BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

149 related articles for article (PubMed ID: 20335038)

  • 1. 'Click chemistry' synthesis of a library of 1,2,3-triazole-substituted galactose derivatives and their evaluation against Trypanosoma cruzi and its cell surface trans-sialidase.
    Carvalho I; Andrade P; Campo VL; Guedes PM; Sesti-Costa R; Silva JS; Schenkman S; Dedola S; Hill L; Rejzek M; Nepogodiev SA; Field RA
    Bioorg Med Chem; 2010 Apr; 18(7):2412-27. PubMed ID: 20335038
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design, synthesis and the effect of 1,2,3-triazole sialylmimetic neoglycoconjugates on Trypanosoma cruzi and its cell surface trans-sialidase.
    Campo VL; Sesti-Costa R; Carneiro ZA; Silva JS; Schenkman S; Carvalho I
    Bioorg Med Chem; 2012 Jan; 20(1):145-56. PubMed ID: 22154559
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Binding of triazole-linked galactosyl arylsulfonamides to galectin-3 affects Trypanosoma cruzi cell invasion.
    Marchiori MF; Riul TB; Oliveira Bortot L; Andrade P; Junqueira GG; Foca G; Doti N; Ruvo M; Dias-Baruffi M; Carvalho I; Campo VL
    Bioorg Med Chem; 2017 Nov; 25(21):6049-6059. PubMed ID: 29032929
    [TBL] [Abstract][Full Text] [Related]  

  • 4. 1,2,3-Triazole-based analogue of benznidazole displays remarkable activity against Trypanosoma cruzi.
    de Andrade P; Galo OA; Carvalho MR; Lopes CD; Carneiro ZA; Sesti-Costa R; de Melo EB; Silva JS; Carvalho I
    Bioorg Med Chem; 2015 Nov; 23(21):6815-26. PubMed ID: 26476667
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Design, synthesis and enzymatic evaluation of 3-O-substituted aryl β-D-galactopyranosides as inhibitors of Trypanosoma cruzi trans-sialidase.
    Silva BL; S Filho JD; Andrade P; Carvalho I; Alves RJ
    Bioorg Med Chem Lett; 2014 Sep; 24(18):4529-4532. PubMed ID: 25149510
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Naphthoquinoidal [1,2,3]-triazole, a new structural moiety active against Trypanosoma cruzi.
    da Silva EN; Menna-Barreto RF; Pinto Mdo C; Silva RS; Teixeira DV; de Souza MC; De Simone CA; De Castro SL; Ferreira VF; Pinto AV
    Eur J Med Chem; 2008 Aug; 43(8):1774-80. PubMed ID: 18045742
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis, molecular docking and biological evaluation of novel phthaloyl derivatives of 3-amino-3-aryl propionic acids as inhibitors of Trypanosoma cruzi trans-sialidase.
    Kashif M; Chacón-Vargas KF; López-Cedillo JC; Nogueda-Torres B; Paz-González AD; Ramírez-Moreno E; Agusti R; Uhrig ML; Reyes-Arellano A; Peralta-Cruz J; Ashfaq M; Rivera G
    Eur J Med Chem; 2018 Aug; 156():252-268. PubMed ID: 30006170
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Trypanosoma cruzi trans-sialidase alternative substrates: Study of the effect of substitution in C-6 in benzyl β-lactoside.
    Morrone-Pozzuto P; Uhrig ML; Agusti R
    Carbohydr Res; 2019 May; 478():33-45. PubMed ID: 31054381
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis of PEGylated lactose analogs for inhibition studies on T.cruzi trans-sialidase.
    Giorgi ME; Ratier L; Agusti R; Frasch AC; de Lederkremer RM
    Glycoconj J; 2010 Jul; 27(5):549-59. PubMed ID: 20645127
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis and in vitro and in silico studies of 1H- and 2H-1,2,3-triazoles as antichagasic agents.
    Silva TB; Ji KNK; Petzold Pauli F; Galvão RMS; Faria AFM; Bello ML; Resende JALC; Campos VR; Forezi LDSM; da Silva FC; Faria RX; Ferreira VF
    Bioorg Chem; 2021 Nov; 116():105250. PubMed ID: 34469833
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis, activity, and molecular modeling studies of 1,2,3-triazole derivatives from natural phenylpropanoids as new trypanocidal agents.
    de Souza TB; Caldas IS; Paula FR; Rodrigues CC; Carvalho DT; Dias DF
    Chem Biol Drug Des; 2020 Jan; 95(1):124-129. PubMed ID: 31569301
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Recent developments in trans-sialidase inhibitors of Trypanosoma cruzi.
    Kashif M; Moreno-Herrera A; Lara-Ramirez EE; Ramírez-Moreno E; Bocanegra-García V; Ashfaq M; Rivera G
    J Drug Target; 2017 Jul; 25(6):485-498. PubMed ID: 28140698
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Effect of 4-amino-3-nitrobenzoic acid on the expression level of the trans-sialidase gene in Trypanosoma cruzi epimastigotes.
    Vázquez-Jiménez LK; Paz-González AD; Kashif M; Juárez-Rendón KJ; Nogueda-Torres B; Bocanegra-García V; Rivera G
    Pak J Pharm Sci; 2019 Mar; 32(2 (Supplementary)):825-829. PubMed ID: 31103978
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Continuous nonradioactive method for screening trypanosomal trans-sialidase activity and its inhibitors.
    Sartor PA; Agusti R; Leguizamón MS; Campetella O; de Lederkremer RM
    Glycobiology; 2010 Aug; 20(8):982-90. PubMed ID: 20375068
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Trypanosoma cruzi trans-sialidase. A tool for the synthesis of sialylated oligosaccharides.
    Agusti R; Gallo-Rodriguez C; de Lederkremer RM
    Carbohydr Res; 2019 Jun; 479():48-58. PubMed ID: 31132642
    [TBL] [Abstract][Full Text] [Related]  

