107 related articles for article (PubMed ID: 20206195)
1. Synthesis of regioisomeric 17beta-N-phenylpyrazolyl steroid derivatives and their inhibitory effect on 17alpha-hydroxylase/C(17,20)-lyase.
Iványi Z; Wölfling J; Görbe T; Szécsi M; Wittmann T; Schneider G
Steroids; 2010 Jun; 75(6):450-6. PubMed ID: 20206195
[TBL] [Abstract][Full Text] [Related]
2. Steroselective synthesis of some steroidal oxazolines, as novel potential inhibitors of 17alpha-hydroxylase-C17,20-lyase.
Ondré D; Wölfling J; Tóth I; Szécsi M; Julesz J; Schneider G
Steroids; 2009; 74(13-14):1025-32. PubMed ID: 19666042
[TBL] [Abstract][Full Text] [Related]
3. Neighboring group participation Part 17 Stereoselective synthesis of some steroidal 2-oxazolidones, as novel potential inhibitors of 17alpha-hydroxylase-C(17,20)-lyase.
Ondré D; Wölfling J; Iványi Z; Schneider G; Tóth I; Szécsi M; Julesz J
Steroids; 2008 Dec; 73(14):1375-84. PubMed ID: 18652838
[TBL] [Abstract][Full Text] [Related]
4. Stereoselective synthesis of some 17beta-dihydrooxazinyl steroids, as novel presumed inhibitors of 17alpha-hydroxylase-C17,20-lyase.
Wölfling J; Oravecz EA; Ondré D; Mernyák E; Schneider G; Tóth I; Szécsi M; Julesz J
Steroids; 2006 Sep; 71(9):809-16. PubMed ID: 16814336
[TBL] [Abstract][Full Text] [Related]
5. Novel series of 17β-pyrazolylandrosta-5,16-diene derivatives and their inhibitory effect on 17α-hydroxylase/C(17,20)-lyase.
Iványi Z; Szabó N; Wölfling J; Szécsi M; Julesz J; Schneider G
Steroids; 2012 Sep; 77(11):1152-9. PubMed ID: 22809751
[TBL] [Abstract][Full Text] [Related]
6. Synthesis of methoxycarbonylpyrazolylandrostene derivatives, and their potential inhibitory effect on androgen biosynthesis and cell proliferation.
Szabó N; Iványi Z; Szécsi M; Julesz J; Mernyák E; Huber J; Wölfling J; Minorics R; Zupkó I; Schneider G
Steroids; 2015 Jun; 98():143-52. PubMed ID: 25804762
[TBL] [Abstract][Full Text] [Related]
7. 17-Imidazolyl, pyrazolyl, and isoxazolyl androstene derivatives. Novel steroidal inhibitors of human cytochrome C17,20-lyase (P450(17 alpha).
Ling YZ; Li JS; Liu Y; Kato K; Klus GT; Brodie A
J Med Chem; 1997 Sep; 40(20):3297-304. PubMed ID: 9379450
[TBL] [Abstract][Full Text] [Related]
8. Determination of 17α-hydroxylase-C17,20-lyase (P45017α) enzyme activities and their inhibition by selected steroidal picolyl and picolinylidene compounds.
Szabó N; Ajduković JJ; Djurendić EA; Sakač MN; Ignáth I; Gardi J; Mahmoud G; Klisurić OR; Jovanović-Šanta S; Penov Gaši KM; Szécsi M
Acta Biol Hung; 2015 Mar; 66(1):41-51. PubMed ID: 25740437
[TBL] [Abstract][Full Text] [Related]
9. Synthesis of novel 17-triazolyl-androst-5-en-3-ol epimers via Cu(I)-catalyzed azide-alkyne cycloaddition and their inhibitory effect on 17α-hydroxylase/C
Kiss A; Herman BE; Görbe T; Mernyák E; Molnár B; Wölfling J; Szécsi M; Schneider G
Steroids; 2018 Jul; 135():79-91. PubMed ID: 29577953
[TBL] [Abstract][Full Text] [Related]
10. Synthesis, biochemical evaluation and rationalisation of the inhibitory activity of a range of phenyl alkyl imidazole-based compounds as potent inhibitors of the enzyme complex 17alpha-hydroxylase/17,20-lyase (P450(17alpha)).
