128 related articles for article (PubMed ID: 20131817)
21. Replacement of the lactone moiety on podophyllotoxin and steganacin analogues with a 1,5-disubstituted 1,2,3-triazole via ruthenium-catalyzed click chemistry.
Imperio D; Pirali T; Galli U; Pagliai F; Cafici L; Canonico PL; Sorba G; Genazzani AA; Tron GC
Bioorg Med Chem; 2007 Nov; 15(21):6748-57. PubMed ID: 17765552
[TBL] [Abstract][Full Text] [Related]
22. Novel synthesis, cytotoxic evaluation, and structure-activity relationship studies of a series of alpha-alkylidene-gamma-lactones and lactams.
Janecki T; Błaszczyk E; Studzian K; Janecka A; Krajewska U; Rózalski M
J Med Chem; 2005 May; 48(10):3516-21. PubMed ID: 15887960
[TBL] [Abstract][Full Text] [Related]
23. Synthesis, solution equilibria and antiproliferative activity of copper(II) aminomethyltriazole and aminomethylthioxotriazoline complexes.
Gaccioli F; Franchi-Gazzola R; Lanfranchi M; Marchiò L; Metta G; Pellinghelli MA; Tardito S; Tegoni M
J Inorg Biochem; 2005 Aug; 99(8):1573-84. PubMed ID: 15953645
[TBL] [Abstract][Full Text] [Related]
24. Phase I trial of the cryptophycin analogue LY355703 administered as an intravenous infusion on a day 1 and 8 schedule every 21 days.
Stevenson JP; Sun W; Gallagher M; Johnson R; Vaughn D; Schuchter L; Algazy K; Hahn S; Enas N; Ellis D; Thornton D; O'Dwyer PJ
Clin Cancer Res; 2002 Aug; 8(8):2524-9. PubMed ID: 12171879
[TBL] [Abstract][Full Text] [Related]
25. Total synthesis and anti-tubulin activity of epi-c3 analogues of cryptophycin-24.
Buck SB; Huff JK; Himes RH; Georg GI
J Med Chem; 2004 Jul; 47(14):3697-9. PubMed ID: 15214797
[TBL] [Abstract][Full Text] [Related]
26. A practical total synthesis of hapalosin, a 12-membered cyclic depsipeptide with multidrug resistance-reversing activity, by employing improved segment coupling and macrolactonization.
Palomo C; Oiarbide M; García JM; González A; Pazos R; Odriozola JM; Bañuelos P; Tello M; Linden A
J Org Chem; 2004 Jun; 69(12):4126-34. PubMed ID: 15176838
[TBL] [Abstract][Full Text] [Related]
27. 1,5-Disubstituted 1,2,3-triazoles as cis-restricted analogues of combretastatin A-4: Synthesis, molecular modeling and evaluation as cytotoxic agents and inhibitors of tubulin.
Odlo K; Hentzen J; dit Chabert JF; Ducki S; Gani OA; Sylte I; Skrede M; Flørenes VA; Hansen TV
Bioorg Med Chem; 2008 May; 16(9):4829-38. PubMed ID: 18396050
[TBL] [Abstract][Full Text] [Related]
28. Homophymines B-E and A1-E1, a family of bioactive cyclodepsipeptides from the sponge Homophymia sp.
Zampella A; Sepe V; Bellotta F; Luciano P; D'Auria MV; Cresteil T; Debitus C; Petek S; Poupat C; Ahond A
Org Biomol Chem; 2009 Oct; 7(19):4037-44. PubMed ID: 19763308
[TBL] [Abstract][Full Text] [Related]
29. Inhibition of macromolecular synthesis by cryptophycin-52.
Subramanian B; Nakeff A; Media JE; Wiegand RA; Valeriote FA
Anticancer Drugs; 2002 Nov; 13(10):1061-8. PubMed ID: 12439340
[TBL] [Abstract][Full Text] [Related]
30. Synthesis of cryptophycin 52 using the sharpless asymmetric dihydroxylation: diol to epoxide transformation optimized for a base-sensitive substrate.
