81 related articles for article (PubMed ID: 20462217)
1. Rational design of a topical androgen receptor antagonist for the suppression of sebum production with properties suitable for follicular delivery.
Mitchell LH; Johnson TR; Lu GW; Du D; Datta K; Grzemski F; Shanmugasundaram V; Spence J; Wade K; Wang Z; Sun K; Lin K; Hu LY; Sexton K; Raheja N; Kostlan C; Pocalyko D
J Med Chem; 2010 Jun; 53(11):4422-7. PubMed ID: 20462217
[TBL] [Abstract][Full Text] [Related]
2. 4-(Alkylthio)- and 4-(arylthio)-benzonitrile derivatives as androgen receptor antagonists for the topical suppression of sebum production.
Mitchell L; Wang Z; Hu LY; Kostlan C; Carroll M; Dettling D; Du D; Pocalyko D; Wade K
Bioorg Med Chem Lett; 2009 Mar; 19(5):1310-3. PubMed ID: 19201190
[TBL] [Abstract][Full Text] [Related]
3. (1R,2S)-4-(2-cyano-cyclohexyl-oxy)-2-trifluoromethyl-benzonitrile, a potent androgen receptor antagonist for stimulating hair growth and reducing sebum production.
Hu LY; Du D; Hoffman J; Smith Y; Fedij V; Kostlan C; Johnson TR; Huang Y; Kesten S; Harter W; Yue WS; Li JJ; Barvian N; Mitchell L; Lei HJ; Lefker B; Carroll M; Dettling D; Krieger-Burke T; Samas B; Yalamanchili R; Lapham K; Pocalyko D; Sliskovic D; Ciotti S; Stoller B; Hena MA; Ding Q; Maiti SN; Stier M; Welgus H
Bioorg Med Chem Lett; 2007 Nov; 17(21):5983-8. PubMed ID: 17827000
[TBL] [Abstract][Full Text] [Related]
4. Pantolactams as androgen receptor antagonists for the topical suppression of sebum production.
Sexton KE; Barrett S; Bridgwood K; Carroll M; Dettling D; Du D; Fakhoury S; Fedij V; Hu LY; Kostlan C; Pocalyko D; Raheja N; Smith Y; Shanmugasundaram V; Wade K
Bioorg Med Chem Lett; 2011 Sep; 21(18):5230-3. PubMed ID: 21831636
[TBL] [Abstract][Full Text] [Related]
5. Diphenyl ethers as androgen receptor antagonists for the topical suppression of sebum production.
Mitchell LH; Hu LY; Nguyen M; Fakhoury S; Smith Y; Iula D; Kostlan C; Carroll M; Dettling D; Du D; Pocalyko D; Wade K; Lefker B
Bioorg Med Chem Lett; 2009 Apr; 19(8):2176-8. PubMed ID: 19286380
[TBL] [Abstract][Full Text] [Related]
6. Preparation of 4-aryl-2-trifluoromethylbenzonitrile derivatives as androgen receptor antagonists for topical suppression of sebum production.
Van Camp JA; Hu LY; Kostlan C; Lefker B; Li J; Mitchell L; Wang Z; Yue WS; Carroll M; Dettling D; Du D; Pocalyko D; Wade K
Bioorg Med Chem Lett; 2007 Oct; 17(20):5529-32. PubMed ID: 17764935
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and biological evaluation of amino-pyridines as androgen receptor antagonists for stimulating hair growth and reducing sebum production.
Hu LY; Lei HJ; Du D; Johnson TR; Fedij V; Kostlan C; Yue WS; Lovdahl M; Li JJ; Carroll M; Dettling D; Asbill J; Fan C; Wade K; Pocalyko D; Lapham K; Yalamanchili R; Samas B; Vrieze D; Ciotti S; Krieger-Burke T; Sliskovic D; Welgus H
Bioorg Med Chem Lett; 2007 Oct; 17(20):5693-7. PubMed ID: 17766112
[TBL] [Abstract][Full Text] [Related]
8. Rational design and synthesis of 4-((1R,2R)-2-hydroxycyclohexyl)-2(trifluoromethyl)benzonitrile (PF-998425), a novel, nonsteroidal androgen receptor antagonist devoid of phototoxicity for dermatological indications.
