These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
2. Flavan-3-ol derivatives are positive modulators of GABA(A) receptors with higher efficacy for the alpha(2) subtype and anxiolytic action in mice. Fernandez SP; Mewett KN; Hanrahan JR; Chebib M; Johnston GA Neuropharmacology; 2008 Oct; 55(5):900-7. PubMed ID: 18657554 [TBL] [Abstract][Full Text] [Related]
3. The modulatory effects of the anxiolytic etifoxine on GABA(A) receptors are mediated by the beta subunit. Hamon A; Morel A; Hue B; Verleye M; Gillardin JM Neuropharmacology; 2003 Sep; 45(3):293-303. PubMed ID: 12871647 [TBL] [Abstract][Full Text] [Related]
4. The anxioselective agent 7-(2-chloropyridin-4-yl)pyrazolo-[1,5-a]-pyrimidin-3-yl](pyridin-2-yl)methanone (DOV 51892) is more efficacious than diazepam at enhancing GABA-gated currents at alpha1 subunit-containing GABAA receptors. Popik P; Kostakis E; Krawczyk M; Nowak G; Szewczyk B; Krieter P; Chen Z; Russek SJ; Gibbs TT; Farb DH; Skolnick P; Lippa AS; Basile AS J Pharmacol Exp Ther; 2006 Dec; 319(3):1244-52. PubMed ID: 16971504 [TBL] [Abstract][Full Text] [Related]
5. 2'-Methoxy-6-methylflavone: a novel anxiolytic and sedative with subtype selective activating and modulating actions at GABA(A) receptors. Karim N; Curmi J; Gavande N; Johnston GA; Hanrahan JR; Tierney ML; Chebib M Br J Pharmacol; 2012 Feb; 165(4):880-96. PubMed ID: 21797842 [TBL] [Abstract][Full Text] [Related]
6. Anxiolytic-like effects of 8-acetylene imidazobenzodiazepines in a rhesus monkey conflict procedure. Fischer BD; Licata SC; Edwankar RV; Wang ZJ; Huang S; He X; Yu J; Zhou H; Johnson EM; Cook JM; Furtmüller R; Ramerstorfer J; Sieghart W; Roth BL; Majumder S; Rowlett JK Neuropharmacology; 2010 Dec; 59(7-8):612-8. PubMed ID: 20727364 [TBL] [Abstract][Full Text] [Related]
7. Novel positive allosteric modulators of GABAA receptors: do subtle differences in activity at alpha1 plus alpha5 versus alpha2 plus alpha3 subunits account for dissimilarities in behavioral effects in rats? Savić MM; Majumder S; Huang S; Edwankar RV; Furtmüller R; Joksimović S; Clayton T; Ramerstorfer J; Milinković MM; Roth BL; Sieghart W; Cook JM Prog Neuropsychopharmacol Biol Psychiatry; 2010 Mar; 34(2):376-86. PubMed ID: 20074611 [TBL] [Abstract][Full Text] [Related]
8. Delineation of the functional properties and the mechanism of action of AA29504, an allosteric agonist and positive allosteric modulator of GABA Olander ER; Madjroh N; Bunch L; Söderhielm PC; Jensen AA Biochem Pharmacol; 2018 Apr; 150():305-319. PubMed ID: 29454619 [TBL] [Abstract][Full Text] [Related]
9. Modulation of GABA(A) receptor function by neuroactive steroids: evidence for heterogeneity of steroid sensitivity of recombinant GABA(A) receptor isoforms. Maitra R; Reynolds JN Can J Physiol Pharmacol; 1998 Sep; 76(9):909-20. PubMed ID: 10066142 [TBL] [Abstract][Full Text] [Related]
10. Pharmacology of the human gamma-aminobutyric acidA receptor alpha 4 subunit expressed in Xenopus laevis oocytes. Whittemore ER; Yang W; Drewe JA; Woodward RM Mol Pharmacol; 1996 Nov; 50(5):1364-75. PubMed ID: 8913369 [TBL] [Abstract][Full Text] [Related]
11. 6-Methylflavanone, a more efficacious positive allosteric modulator of gamma-aminobutyric acid (GABA) action at human recombinant alpha2beta2gamma2L than at alpha1beta2gamma2L and alpha1beta2 GABA(A) receptors expressed in Xenopus oocytes. Hall BJ; Chebib M; Hanrahan JR; Johnston GA Eur J Pharmacol; 2005 Apr; 512(2-3):97-104. PubMed ID: 15840393 [TBL] [Abstract][Full Text] [Related]
12. Thymol, a constituent of thyme essential oil, is a positive allosteric modulator of human GABA(A) receptors and a homo-oligomeric GABA receptor from Drosophila melanogaster. Priestley CM; Williamson EM; Wafford KA; Sattelle DB Br J Pharmacol; 2003 Dec; 140(8):1363-72. PubMed ID: 14623762 [TBL] [Abstract][Full Text] [Related]
13. Barbiturate interactions at the human GABAA receptor: dependence on receptor subunit combination. Thompson SA; Whiting PJ; Wafford KA Br J Pharmacol; 1996 Feb; 117(3):521-527. PubMed ID: 8821543 [TBL] [Abstract][Full Text] [Related]
14. GABAA α5 subunit-containing receptors do not contribute to reversal of inflammatory-induced spinal sensitization as indicated by the unique selectivity profile of the GABAA receptor allosteric modulator NS16085. de Lucas AG; Ahring PK; Larsen JS; Rivera-Arconada I; Lopez-Garcia JA; Mirza NR; Munro G Biochem Pharmacol; 2015 Feb; 93(3):370-9. PubMed ID: 25542996 [TBL] [Abstract][Full Text] [Related]