These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

339 related articles for article (PubMed ID: 19524602)

  • 1. 6beta,19-Bridged androstenedione analogs as aromatase inhibitors.
    Komatsu S; Yaguchi A; Yamashita K; Nagaoka M; Numazawa M
    Steroids; 2009 Nov; 74(12):884-9. PubMed ID: 19524602
    [TBL] [Abstract][Full Text] [Related]  

  • 2. An efficient steroid pharmacophore-based strategy to identify new aromatase inhibitors.
    Neves MA; Dinis TC; Colombo G; Sá e Melo ML
    Eur J Med Chem; 2009 Oct; 44(10):4121-7. PubMed ID: 19500885
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Structure-activity relationships of new A,D-ring modified steroids as aromatase inhibitors: design, synthesis, and biological activity evaluation.
    Cepa MM; Tavares da Silva EJ; Correia-da-Silva G; Roleira FM; Teixeira NA
    J Med Chem; 2005 Oct; 48(20):6379-85. PubMed ID: 16190763
    [TBL] [Abstract][Full Text] [Related]  

  • 4. 4- and 6-(p-Sulphamoylphenyl)androstenediones: Studies of aromatase inhibitor-based oestrone sulphatase inhibition.
    Watari Y; Yamaguchi S; Takahashi M; Nagaoka M; Numazawa M
    Steroids; 2010 Dec; 75(12):891-6. PubMed ID: 20546769
    [TBL] [Abstract][Full Text] [Related]  

  • 5. New structure-activity relationships of A- and D-ring modified steroidal aromatase inhibitors: design, synthesis, and biochemical evaluation.
    Varela C; Tavares da Silva EJ; Amaral C; Correia da Silva G; Baptista T; Alcaro S; Costa G; Carvalho RA; Teixeira NA; Roleira FM
    J Med Chem; 2012 Apr; 55(8):3992-4002. PubMed ID: 22475216
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis of some epoxy and/or N-oxy 17-picolyl and 17-picolinylidene-androst-5-ene derivatives and evaluation of their biological activity.
    Djurendić E; Daljev J; Sakac M; Canadi J; Santa SJ; Andrić S; Klisurić O; Kojić V; Bogdanović G; Djurendić-Brenesel M; Novaković S; Gasi KP
    Steroids; 2008 Jan; 73(1):129-38. PubMed ID: 17963806
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Probing the binding pocket of the active site of aromatase with 6-ether or 6-ester substituted androst-4-ene-3,17-diones and their diene and triene analogs.
    Numazawa M; Shelangouski M; Nagasaka M
    Steroids; 2000 Dec; 65(12):871-82. PubMed ID: 11077085
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Substituted C19 steroid analogs as inhibitors of aromatase.
    Brueggemeier RW; Snider CE; Counsell RE
    Cancer Res; 1982 Aug; 42(8 Suppl):3334s-3337s. PubMed ID: 7083196
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and biochemical studies of 17-substituted androst-3-enes and 3,4-epoxyandrostanes as aromatase inhibitors.
    Cepa MM; Tavares da Silva EJ; Correia-da-Silva G; Roleira FM; Teixeira NA
    Steroids; 2008 Dec; 73(14):1409-15. PubMed ID: 18691607
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis and biochemical properties of 6-bromoandrostenedione derivatives with a 2,2-dimethyl or 2-methyl group as aromatase inhibitors.
    Numazawa M; Handa W; Yamada K
    Biol Pharm Bull; 2004 Nov; 27(11):1878-82. PubMed ID: 15516742
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Time-dependent inactivation of aromatase by 6-alkylandrosta-1,4-diene-3,17-diones. Effects of length and configuration of 6-alkyl group.
    Numazawa M; Oshibe M; Yamaguchi S; Tachibana M
    J Med Chem; 1996 Mar; 39(5):1033-8. PubMed ID: 8676338
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Biochemistry and pharmacology of 7alpha-substituted androstenediones as aromatase inhibitors.
    Brueggemeier RW; O'Reilly JM; Lovely CJ; Ward PJ; Quinn AL; Baker D; Darby MV; Gu XJ; Gilbert NE
    J Steroid Biochem Mol Biol; 1997 Apr; 61(3-6):247-54. PubMed ID: 9365197
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Aromatase inhibition by 4 beta,5 beta-epoxides of 16 alpha-hydroxyandrostenedione and its 19-oxygenated analogs, potential precursors of estriol production in the feto-placental unit.
    Numazawa M; Yoshimura A; Watari Y; Matsuzaki H
    Biol Pharm Bull; 2002 Dec; 25(12):1566-9. PubMed ID: 12499641
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Androst-5-ene-7,17-dione: a novel class of suicide substrate of aromatase.
    Numazawa M; Mutsumi A; Hoshi K; Tanaka Y
    Biochem Biophys Res Commun; 1992 Jul; 186(1):32-9. PubMed ID: 1632774
    [TBL] [Abstract][Full Text] [Related]  

  • 15. 6beta-Methyl-B-norandrostenedione.
    Andrade LC; de Almeida MJ; Neves MA; Dinis TC; Sá e Melo ML
    Acta Crystallogr C; 2010 Apr; 66(Pt 4):o185-6. PubMed ID: 20354306
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Structure-activity relationships of 2-, 4-, or 6-substituted estrogens as aromatase inhibitors.
    Numazawa M; Ando M; Watari Y; Tominaga T; Hayata Y; Yoshimura A
    J Steroid Biochem Mol Biol; 2005 Jun; 96(1):51-8. PubMed ID: 16039845
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Gas chromatography-mass spectrometric study of 19-oxygenation of the aromatase inhibitor 19-methylandrostenedione with human placental microsomes.
    Numazawa M; Nagaoka M; Handa W; Yamada A
    Biol Pharm Bull; 2006 Jun; 29(6):1242-5. PubMed ID: 16755025
    [TBL] [Abstract][Full Text] [Related]  

  • 18. 6-Phenylaliphatic-substituted androst-4-ene-3,17-diones as aromatase inhibitors: structure-activity relationships.
    Numazawa M; Yamaguchi S
    J Steroid Biochem Mol Biol; 1998 Oct; 67(1):41-8. PubMed ID: 9780028
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Probing the binding pocket of the active site of aromatase with 2-phenylaliphatic androsta-1,4-diene-3,17-dione steroids.
    Takahashi M; Yamashita K; Numazawa M
    Steroids; 2010 Apr; 75(4-5):330-7. PubMed ID: 20096721
    [TBL] [Abstract][Full Text] [Related]  

  • 20. 19-oxygenated derivatives of androst-4-ene-6,17-dione and androst-5-ene-4,17-dione as catalytic probes for the active site of aromatase.
    Numazawa M; Yamada K; Kidokoro K
    Biol Pharm Bull; 1999 Oct; 22(10):1134-6. PubMed ID: 10549872
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 17.