Owen CP; Shahid I; Olusanjo MS; Patel CH; Dhanani S; Ahmed S
J Steroid Biochem Mol Biol; 2008 Jul; 111(1-2):117-27. PubMed ID: 18620055
[TBL] [Abstract][Full Text] [Related]
11. Neighboring group participation. Part 15. Stereoselective synthesis of some steroidal tetrahydrooxazin-2-ones, as novel presumed inhibitors of human 5alpha-reductase.
Wölfling J; Hackler L; Mernyák E; Schneider G; Tóth I; Szécsi M; Julesz J; Sohár P; Csámpai A
Steroids; 2004 Jul; 69(7):451-60. PubMed ID: 15246775
[TBL] [Abstract][Full Text] [Related]
12. Synthesis and biochemical evaluation of a range of (4-substituted phenyl)sulfonate derivatives of 4-hydroxybenzyl imidazole-based compounds as potent inhibitors of 17alpha-hydroxylase/17,20-lyase (P45017alpha) derived from rat testicular microsomes.
Owen CP; Shahid I; Lee WY; Ahmed S
Bioorg Med Chem Lett; 2010 Sep; 20(17):5345-8. PubMed ID: 20675132
[TBL] [Abstract][Full Text] [Related]
13. Synthesis of D-ring-substituted (5'R)- and (5'S)-17β-pyrazolinylandrostene epimers and comparison of their potential anticancer activities.
Iványi Z; Szabó N; Huber J; Wölfling J; Zupkó I; Szécsi M; Wittmann T; Schneider G
Steroids; 2012 Apr; 77(5):566-74. PubMed ID: 22342542
[TBL] [Abstract][Full Text] [Related]
14. The 16,17-double bond is needed for irreversible inhibition of human cytochrome p45017alpha by abiraterone (17-(3-pyridyl)androsta-5, 16-dien-3beta-ol) and related steroidal inhibitors.
Jarman M; Barrie SE; Llera JM
J Med Chem; 1998 Dec; 41(27):5375-81. PubMed ID: 9876107
[TBL] [Abstract][Full Text] [Related]
15. Synthesis and biochemical evaluation of a range of sulfonated derivatives of 4-hydroxybenzyl imidazole as highly potent inhibitors of rat testicular 17alpha-hydroxylase/17,20-lyase (P-450(17alpha)).
Ahmed S; Shahid I; Dhanani S; Owen CP
Bioorg Med Chem Lett; 2009 Aug; 19(16):4698-701. PubMed ID: 19608417
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and evaluation of 17-aliphatic heterocycle-substituted steroidal inhibitors of 17alpha-hydroxylase/C17-20-lyase (P450 17).
Hartmann RW; Hector M; Wachall BG; Palusczak A; Palzer M; Huch V; Veith M
J Med Chem; 2000 Nov; 43(23):4437-45. PubMed ID: 11087568
[TBL] [Abstract][Full Text] [Related]
17. An efficient approach to novel 17-5'-(1',2',4')-oxadiazolyl androstenes via the cyclodehydration of cytotoxic O-steroidacylamidoximes, and an evaluation of their inhibitory action on 17α-hydroxylase/C₁₇,₂₀-lyase.
Kovács D; Wölfling J; Szabó N; Szécsi M; Kovács I; Zupkó I; Frank E
Eur J Med Chem; 2013; 70():649-60. PubMed ID: 24211641
[TBL] [Abstract][Full Text] [Related]
18. Synthesis and evaluation of pregnane derivatives as inhibitors of human testicular 17 alpha-hydroxylase/C17,20-lyase.
Li JS; Li Y; Son C; Brodie AM
J Med Chem; 1996 Oct; 39(21):4335-9. PubMed ID: 8863811
[TBL] [Abstract][Full Text] [Related]
19. Synthesis, biochemical evaluation of a range of potent 4-substituted phenyl alkyl imidazole-based inhibitors of the enzyme complex 17alpha-Hydroxylase/17,20-Lyase (P45017alpha).
Shahid I; Patel CH; Dhanani S; Owen CP; Ahmed S
J Steroid Biochem Mol Biol; 2008 May; 110(1-2):18-29. PubMed ID: 18407491
[TBL] [Abstract][Full Text] [Related]
20. Efficient access to novel androsteno-17-(1',3',4')-oxadiazoles and 17β-(1',3',4')-thiadiazoles via N-substituted hydrazone and N,N'-disubstituted hydrazine intermediates, and their pharmacological evaluation in vitro.
Kovács D; Wölfling J; Szabó N; Szécsi M; Minorics R; Zupkó I; Frank É
Eur J Med Chem; 2015 Jun; 98():13-29. PubMed ID: 25993309
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]