Liang J; Moher ED; Moore RE; Hoard DW
J Org Chem; 2000 May; 65(10):3143-7. PubMed ID: 10814209
[TBL] [Abstract][Full Text] [Related]
31. Incrementally increasing the length of a peptide backbone: effect on macrocyclisation efficiency.
Ahmed MI; Harper JB; Hunter L
Org Biomol Chem; 2014 Jul; 12(26):4598-601. PubMed ID: 24891254
[TBL] [Abstract][Full Text] [Related]
32. Acute vulvar vestibulitis occurring during chemotherapy with cryptophycin analogue LY355703.
De Pas TM; Mandalà M; Curigliano G; Peccatori F
Obstet Gynecol; 2000 Jun; 95(6 Pt 2):1030. PubMed ID: 10808018
[No Abstract] [Full Text] [Related]
33. Synthesis, 3D-QSAR, and docking studies of 1-phenyl-1H-1,2,3-triazoles as selective antagonists for beta3 over alpha1beta2gamma2 GABA receptors.
Alam MS; Huang J; Ozoe F; Matsumura F; Ozoe Y
Bioorg Med Chem; 2007 Aug; 15(15):5090-104. PubMed ID: 17544280
[TBL] [Abstract][Full Text] [Related]
34. Synthesis and properties of bioactive 2- and 3-amino-8-methyl-8H-quino[4,3,2-kl]acridine and 8,13-dimethyl-8H-quino[4,3,2-kl]acridinium salts.
Hutchinson I; McCarroll AJ; Heald RA; Stevens MF
Org Biomol Chem; 2004 Jan; 2(2):220-8. PubMed ID: 14737646
[TBL] [Abstract][Full Text] [Related]
35. Synthesis and biological activities of hapalosin derivatives with modification at the C12 position.
Kashihara N; To-e S; Nakamura K; Umezawa K; Yamamura S; Nishiyama S
Bioorg Med Chem Lett; 2000 Jan; 10(2):101-3. PubMed ID: 10673089
[TBL] [Abstract][Full Text] [Related]
36. Approaches for the synthesis of functionalized cryptophycins.
Sammet B; Bogner T; Nahrwold M; Weiss C; Sewald N
J Org Chem; 2010 Oct; 75(20):6953-60. PubMed ID: 20857920
[TBL] [Abstract][Full Text] [Related]
37. Total synthesis and biological evaluation of halipeptins A and D and analogues.
Nicolaou KC; Lizos DE; Kim DW; Schlawe D; de Noronha RG; Longbottom DA; Rodriquez M; Bucci M; Cirino G
J Am Chem Soc; 2006 Apr; 128(13):4460-70. PubMed ID: 16569024
[TBL] [Abstract][Full Text] [Related]
38. Cryptophycins-309, 249 and other cryptophycin analogs: preclinical efficacy studies with mouse and human tumors.
Liang J; Moore RE; Moher ED; Munroe JE; Al-awar RS; Hay DA; Varie DL; Zhang TY; Aikins JA; Martinelli MJ; Shih C; Ray JE; Gibson LL; Vasudevan V; Polin L; White K; Kushner J; Simpson C; Pugh S; Corbett TH
Invest New Drugs; 2005 Jun; 23(3):213-24. PubMed ID: 15868377
[TBL] [Abstract][Full Text] [Related]
39. Diversity-oriented asymmetric synthesis of hapalosin: construction of three small C9/C4/C3-modified hapalosin analogue libraries.
Dai CF; Cheng F; Xu HC; Ruan YP; Huang PQ
J Comb Chem; 2007; 9(3):386-94. PubMed ID: 17358084
[TBL] [Abstract][Full Text] [Related]
40. Annonaceous acetogenin mimics bearing a terminal lactam and their cytotoxicity against cancer cells.
Liu HX; Huang GR; Zhang HM; Wu JR; Yao ZJ
Bioorg Med Chem Lett; 2007 Jun; 17(12):3426-30. PubMed ID: 17433671
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
