BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

157 related articles for article (PubMed ID: 20501662)

  • 1. Identification of novel specific allosteric modulators of the glycine receptor using phage display.
    Tipps ME; Lawshe JE; Ellington AD; Mihic SJ
    J Biol Chem; 2010 Jul; 285(30):22840-5. PubMed ID: 20501662
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Identification and characterization of heptapeptide modulators of the glycine receptor.
    Cornelison GL; Pflanz NC; Tipps ME; Mihic SJ
    Eur J Pharmacol; 2016 Jun; 780():252-9. PubMed ID: 27038522
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Positive allosteric modulators differentially affect full versus partial agonist activation of the glycine receptor.
    Kirson D; Todorovic J; Mihic SJ
    J Pharmacol Exp Ther; 2012 Jul; 342(1):61-70. PubMed ID: 22473615
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Effects of a mutation in the TM2-TM3 linker region of the glycine receptor alpha1 subunit on gating and allosteric modulation.
    Dupre ML; Broyles JM; Mihic SJ
    Brain Res; 2007 Jun; 1152():1-9. PubMed ID: 17434460
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Interactions between Zinc and Allosteric Modulators of the Glycine Receptor.
    Cornelison GL; Daszkowski AW; Pflanz NC; Mihic SJ
    J Pharmacol Exp Ther; 2017 Apr; 361(1):1-8. PubMed ID: 28087784
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Molecular sites for the positive allosteric modulation of glycine receptors by endocannabinoids.
    Yévenes GE; Zeilhofer HU
    PLoS One; 2011; 6(8):e23886. PubMed ID: 21901142
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Glucose is a positive modulator for the activation of human recombinant glycine receptors.
    Breitinger U; Raafat KM; Breitinger HG
    J Neurochem; 2015 Sep; 134(6):1055-66. PubMed ID: 26118987
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Identification of Positive Allosteric Modulators of Glycine Receptors from a High-Throughput Screen Using a Fluorescent Membrane Potential Assay.
    Stead C; Brown A; Adams C; Nickolls SJ; Young G; Kammonen J; Pryde D; Cawkill D
    J Biomol Screen; 2016 Dec; 21(10):1042-1053. PubMed ID: 27412533
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Anesthetic and ethanol effects on spontaneously opening glycine receptor channels.
    Beckstead MJ; Phelan R; Trudell JR; Bianchini MJ; Mihic SJ
    J Neurochem; 2002 Sep; 82(6):1343-51. PubMed ID: 12354281
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Mapping a molecular link between allosteric inhibition and activation of the glycine receptor.
    Miller PS; Topf M; Smart TG
    Nat Struct Mol Biol; 2008 Oct; 15(10):1084-93. PubMed ID: 18806798
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Allosteric modulation of the glycine receptor activated by agonists differing in efficacy.
    Farley NM; Mihic SJ
    Brain Res; 2015 May; 1606():95-101. PubMed ID: 25721789
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Single-channel analysis of ethanol enhancement of glycine receptor function.
    Welsh BT; Goldstein BE; Mihic SJ
    J Pharmacol Exp Ther; 2009 Jul; 330(1):198-205. PubMed ID: 19380602
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Molecular pharmacology of the glycine receptor chloride channel.
    Webb TI; Lynch JW
    Curr Pharm Des; 2007; 13(23):2350-67. PubMed ID: 17692006
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Alanine-scanning mutagenesis in the signature disulfide loop of the glycine receptor alpha 1 subunit: critical residues for activation and modulation.
    Schofield CM; Trudell JR; Harrison NL
    Biochemistry; 2004 Aug; 43(31):10058-63. PubMed ID: 15287733
    [TBL] [Abstract][Full Text] [Related]  

  • 15. In vitro interaction of the glycine receptor with the leptin receptor.
    Leite JF; Gribble B; Randolph N; Cascio M
    Physiol Behav; 2002 Dec; 77(4-5):565-9. PubMed ID: 12527000
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Identification of N-acyl amino acids that are positive allosteric modulators of glycine receptors.
    Gallagher CI; Sheipouri D; Shimmon S; Rawling T; Vandenberg RJ
    Biochem Pharmacol; 2020 Oct; 180():114117. PubMed ID: 32579961
    [TBL] [Abstract][Full Text] [Related]  

  • 17. A System for Assessing Dual Action Modulators of Glycine Transporters and Glycine Receptors.
    Sheipouri D; Gallagher CI; Shimmon S; Rawling T; Vandenberg RJ
    Biomolecules; 2020 Nov; 10(12):. PubMed ID: 33266066
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Loop 2 structure in glycine and GABA(A) receptors plays a key role in determining ethanol sensitivity.
    Perkins DI; Trudell JR; Crawford DK; Asatryan L; Alkana RL; Davies DL
    J Biol Chem; 2009 Oct; 284(40):27304-14. PubMed ID: 19656948
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Structure and Pharmacologic Modulation of Inhibitory Glycine Receptors.
    Burgos CF; Yévenes GE; Aguayo LG
    Mol Pharmacol; 2016 Sep; 90(3):318-25. PubMed ID: 27401877
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Mutations within the agonist-binding site convert the homomeric alpha1 glycine receptor into a Zn2+-activated chloride channel.
    Grudzinska J; Schumann T; Schemm R; Betz H; Laube B
    Channels (Austin); 2008; 2(1):13-8. PubMed ID: 18690053
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.