  • 16. The synthesis and kinetic evaluation of aryl α-aminophosphonates as novel inhibitors of T. cruzi trans-sialidase.
    Chen Z; Marcé P; Resende R; Alzari PM; Frasch AC; van den Elsen JMH; Crennell SJ; Watts AG
    Eur J Med Chem; 2018 Oct; 158():25-33. PubMed ID: 30199703
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Design and synthesis of aryloxyethyl thiocyanate derivatives as potent inhibitors of Trypanosoma cruzi proliferation.
    Szajnman SH; Yan W; Bailey BN; Docampo R; Elhalem E; Rodriguez JB
    J Med Chem; 2000 May; 43(9):1826-40. PubMed ID: 10794699
    [TBL] [Abstract][Full Text] [Related]  

  • 18. α-Selective glycosylation affords mucin-related GalNAc amino acids and diketopiperazines active on Trypanosoma cruzi.
    Martins-Teixeira MB; Campo VL; Biondo M; Sesti-Costa R; Carneiro ZA; Silva JS; Carvalho I
    Bioorg Med Chem; 2013 Apr; 21(7):1978-87. PubMed ID: 23415086
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Temperature differences for trans-glycosylation and hydrolysis reaction reveal an acceptor binding site in the catalytic mechanism of Trypanosoma cruzi trans-sialidase.
    Ribeirão M; Pereira-Chioccola VL; Eichinger D; Rodrigues MM; Schenkman S
    Glycobiology; 1997 Dec; 7(8):1237-46. PubMed ID: 9455925
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Enzymatically inactive trans-sialidase from Trypanosoma cruzi binds sialyl and beta-galactopyranosyl residues in a sequential ordered mechanism.
    Todeschini AR; Dias WB; Girard MF; Wieruszeski JM; Mendonça-Previato L; Previato JO
    J Biol Chem; 2004 Feb; 279(7):5323-8. PubMed ID: 14634017
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.