515 related articles for article (PubMed ID: 19926176)
1. Synthesis and antimalarial evaluation of 1, 3, 5-trisubstituted pyrazolines.
Acharya BN; Saraswat D; Tiwari M; Shrivastava AK; Ghorpade R; Bapna S; Kaushik MP
Eur J Med Chem; 2010 Feb; 45(2):430-8. PubMed ID: 19926176
[TBL] [Abstract][Full Text] [Related]
2. Novel oxazine skeletons as potential antiplasmodial active ingredients: Synthesis, in vitro and in vivo biology of some oxazine entities produced via cyclization of novel chalcone intermediates.
Tiwari V; Meshram J; Ali P; Sheikh J; Tripathi U
J Enzyme Inhib Med Chem; 2011 Aug; 26(4):569-78. PubMed ID: 21171899
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and evaluation of sulfonylurea derivatives as novel antimalarials.
León C; Rodrigues J; Gamboa de Domínguez N; Charris J; Gut J; Rosenthal PJ; Domínguez JN
Eur J Med Chem; 2007 Jun; 42(6):735-42. PubMed ID: 17321641
[TBL] [Abstract][Full Text] [Related]
4. Synthesis of novel alpha-pyranochalcones and pyrazoline derivatives as Plasmodium falciparum growth inhibitors.
Wanare G; Aher R; Kawathekar N; Ranjan R; Kaushik NK; Sahal D
Bioorg Med Chem Lett; 2010 Aug; 20(15):4675-8. PubMed ID: 20576433
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and antimalarial activity in vitro and in vivo of a new ferrocene-chloroquine analogue.
Biot C; Glorian G; Maciejewski LA; Brocard JS
J Med Chem; 1997 Nov; 40(23):3715-8. PubMed ID: 9371235
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and in vitro evaluation of new chloroquine-chalcone hybrids against chloroquine-resistant strain of Plasmodium falciparum.
Sashidhara KV; Avula SR; Palnati GR; Singh SV; Srivastava K; Puri SK; Saxena JK
Bioorg Med Chem Lett; 2012 Sep; 22(17):5455-9. PubMed ID: 22850213
[TBL] [Abstract][Full Text] [Related]
7. A new class of phenazines with activity against a chloroquine resistant Plasmodium falciparum strain and antimicrobial activity.
Hussain H; Specht S; Sarite SR; Saeftel M; Hoerauf A; Schulz B; Krohn K
J Med Chem; 2011 Jul; 54(13):4913-7. PubMed ID: 21591758
[TBL] [Abstract][Full Text] [Related]
8. Dibenzylideneacetone analogues as novel Plasmodium falciparum inhibitors.
Aher RB; Wanare G; Kawathekar N; Kumar RR; Kaushik NK; Sahal D; Chauhan VS
Bioorg Med Chem Lett; 2011 May; 21(10):3034-6. PubMed ID: 21493068
[TBL] [Abstract][Full Text] [Related]
9. 4, 5-Dihydrooxazole-pyrazoline hybrids: Synthesis and their evaluation as potential antimalarial agents.
Pandey AK; Sharma S; Pandey M; Alam MM; Shaquiquzzaman M; Akhter M
Eur J Med Chem; 2016 Nov; 123():476-486. PubMed ID: 27494165
[TBL] [Abstract][Full Text] [Related]
10. Antimalarial acridines: synthesis, in vitro activity against P. falciparum and interaction with hematin.
Guetzoyan L; Yu XM; Ramiandrasoa F; Pethe S; Rogier C; Pradines B; Cresteil T; Perrée-Fauvet M; Mahy JP
Bioorg Med Chem; 2009 Dec; 17(23):8032-9. PubMed ID: 19879150
[TBL] [Abstract][Full Text] [Related]
