwave-assisted ring opening of epoxides: a general route to the synthesis of 1-aminopropan-2-ols with anti malaria parasite activities.
Robin A; Brown F; Bahamontes-Rosa N; Wu B; Beitz E; Kun JF; Flitsch SL
J Med Chem; 2007 Aug; 50(17):4243-9. PubMed ID: 17665900
[TBL] [Abstract][Full Text] [Related]
3. Novel oxazine skeletons as potential antiplasmodial active ingredients: Synthesis, in vitro and in vivo biology of some oxazine entities produced via cyclization of novel chalcone intermediates.
Tiwari V; Meshram J; Ali P; Sheikh J; Tripathi U
J Enzyme Inhib Med Chem; 2011 Aug; 26(4):569-78. PubMed ID: 21171899
[TBL] [Abstract][Full Text] [Related]
4. Synthesis, biological evaluation and mechanistic studies of totarol amino alcohol derivatives as potential antimalarial agents.
Tacon C; Guantai EM; Smith PJ; Chibale K
Bioorg Med Chem; 2012 Jan; 20(2):893-902. PubMed ID: 22196513
[TBL] [Abstract][Full Text] [Related]
5. Conformationally restrained aromatic analogues of fosmidomycin and FR900098.
Kurz T; Schlüter K; Pein M; Behrendt C; Bergmann B; Walter RD
Arch Pharm (Weinheim); 2007 Jul; 340(7):339-44. PubMed ID: 17611943
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and antimalarial activities of some furoxan sulfones and related furazans.
Galli U; Lazzarato L; Bertinaria M; Sorba G; Gasco A; Parapini S; Taramelli D
Eur J Med Chem; 2005 Dec; 40(12):1335-40. PubMed ID: 15979766
[TBL] [Abstract][Full Text] [Related]
7. Application of multicomponent reactions to antimalarial drug discovery. Part 3: discovery of aminoxazole 4-aminoquinolines with potent antiplasmodial activity in vitro.
Musonda CC; Little S; Yardley V; Chibale K
Bioorg Med Chem Lett; 2007 Sep; 17(17):4733-6. PubMed ID: 17644333
[TBL] [Abstract][Full Text] [Related]
8. Pharmacomodulation on the 3-acetylursolic acid skeleton: Design, synthesis, and biological evaluation of novel N-{3-[4-(3-aminopropyl)piperazinyl]propyl}-3-O-acetylursolamide derivatives as antimalarial agents.
Gnoatto SC; Susplugas S; Dalla Vechia L; Ferreira TB; Dassonville-Klimpt A; Zimmer KR; Demailly C; Da Nascimento S; Guillon J; Grellier P; Verli H; Gosmann G; Sonnet P
Bioorg Med Chem; 2008 Jan; 16(2):771-82. PubMed ID: 17967541
[TBL] [Abstract][Full Text] [Related]
9. In vitro efficiency of new acridyl derivatives against Plasmodium falciparum.
Guetzoyan L; Ramiandrasoa F; Dorizon H; Desprez C; Bridoux A; Rogier C; Pradines B; Perrée-Fauvet M
Bioorg Med Chem; 2007 May; 15(9):3278-89. PubMed ID: 17339112
[TBL] [Abstract][Full Text] [Related]
10. Synthesis, structural characterization and biological evaluation of novel stilbene derivatives as potential antimalarial agents.
Jung M; Park WH; Jung JC; Lim E; Lee Y; Oh S; Moon HI
Chem Biol Drug Des; 2009 Mar; 73(3):346-54. PubMed ID: 19207471
[TBL] [Abstract][Full Text] [Related]
11. Synthesis of aminoquinoline-based aminoalcohols and oxazolidinones and their antiplasmodial activity.
Kobarfard F; Yardley V; Little S; Daryaee F; Chibale K
Chem Biol Drug Des; 2012 Mar; 79(3):326-31. PubMed ID: 22129095
[TBL] [Abstract][Full Text] [Related]
12. gamma-Substituted bis(pivaloyloxymethyl)ester analogues of fosmidomycin and FR900098.
Kurz T; Behrendt C; Pein M; Kaula U; Bergmann B; Walter RD
Arch Pharm (Weinheim); 2007 Dec; 340(12):661-6. PubMed ID: 17994605
[TBL] [Abstract][Full Text] [Related]
13. In vitro and in vivo antimalarial activity of derivatives of 1,10-phenanthroline framework.
Yapi AD; Valentin A; Chezal JM; Chavignon O; Chaillot B; Gerhardt R; Teulade JC; Blache Y
Arch Pharm (Weinheim); 2006 Apr; 339(4):201-6. PubMed ID: 16586427
[TBL] [Abstract][Full Text] [Related]
14. Application of multicomponent reactions to antimalarial drug discovery. Part 2: New antiplasmodial and antitrypanosomal 4-aminoquinoline gamma- and delta-lactams via a 'catch and release' protocol.
Musonda CC; Gut J; Rosenthal PJ; Yardley V; Carvalho de Souza RC; Chibale K
Bioorg Med Chem; 2006 Aug; 14(16):5605-15. PubMed ID: 16690319
[TBL] [Abstract][Full Text] [Related]
15. Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline.
Delarue-Cochin S; Grellier P; Maes L; Mouray E; Sergheraert C; Melnyk P
Eur J Med Chem; 2008 Oct; 43(10):2045-55. PubMed ID: 18226428
[TBL] [Abstract][Full Text] [Related]
16. Design, synthesis and anti-plasmodial evaluation in vitro of new 4-aminoquinoline isatin derivatives.
Chiyanzu I; Clarkson C; Smith PJ; Lehman J; Gut J; Rosenthal PJ; Chibale K
Bioorg Med Chem; 2005 May; 13(9):3249-61. PubMed ID: 15809160
[TBL] [Abstract][Full Text] [Related]
17. Antimalarial and antitrypanosomal activity of a series of amide and sulfonamide derivatives of a 2,5-diaminobenzophenone.
Altenkämper M; Bechem B; Perruchon J; Heinrich S; Mädel A; Ortmann R; Dahse HM; Freunscht E; Wang Y; Rath J; Stich A; Hitzler M; Chiba P; Lanzer M; Schlitzer M
Bioorg Med Chem; 2009 Nov; 17(22):7690-7. PubMed ID: 19819706
[TBL] [Abstract][Full Text] [Related]
18. Synthesis and in vitro antiprotozoal activities of water-soluble, inexpensive 3,7-bis(dialkylamino)phenoxazin-5-ium derivatives.
Ge JF; Arai C; Kaiser M; Wittlin S; Brun R; Ihara M
J Med Chem; 2008 Jun; 51(12):3654-8. PubMed ID: 18476684
[TBL] [Abstract][Full Text] [Related]
19. Synthesis of new 7-chloroquinolinyl thioureas and their biological investigation as potential antimalarial and anticancer agents.
Mahajan A; Yeh S; Nell M; van Rensburg CE; Chibale K
Bioorg Med Chem Lett; 2007 Oct; 17(20):5683-5. PubMed ID: 17768052
[TBL] [Abstract][Full Text] [Related]
20. Synthesis of 2-[3-(7-Chloro-quinolin-4-ylamino)-alkyl]-1-(substituted phenyl)-2,3,4,9-tetrahydro-1H-beta-carbolines as a new class of antimalarial agents.
Gupta L; Srivastava K; Singh S; Puri SK; Chauhan PM
Bioorg Med Chem Lett; 2008 Jun; 18(11):3306-9. PubMed ID: 18442907
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
