131 related articles for article (PubMed ID: 19748781)
1. Synthesis and biological evaluation of new heterocyclic quinolinones as anti-parasite and anti-HIV drug candidates.
Darque A; Dumètre A; Hutter S; Casano G; Robin M; Pannecouque C; Azas N
Bioorg Med Chem Lett; 2009 Oct; 19(20):5962-4. PubMed ID: 19748781
[TBL] [Abstract][Full Text] [Related]
2. Synthesis and biological evaluation of 2,3-dihydroimidazo[1,2-a]benzimidazole derivatives against Leishmania donovani and Trypanosoma cruzi.
Oh S; Kim S; Kong S; Yang G; Lee N; Han D; Goo J; Siqueira-Neto JL; Freitas-Junior LH; Song R
Eur J Med Chem; 2014 Sep; 84():395-403. PubMed ID: 25036797
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and antiparasitic and antifungal evaluation of 2'-arylsubstituted-1H,1'H-[2,5']bisbenzimidazolyl-5-carboxamidines.
Alp M; Göker H; Brun R; Yildiz S
Eur J Med Chem; 2009 May; 44(5):2002-8. PubMed ID: 19010569
[TBL] [Abstract][Full Text] [Related]
4. Synthesis, characterization, antiparasitic and cytotoxic evaluation of thioureas conjugated to polyamine scaffolds.
Stringer T; Taylor D; de Kock C; Guzgay H; Au A; An SH; Sanchez B; O'Connor R; Patel N; Land KM; Smith PJ; Hendricks DT; Egan TJ; Smith GS
Eur J Med Chem; 2013 Nov; 69():90-8. PubMed ID: 24012713
[TBL] [Abstract][Full Text] [Related]
5. Synthesis of novel guttiferone A derivatives: in-vitro evaluation toward Plasmodium falciparum, Trypanosoma brucei and Leishmania donovani.
Fromentin Y; Gaboriaud-Kolar N; Lenta BN; Wansi JD; Buisson D; Mouray E; Grellier P; Loiseau PM; Lallemand MC; Michel S
Eur J Med Chem; 2013 Jul; 65():284-94. PubMed ID: 23727538
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and antiparasitic evaluation of bis-2,5-[4-guanidinophenyl]thiophenes.
Gonzalez JL; Stephens CE; Wenzler T; Brun R; Tanious FA; Wilson WD; Barszcz T; Werbovetz KA; Boykin DW
Eur J Med Chem; 2007 Apr; 42(4):552-7. PubMed ID: 17178177
[TBL] [Abstract][Full Text] [Related]
7. Biological evaluation of substituted quinolines.
Franck X; Fournet A; Prina E; Mahieux R; Hocquemiller R; Figadère B
Bioorg Med Chem Lett; 2004 Jul; 14(14):3635-8. PubMed ID: 15203133
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and antikinetoplastid activities of 3-substituted quinolinones derivatives.
Audisio D; Messaoudi S; Cojean S; Peyrat JF; Brion JD; Bories C; Huteau F; Loiseau PM; Alami M
Eur J Med Chem; 2012 Jun; 52():44-50. PubMed ID: 22472166
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and antiprotozoal activity of some new synthetic substituted quinoxalines.
Hui X; Desrivot J; Bories C; Loiseau PM; Franck X; Hocquemiller R; Figadère B
Bioorg Med Chem Lett; 2006 Feb; 16(4):815-20. PubMed ID: 16309903
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and evaluation of 2-pyridyl pyrimidines with in vitro antiplasmodial and antileishmanial activity.
Musonda CC; Whitlock GA; Witty MJ; Brun R; Kaiser M
Bioorg Med Chem Lett; 2009 Jan; 19(2):401-5. PubMed ID: 19091562
[TBL] [Abstract][Full Text] [Related]
11. Antiparasitic activity of highly conjugated pyrimidine-2,4-dione derivatives.
Azas N; Rathelot P; Djekou S; Delmas F; Gellis A; Di Giorgio C; Vanelle P; Timon-David P
Farmaco; 2003 Dec; 58(12):1263-70. PubMed ID: 14630237
[TBL] [Abstract][Full Text] [Related]
12. 1,3-Diphenylpyrazoles: synthesis and antiparasitic activities of azomethine derivatives.
Rathelot P; Azas N; El-Kashef H; Delmas F; Di Giorgio C; Timon-David P; Maldonado J; Vanelle P
Eur J Med Chem; 2002 Aug; 37(8):671-9. PubMed ID: 12161064
[TBL] [Abstract][Full Text] [Related]
13. Polyamine quinoline rhodium complexes: synthesis and pharmacological evaluation as antiparasitic agents against Plasmodium falciparum and Trichomonas vaginalis.
Stringer T; Taylor D; Guzgay H; Shokar A; Au A; Smith PJ; Hendricks DT; Land KM; Egan TJ; Smith GS
Dalton Trans; 2015 Sep; 44(33):14906-17. PubMed ID: 26226082
[TBL] [Abstract][Full Text] [Related]
14. In vitro and in silico studies of polycondensed diazine systems as anti-parasitic agents.
Almerico AM; Tutone M; Guarcello A; Lauria A
Bioorg Med Chem Lett; 2012 Jan; 22(2):1000-4. PubMed ID: 22197138
[TBL] [Abstract][Full Text] [Related]
15. Multifunctional host defense peptides: antiparasitic activities.
Mor A
FEBS J; 2009 Nov; 276(22):6474-82. PubMed ID: 19817857
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and antiparasitic properties of new 4-N-benzylamino-4-hetarylbut-1-enes.
Kouznetsov VV; Castro JR; Puentes CO; Stashenko EE; Martínez JR; Ochoa C; Pereira DM; Ruiz JJ; Portillo CF; Serrano SM; Barrio AG; Bahsas A; Amaro-Luis J
Arch Pharm (Weinheim); 2005 Jan; 338(1):32-7. PubMed ID: 15674802
[TBL] [Abstract][Full Text] [Related]
17. Lowering of 5-nitroimidazole's mutagenicity: towards optimal antiparasitic pharmacophore.
Crozet MD; Botta C; Gasquet M; Curti C; Rémusat V; Hutter S; Chapelle O; Azas N; De Méo M; Vanelle P
Eur J Med Chem; 2009 Feb; 44(2):653-9. PubMed ID: 18590939
[TBL] [Abstract][Full Text] [Related]
18. 2-Phenylquinolones as inhibitors of the HIV-1 Tat-TAR interaction.
Gatto B; Tabarrini O; Massari S; Giaretta G; Sabatini S; Del Vecchio C; Parolin C; Fravolini A; Palumbo M; Cecchetti V
ChemMedChem; 2009 Jun; 4(6):935-8. PubMed ID: 19283692
[TBL] [Abstract][Full Text] [Related]
19. Synthesis and biological evaluation of a novel series of aryl S,N-ketene acetals as antileishmanial agents.
Suryawanshi SN; Kumar S; Tiwari A; Shivahare R; Chhonker YS; Pandey S; Shakya N; Bhatta RS; Gupta S
Bioorg Med Chem Lett; 2013 Jul; 23(13):3979-82. PubMed ID: 23673014
[TBL] [Abstract][Full Text] [Related]
20. Lead selection of antiparasitic compounds from a focused library of benzenesulfonyl derivatives of heterocycles.
Pagliero RJ; Kaiser M; Brun R; Nieto MJ; Mazzieri MR
Bioorg Med Chem Lett; 2017 Sep; 27(17):3945-3949. PubMed ID: 28789893
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]