11. Design and synthesis of new antimalarial agents from 4-aminoquinoline.
Solomon VR; Puri SK; Srivastava K; Katti SB
Bioorg Med Chem; 2005 Mar; 13(6):2157-65. PubMed ID: 15727868
[TBL] [Abstract][Full Text] [Related]
12. Antimalarial activity of 4-(5-trifluoromethyl-1H-pyrazol-1-yl)-chloroquine analogues.
Cunico W; Cechinel CA; Bonacorso HG; Martins MA; Zanatta N; de Souza MV; Freitas IO; Soares RP; Krettli AU
Bioorg Med Chem Lett; 2006 Feb; 16(3):649-53. PubMed ID: 16257205
[TBL] [Abstract][Full Text] [Related]
13. Synthesis of three classes of rhodacyanine dyes and evaluation of their in vitro and in vivo antimalarial activity.
Pudhom K; Kasai K; Terauchi H; Inoue H; Kaiser M; Brun R; Ihara M; Takasu K
Bioorg Med Chem; 2006 Dec; 14(24):8550-63. PubMed ID: 16971131
[TBL] [Abstract][Full Text] [Related]
14. Synthesis of some cryptolepine analogues, assessment of their antimalarial and cytotoxic activities, and consideration of their antimalarial mode of action.
Onyeibor O; Croft SL; Dodson HI; Feiz-Haddad M; Kendrick H; Millington NJ; Parapini S; Phillips RM; Seville S; Shnyder SD; Taramelli D; Wright CW
J Med Chem; 2005 Apr; 48(7):2701-9. PubMed ID: 15801861
[TBL] [Abstract][Full Text] [Related]
15. Bisquinolines. 2. Antimalarial N,N-bis(7-chloroquinolin-4-yl)heteroalkanediamines.
Vennerstrom JL; Ager AL; Dorn A; Andersen SL; Gerena L; Ridley RG; Milhous WK
J Med Chem; 1998 Oct; 41(22):4360-4. PubMed ID: 9784111
[TBL] [Abstract][Full Text] [Related]
16. Quinoline antimalarials containing a dibemethin group are active against chloroquinone-resistant Plasmodium falciparum and inhibit chloroquine transport via the P. falciparum chloroquine-resistance transporter (PfCRT).
Zishiri VK; Joshi MC; Hunter R; Chibale K; Smith PJ; Summers RL; Martin RE; Egan TJ
J Med Chem; 2011 Oct; 54(19):6956-68. PubMed ID: 21875063
[TBL] [Abstract][Full Text] [Related]
17. Parallel solution-phase synthesis of conformationally restricted congeners of pentamidine and evaluation of their antiplasmodial activities.
Mayence A; Vanden Eynde JJ; Krogstad FM; Krogstad DJ; Cushion MT; Huang TL
J Med Chem; 2004 May; 47(10):2700-5. PubMed ID: 15115412
[TBL] [Abstract][Full Text] [Related]
18. Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline.
Delarue-Cochin S; Grellier P; Maes L; Mouray E; Sergheraert C; Melnyk P
Eur J Med Chem; 2008 Oct; 43(10):2045-55. PubMed ID: 18226428
[TBL] [Abstract][Full Text] [Related]
19. Synthesis of N1-arylidene-N2-quinolyl- and N2-acrydinylhydrazones as potent antimalarial agents active against CQ-resistant P. falciparum strains.
Gemma S; Kukreja G; Fattorusso C; Persico M; Romano MP; Altarelli M; Savini L; Campiani G; Fattorusso E; Basilico N; Taramelli D; Yardley V; Butini S
Bioorg Med Chem Lett; 2006 Oct; 16(20):5384-8. PubMed ID: 16890433
[TBL] [Abstract][Full Text] [Related]
20. 4-Aminoquinoline quinolizidinyl- and quinolizidinylalkyl-derivatives with antimalarial activity.
Sparatore A; Basilico N; Parapini S; Romeo S; Novelli F; Sparatore F; Taramelli D
Bioorg Med Chem; 2005 Sep; 13(18):5338-45. PubMed ID: 16054368
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]