BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

203 related articles for article (PubMed ID: 19481943)

  • 1. Synthesis of hybrid analogues of caffeine and eudistomin D and its affinity for adenosine receptors.
    Ishiyama H; Nakajima H; Nakata H; Kobayashi J
    Bioorg Med Chem; 2009 Jul; 17(13):4280-4. PubMed ID: 19481943
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis of hybrid molecules of caffeine and eudistomin D and its effects on adenosine receptors.
    Ohshita K; Ishiyama H; Oyanagi K; Nakata H; Kobayashi J
    Bioorg Med Chem; 2007 May; 15(9):3235-40. PubMed ID: 17350268
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis of eudistomin D analogues and its effects on adenosine receptors.
    Ishiyama H; Ohshita K; Abe T; Nakata H; Kobayashi J
    Bioorg Med Chem; 2008 Apr; 16(7):3825-30. PubMed ID: 18262425
    [TBL] [Abstract][Full Text] [Related]  

  • 4. 1,3-dialkyl-8-N-substituted benzyloxycarbonylamino-9-deazaxanthines as potent adenosine receptor ligands: Design, synthesis, structure-affinity and structure-selectivity relationships.
    Fernández F; Caamaño O; Isabel Nieto M; López C; García-Mera X; Stefanachi A; Nicolotti O; Isabel Loza M; Brea J; Esteve C; Segarra V; Vidal B; Carotti A
    Bioorg Med Chem; 2009 May; 17(10):3618-29. PubMed ID: 19398343
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and evaluation of analogues of the partial agonist 6-(propyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (6-PBC) and the full agonist 6-(benzyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (Zk 93423) at wild type and recombinant GABAA receptors.
    Cox ED; Diaz-Arauzo H; Huang Q; Reddy MS; Ma C; Harris B; McKernan R; Skolnick P; Cook JM
    J Med Chem; 1998 Jul; 41(14):2537-52. PubMed ID: 9651158
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Binding of tetrahydrocarboline derivatives at human 5-HT5A receptors.
    Khorana N; Smith C; Herrick-Davis K; Purohit A; Teitler M; Grella B; Dukat M; Glennon RA
    J Med Chem; 2003 Aug; 46(18):3930-7. PubMed ID: 12930153
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Tricyclic oxazolo[2,3-f]purinediones: potency as adenosine receptor ligands and anticonvulsants.
    Drabczyńska A; Müller CE; Schumacher B; Hinz S; Karolak-Wojciechowska J; Michalak B; Pekala E; Kieć-Kononowicz K
    Bioorg Med Chem; 2004 Sep; 12(18):4895-908. PubMed ID: 15336269
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis, biological evaluation, and molecular modeling of ribose-modified adenosine analogues as adenosine receptor agonists.
    Cappellacci L; Franchetti P; Pasqualini M; Petrelli R; Vita P; Lavecchia A; Novellino E; Costa B; Martini C; Klotz KN; Grifantini M
    J Med Chem; 2005 Mar; 48(5):1550-62. PubMed ID: 15743197
    [TBL] [Abstract][Full Text] [Related]  

  • 9. 2-(N-acyl) and 2-N-acyl-N(6)-substituted analogues of adenosine and their affinity at the human adenosine receptors.
    Jagtap PG; Chen Z; Szabó C; Klotz KN
    Bioorg Med Chem Lett; 2004 Mar; 14(6):1495-8. PubMed ID: 15006389
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis and biological activity of new potential agonists for the human adenosine A2A receptor.
    Bosch MP; Campos F; Niubó I; Rosell G; Díaz JL; Brea J; Loza MI; Guerrero A
    J Med Chem; 2004 Jul; 47(16):4041-53. PubMed ID: 15267242
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Phenylethyl-substituted pyrimido[2,1-f]purinediones and related compounds: structure-activity relationships as adenosine A(1) and A(2A) receptor ligands.
    Drabczyńska A; Müller CE; Schiedel A; Schumacher B; Karolak-Wojciechowska J; Fruziński A; Zobnina W; Yuzlenko O; Kieć-Kononowicz K
    Bioorg Med Chem; 2007 Nov; 15(22):6956-74. PubMed ID: 17827019
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Development of spin-labeled probes for adenosine receptors.
    Ilas J; Pecar S; Hockemeyer J; Euler H; Kirfel A; Müller CE
    J Med Chem; 2005 Mar; 48(6):2108-14. PubMed ID: 15771453
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis and adenosine receptor binding studies of some novel triazolothienopyrimidines.
    Raghu Prasad M; Raghuram Rao A; Shanthan Rao P; Rajan KS; Meena S; Madhavi K
    Eur J Med Chem; 2008 Mar; 43(3):614-20. PubMed ID: 17602796
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and pharmacological evaluation of novel 1- and 8-substituted-3-furfuryl xanthines as adenosine receptor antagonists.
    Balo MC; Brea J; Caamaño O; Fernández F; García-Mera X; López C; Loza MI; Nieto MI; Rodríguez-Borges JE
    Bioorg Med Chem; 2009 Sep; 17(18):6755-60. PubMed ID: 19682912
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis, adenosine receptor binding and 3D-QSAR of 4-substituted 2-(2'-furyl)-1,2,4-triazolo[1,5-a]quinoxalines.
    Martínez A; Gutiérrez-de-Terán H; Brea J; Raviña E; Loza MI; Cadavid MI; Sanz F; Vidal B; Segarra V; Sotelo E
    Bioorg Med Chem; 2008 Feb; 16(4):2103-13. PubMed ID: 18249548
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis of a new series of 1H-imidazol-1-yl substituted 8-phenylxanthines as adenosine receptor ligands.
    Bansal R; Kumar G; Gandhi D; Young LC; Harvey AL
    Chem Biodivers; 2011 Jul; 8(7):1290-300. PubMed ID: 21766450
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Molecular determinants of beta-carboline inhibition of the glycine receptor.
    Chen X; Cromer BA; Lynch JW
    J Neurochem; 2009 Sep; 110(5):1685-94. PubMed ID: 19619142
    [TBL] [Abstract][Full Text] [Related]  

  • 18. 5'-Carbamoyl derivatives of 2'-C-methyl-purine nucleosides as selective A1 adenosine receptor agonists: affinity, efficacy, and selectivity for A1 receptor from different species.
    Cappellacci L; Franchetti P; Vita P; Petrelli R; Lavecchia A; Costa B; Spinetti F; Martini C; Klotz KN; Grifantini M
    Bioorg Med Chem; 2008 Jan; 16(1):336-53. PubMed ID: 17933541
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Binding of beta-carbolines at imidazoline I2 receptors: a structure-affinity investigation.
    Glennon RA; Grella B; Tyacke RJ; Lau A; Westaway J; Hudson AL
    Bioorg Med Chem Lett; 2004 Feb; 14(4):999-1002. PubMed ID: 15013009
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Dual inhibition of monoamine oxidase B and antagonism of the adenosine A(2A) receptor by (E,E)-8-(4-phenylbutadien-1-yl)caffeine analogues.
    Pretorius J; Malan SF; Castagnoli N; Bergh JJ; Petzer JP
    Bioorg Med Chem; 2008 Sep; 16(18):8676-84. PubMed ID: 18723354
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 11.