267 related articles for article (PubMed ID: 19959746)
1. No evidence for functional selectivity of proxyfan at the human histamine H3 receptor coupled to defined Gi/Go protein heterotrimers.
Schnell D; Burleigh K; Trick J; Seifert R
J Pharmacol Exp Ther; 2010 Mar; 332(3):996-1005. PubMed ID: 19959746
[TBL] [Abstract][Full Text] [Related]
2. Modulation of histamine H(3) receptor function by monovalent ions.
Schnell D; Seifert R
Neurosci Lett; 2010 Mar; 472(2):114-8. PubMed ID: 20132865
[TBL] [Abstract][Full Text] [Related]
3. G protein-dependent pharmacology of histamine H3 receptor ligands: evidence for heterogeneous active state receptor conformations.
Krueger KM; Witte DG; Ireland-Denny L; Miller TR; Baranowski JL; Buckner S; Milicic I; Esbenshade TA; Hancock AA
J Pharmacol Exp Ther; 2005 Jul; 314(1):271-81. PubMed ID: 15821027
[TBL] [Abstract][Full Text] [Related]
4. Histamine H(4) receptor-RGS fusion proteins expressed in Sf9 insect cells: a sensitive and reliable approach for the functional characterization of histamine H(4) receptor ligands.
Schneider EH; Seifert R
Biochem Pharmacol; 2009 Sep; 78(6):607-16. PubMed ID: 19464266
[TBL] [Abstract][Full Text] [Related]
5. Constitutive activity and ligand selectivity of human, guinea pig, rat, and canine histamine H2 receptors.
Preuss H; Ghorai P; Kraus A; Dove S; Buschauer A; Seifert R
J Pharmacol Exp Ther; 2007 Jun; 321(3):983-95. PubMed ID: 17332265
[TBL] [Abstract][Full Text] [Related]
6. Mutations of Cys-17 and Ala-271 in the human histamine H2 receptor determine the species selectivity of guanidine-type agonists and increase constitutive activity.
Preuss H; Ghorai P; Kraus A; Dove S; Buschauer A; Seifert R
J Pharmacol Exp Ther; 2007 Jun; 321(3):975-82. PubMed ID: 17347323
[TBL] [Abstract][Full Text] [Related]
7. Sf9 cells: a versatile model system to investigate the pharmacological properties of G protein-coupled receptors.
Schneider EH; Seifert R
Pharmacol Ther; 2010 Dec; 128(3):387-418. PubMed ID: 20705094
[TBL] [Abstract][Full Text] [Related]
8. G protein coupling and ligand selectivity of the D2L and D3 dopamine receptors.
Lane JR; Powney B; Wise A; Rees S; Milligan G
J Pharmacol Exp Ther; 2008 Apr; 325(1):319-30. PubMed ID: 18218829
[TBL] [Abstract][Full Text] [Related]
9. Protean agonism at the dopamine D2 receptor: (S)-3-(3-hydroxyphenyl)-N-propylpiperidine is an agonist for activation of Go1 but an antagonist/inverse agonist for Gi1,Gi2, and Gi3.
Lane JR; Powney B; Wise A; Rees S; Milligan G
Mol Pharmacol; 2007 May; 71(5):1349-59. PubMed ID: 17287401
[TBL] [Abstract][Full Text] [Related]
10. Structural requirements for inverse agonism and neutral antagonism of indole-, benzimidazole-, and thienopyrrole-derived histamine H4 receptor ligands.
Schneider EH; Strasser A; Thurmond RL; Seifert R
J Pharmacol Exp Ther; 2010 Aug; 334(2):513-21. PubMed ID: 20484153
[TBL] [Abstract][Full Text] [Related]
11. Probing ligand-specific histamine H1- and H2-receptor conformations with NG-acylated Imidazolylpropylguanidines.
Xie SX; Ghorai P; Ye QZ; Buschauer A; Seifert R
J Pharmacol Exp Ther; 2006 Apr; 317(1):139-46. PubMed ID: 16394198
[TBL] [Abstract][Full Text] [Related]
12. Functional coupling of the human dopamine D2 receptor with G alpha i1, G alpha i2, G alpha i3 and G alpha o G proteins: evidence for agonist regulation of G protein selectivity.
Gazi L; Nickolls SA; Strange PG
Br J Pharmacol; 2003 Mar; 138(5):775-86. PubMed ID: 12642378
[TBL] [Abstract][Full Text] [Related]
13. Interactions of histamine H1-receptor agonists and antagonists with the human histamine H4-receptor.
Deml KF; Beermann S; Neumann D; Strasser A; Seifert R
Mol Pharmacol; 2009 Nov; 76(5):1019-30. PubMed ID: 19720730
[TBL] [Abstract][Full Text] [Related]
14. High constitutive activity and a G-protein-independent high-affinity state of the human histamine H(4)-receptor.
Schneider EH; Schnell D; Papa D; Seifert R
Biochemistry; 2009 Feb; 48(6):1424-38. PubMed ID: 19166345
[TBL] [Abstract][Full Text] [Related]
15. Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors.
Rouleau A; Ligneau X; Tardivel-Lacombe J; Morisset S; Gbahou F; Schwartz JC; Arrang JM
Br J Pharmacol; 2002 Jan; 135(2):383-92. PubMed ID: 11815373
[TBL] [Abstract][Full Text] [Related]
16. Similar apparent constitutive activity of human histamine H(2)-receptor fused to long and short splice variants of G(salpha).
Wenzel-Seifert K; Kelley MT; Buschauer A; Seifert R
J Pharmacol Exp Ther; 2001 Dec; 299(3):1013-20. PubMed ID: 11714890
[TBL] [Abstract][Full Text] [Related]
17. D2 dopamine receptor activation of potassium channels is selectively decoupled by Galpha-specific GoLoco motif peptides.
Webb CK; McCudden CR; Willard FS; Kimple RJ; Siderovski DP; Oxford GS
J Neurochem; 2005 Mar; 92(6):1408-18. PubMed ID: 15748159
[TBL] [Abstract][Full Text] [Related]
18. RGS-insensitive G-protein mutations to study the role of endogenous RGS proteins.
Fu Y; Zhong H; Nanamori M; Mortensen RM; Huang X; Lan K; Neubig RR
Methods Enzymol; 2004; 389():229-43. PubMed ID: 15313569
[TBL] [Abstract][Full Text] [Related]
19. Development of generic calcium imaging assay for monitoring Gi-coupled receptors and G-protein interaction.
Ueda T; Ugawa S; Ishida Y; Hondoh A; Shimada S
J Biomol Screen; 2009 Aug; 14(7):781-8. PubMed ID: 19541673
[TBL] [Abstract][Full Text] [Related]
20. Effects of partial agonists and Mg2+ ions on the interaction of M2 muscarinic acetylcholine receptor and G protein Galpha i1 subunit in the M2-Galpha i1 fusion protein.
Zhang Q; Okamura M; Guo ZD; Niwa S; Haga T
J Biochem; 2004 May; 135(5):589-96. PubMed ID: 15173197
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