Li JJ; Iula DM; Nguyen MN; Hu LY; Dettling D; Johnson TR; Du DY; Shanmugasundaram V; Van Camp JA; Wang Z; Harter WG; Yue WS; Boys ML; Wade KJ; Drummond EM; Samas BM; Lefker BA; Hoge GS; Lovdahl MJ; Asbill J; Carroll M; Meade MA; Ciotti SM; Krieger-Burke T
J Med Chem; 2008 Nov; 51(21):7010-4. PubMed ID: 18921992
[TBL] [Abstract][Full Text] [Related]
9. Deposition of salicylic acid into hamster sebaceous.
Motwani MR; Rhein LD; Zatz JL
J Cosmet Sci; 2004; 55(6):519-31. PubMed ID: 15645108
[TBL] [Abstract][Full Text] [Related]
10. Local inhibition of sebaceous gland growth by topically applied RU 58841.
Matias JR; Gaillard M
Ann N Y Acad Sci; 1995 Jun; 761():56-65. PubMed ID: 7625751
[TBL] [Abstract][Full Text] [Related]
11. Comparison of artificial sebum with human and hamster sebum samples.
Lu GW; Valiveti S; Spence J; Zhuang C; Robosky L; Wade K; Love A; Hu LY; Pole D; Mollan M
Int J Pharm; 2009 Feb; 367(1-2):37-43. PubMed ID: 18929636
[TBL] [Abstract][Full Text] [Related]
12. Inhibition of sebum production and Propionibacterium acnes lipase activity by fullerenol, a novel polyhydroxylated fullerene: potential as a therapeutic reagent for acne.
Inui S; Aoshima H; Ito M; Kobuko K; Itami S
J Cosmet Sci; 2012; 63(4):259-65. PubMed ID: 23193890
[TBL] [Abstract][Full Text] [Related]
13. Effects of sex steroid deprivation/administration on hair growth and skin sebum production in transsexual males and females.
Giltay EJ; Gooren LJ
J Clin Endocrinol Metab; 2000 Aug; 85(8):2913-21. PubMed ID: 10946903
[TBL] [Abstract][Full Text] [Related]
14. Applications and limitations of lipid nanoparticles in dermal and transdermal drug delivery via the follicular route.
Lauterbach A; Müller-Goymann CC
Eur J Pharm Biopharm; 2015 Nov; 97(Pt A):152-63. PubMed ID: 26144664
[TBL] [Abstract][Full Text] [Related]
15. The pilosebaceous unit: a pivotal route for topical drug delivery.
Agarwal R; Katare OP; Vyas SP
Methods Find Exp Clin Pharmacol; 2000 Mar; 22(2):129-33. PubMed ID: 10849897
[TBL] [Abstract][Full Text] [Related]
16. Biological properties of androgen receptor pure antagonist for treatment of castration-resistant prostate cancer: optimization from lead compound to CH5137291.
Kawata H; Arai S; Nakagawa T; Ishikura N; Nishimoto A; Yoshino H; Shiraishi T; Tachibana K; Nakamura R; Sato H
Prostate; 2011 Sep; 71(12):1344-56. PubMed ID: 21308717
[TBL] [Abstract][Full Text] [Related]
17. [Effect of topical retinoid therapy on seborrhea using iontophoresis].
Knor T
Med Arh; 2003; 57(5-6):295-8. PubMed ID: 15022582
[TBL] [Abstract][Full Text] [Related]
18. A novel deformable liposomal hydrogel loaded with a SREBP-1-inhibiting polypeptide for reducing sebum synthesis in golden hamster model.
Lv Z; Bao H; Zhu M; Xie Y; Tang H; Miao D; Guo X; Zhai X; Wang S; Chen H; Cong D; Liu X; Pei J
Eur J Pharm Sci; 2023 Aug; 187():106483. PubMed ID: 37268093
[TBL] [Abstract][Full Text] [Related]
19. Topical minoxidil does not act as an antiandrogen in the flank organ of the golden Syrian hamster.
Nuck BA; Fogelson SL; Lucky AW
Arch Dermatol; 1987 Jan; 123(1):59-61. PubMed ID: 3800423
[TBL] [Abstract][Full Text] [Related]
20. Effect of topical cyproterone acetate on sebum excretion in man.
Bingham KD; Low M; Wyatt EH
Lancet; 1979 Aug; 2(8137):304-5. PubMed ID: 88632
[No Abstract] [Full Text] [Related]
[Next] [New Search]