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5. Novel quinuclidine-based ligands for the muscarinic cholinergic receptor. Saunders J; Cassidy M; Freedman SB; Harley EA; Iversen LL; Kneen C; MacLeod AM; Merchant KJ; Snow RJ; Baker R J Med Chem; 1990 Apr; 33(4):1128-38. PubMed ID: 2319559 [TBL] [Abstract][Full Text] [Related]
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8. Design, synthesis, and neurochemical evaluation of 5-(3-alkyl-1,2,4- oxadiazol-5-yl)-1,4,5,6-tetrahydropyrimidines as M1 muscarinic receptor agonists. Dunbar PG; Durant GJ; Fang Z; Abuh YF; el-Assadi AA; Ngur DO; Periyasamy S; Hoss WP; Messer WS J Med Chem; 1993 Apr; 36(7):842-7. PubMed ID: 8464038 [TBL] [Abstract][Full Text] [Related]
9. Resolved pyrrolidine, piperidine, and perhydroazepine analogues of the muscarinic agent N-methyl-N-(1-methyl-4-pyrrolidino-2-butynyl)acetamide. Lundkvist JR; Vargas HM; Caldirola P; Ringdahl B; Hacksell U J Med Chem; 1990 Dec; 33(12):3182-9. PubMed ID: 2258904 [TBL] [Abstract][Full Text] [Related]
10. Novel functional M1 selective muscarinic agonists. 2. Synthesis and structure-activity relationships of 3-pyrazinyl-1,2,5,6-tetrahydro-1-methylpyridines. Construction of a molecular model for the M1 pharmacophore. Ward JS; Merritt L; Klimkowski VJ; Lamb ML; Mitch CH; Bymaster FP; Sawyer B; Shannon HE; Olesen PH; Honoré T J Med Chem; 1992 Oct; 35(22):4011-9. PubMed ID: 1433209 [TBL] [Abstract][Full Text] [Related]
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13. Synthesis and in vitro biological profile of all four isomers of the potent muscarinic agonist 3-(3-methyl-1,2,4-oxadiazol-5-yl)-1-azabicyclo[2.2.1]heptane. Showell GA; Baker R; Davis J; Hargreaves R; Freedman SB; Hoogsteen K; Patel S; Snow RJ J Med Chem; 1992 Mar; 35(5):911-6. PubMed ID: 1548680 [TBL] [Abstract][Full Text] [Related]
14. Synthesis and muscarinic activities of quinuclidin-3-yltriazole and -tetrazole derivatives. Wadsworth HJ; Jenkins SM; Orlek BS; Cassidy F; Clark MS; Brown F; Riley GJ; Graves D; Hawkins J; Naylor CB J Med Chem; 1992 Apr; 35(7):1280-90. PubMed ID: 1560440 [TBL] [Abstract][Full Text] [Related]
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16. A novel series of non-quaternary oxadiazoles acting as full agonists at muscarinic receptors. Freedman SB; Harley EA; Patel S; Newberry NR; Gilbert MJ; McKnight AT; Tang JK; Maguire JJ; Mudunkotuwa NT; Baker R Br J Pharmacol; 1990 Nov; 101(3):575-80. PubMed ID: 2076477 [TBL] [Abstract][Full Text] [Related]
17. Conformational aspects of the muscarinic receptor interactions of bicyclic isoxazole ester bioisosteres of arecoline. Lagersted A; Falch E; Ebert B; Krogsgaard-Larsen P Drug Des Discov; 1993; 9(3-4):237-50. PubMed ID: 8400005 [TBL] [Abstract][Full Text] [Related]
18. Synthesis and muscarinic activity of quinuclidinyl- and (1-azanorbornyl)pyrazine derivatives. Street LJ; Baker R; Book T; Reeve AJ; Saunders J; Willson T; Marwood RS; Patel S; Freedman SB J Med Chem; 1992 Jan; 35(2):295-305. PubMed ID: 1732546 [TBL] [Abstract][Full Text] [Related]
19. Recognition of cholinergic agonists by the muscarinic receptor. 1. Acetylcholine and other agonists with the NCCOCC backbone. Schulman JM; Sabio ML; Disch RL J Med Chem; 1983 Jun; 26(6):817-23. PubMed ID: 6854585 [TBL] [Abstract][Full Text] [Related]