BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

228 related articles for article (PubMed ID: 20144593)

  • 1. Synthesis and evaluation of novel analogues of vitamin B6 as reactivators of tabun and paraoxon inhibited acetylcholinesterase.
    Gaso-Sokac D; Katalinić M; Kovarik Z; Busić V; Kovac S
    Chem Biol Interact; 2010 Sep; 187(1-3):234-7. PubMed ID: 20144593
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Novel series of bispyridinium compounds bearing a (Z)-but-2-ene linker--synthesis and evaluation of their reactivation activity against tabun and paraoxon-inhibited acetylcholinesterase.
    Musilek K; Holas O; Kuca K; Jun D; Dohnal V; Opletalova V; Dolezal M
    Bioorg Med Chem Lett; 2007 Jun; 17(11):3172-6. PubMed ID: 17383875
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Pseudo-catalytic scavenging: searching for a suitable reactivator of phosphorylated butyrylcholinesterase.
    Kovarik Z; Katalinić M; Sinko G; Binder J; Holas O; Jung YS; Musilova L; Jun D; Kuca K
    Chem Biol Interact; 2010 Sep; 187(1-3):167-71. PubMed ID: 20206154
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Kinetic analysis of interactions of different sarin and tabun analogues with human acetylcholinesterase and oximes: is there a structure-activity relationship?
    Aurbek N; Herkert NM; Koller M; Thiermann H; Worek F
    Chem Biol Interact; 2010 Sep; 187(1-3):215-9. PubMed ID: 20105433
    [TBL] [Abstract][Full Text] [Related]  

  • 5. In vitro and in vivo evaluation of pyridinium oximes: mode of interaction with acetylcholinesterase, effect on tabun- and soman-poisoned mice and their cytotoxicity.
    Calić M; Vrdoljak AL; Radić B; Jelić D; Jun D; Kuca K; Kovarik Z
    Toxicology; 2006 Feb; 219(1-3):85-96. PubMed ID: 16332406
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Fluorinated pyridinium oximes as potential reactivators for acetylcholinesterases inhibited by paraoxon organophosphorus agent.
    Jeong HC; Park NJ; Chae CH; Musilek K; Kassa J; Kuca K; Jung YS
    Bioorg Med Chem; 2009 Sep; 17(17):6213-7. PubMed ID: 19665386
    [TBL] [Abstract][Full Text] [Related]  

  • 7. In vitro oxime reactivation of red blood cell acetylcholinesterase inhibited by methyl-paraoxon.
    Petroianu GA; Arafat K; Nurulain SM; Kuca K; Kassa J
    J Appl Toxicol; 2007; 27(2):168-75. PubMed ID: 17265452
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and evaluation of novel bis-pyridinium oximes as reactivators of DFP-inhibited acetylcholinesterase.
    Acharya J; Gupta AK; Dubey DK; Raza SK
    Eur J Med Chem; 2009 Mar; 44(3):1335-40. PubMed ID: 18396353
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Monoquaternary pyridinium salts with modified side chain-synthesis and evaluation on model of tabun- and paraoxon-inhibited acetylcholinesterase.
    Musilek K; Kucera J; Jun D; Dohnal V; Opletalova V; Kuca K
    Bioorg Med Chem; 2008 Sep; 16(17):8218-23. PubMed ID: 18676153
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Effective bisquaternary reactivators of tabun-inhibited AChE.
    Kuca K; Cabal J; Musilek K; Jun D; Bajgar J
    J Appl Toxicol; 2005; 25(6):491-5. PubMed ID: 16092078
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Interactions of oxime reactivators with diethylphosphoryl adducts of human acetylcholinesterase and its mutant derivatives.
    Grosfeld H; Barak D; Ordentlich A; Velan B; Shafferman A
    Mol Pharmacol; 1996 Sep; 50(3):639-49. PubMed ID: 8794905
    [TBL] [Abstract][Full Text] [Related]  

  • 12. In silico pharmacophore model for tabun-inhibited acetylcholinesterase reactivators: a study of their stereoelectronic properties.
    Bhattacharjee AK; Kuca K; Musilek K; Gordon RK
    Chem Res Toxicol; 2010 Jan; 23(1):26-36. PubMed ID: 20028185
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Monooxime reactivators of acetylcholinesterase with (E)-but-2-ene linker: preparation and reactivation of tabun- and paraoxon-inhibited acetylcholinesterase.
    Musilek K; Holas O; Jun D; Dohnal V; Gunn-Moore F; Opletalova V; Dolezal M; Kuca K
    Bioorg Med Chem; 2007 Nov; 15(21):6733-41. PubMed ID: 17764957
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Quaternary salts of 4,3' and 4,4' bis-pyridinium monooximes: synthesis and biological activity.
    Chennamaneni SR; Vobalaboina V; Garlapati A
    Bioorg Med Chem Lett; 2005 Jun; 15(12):3076-80. PubMed ID: 15908205
    [TBL] [Abstract][Full Text] [Related]  

  • 15. New oxime reactivators connected with CH2O(CH2)nOCH2 linker and their reactivation potency for organophosphorus agents-inhibited acetylcholinesterase.
    Yang GY; Oh KA; Park NJ; Jung YS
    Bioorg Med Chem; 2007 Dec; 15(24):7704-10. PubMed ID: 17869525
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis of asymmetrical bispyridinium compounds bearing cyano-moiety and evaluation of their reactivation activity against tabun and paraoxon-inhibited acetylcholinesterase.
    Musilek K; Holas O; Kuca K; Jun D; Dohnal V; Dolezal M
    Bioorg Med Chem Lett; 2006 Nov; 16(21):5673-6. PubMed ID: 16934462
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Kinetic analysis of reactivation and aging of human acetylcholinesterase inhibited by different phosphoramidates.
    Worek F; Aurbek N; Koller M; Becker C; Eyer P; Thiermann H
    Biochem Pharmacol; 2007 Jun; 73(11):1807-17. PubMed ID: 17382909
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Reactivation of DFP- and paraoxon-inhibited acetylcholinesterases by pyridinium oximes.
    Oh KA; Park NJ; Park NS; Kuca K; Jun D; Jung YS
    Chem Biol Interact; 2008 Sep; 175(1-3):365-7. PubMed ID: 18565503
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Evaluation of monoquaternary pyridinium oximes potency to reactivate tabun-inhibited human acetylcholinesterase.
    Odzak R; Calić M; Hrenar T; Primozic I; Kovarik Z
    Toxicology; 2007 Apr; 233(1-3):85-96. PubMed ID: 16962227
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Oximes: Reactivators of phosphorylated acetylcholinesterase and antidotes in therapy against tabun poisoning.
    Kovarik Z; Calić M; Sinko G; Bosak A; Berend S; Vrdoljak AL; Radić B
    Chem Biol Interact; 2008 Sep; 175(1-3):173-9. PubMed ID: 18501341
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 12.