156 related articles for article (PubMed ID: 20570156)
1. Synthesis and inhibitory activities of novel C-3 substituted azafagomines: a new type of selective inhibitors of α-L-fucosidases.
Moreno-Clavijo E; Carmona AT; Moreno-Vargas AJ; Rodríguez-Carvajal MA; Robina I
Bioorg Med Chem; 2010 Jul; 18(13):4648-60. PubMed ID: 20570156
[TBL] [Abstract][Full Text] [Related]
2. Synthesis of novel pyrrolidine 3,4-diol derivatives as inhibitors of alpha-L-fucosidases.
Moreno-Clavijo E; Carmona AT; Vera-Ayoso Y; Moreno-Vargas AJ; Bello C; Vogel P; Robina I
Org Biomol Chem; 2009 Mar; 7(6):1192-202. PubMed ID: 19262940
[TBL] [Abstract][Full Text] [Related]
3. Stereoselective synthesis of (2S,3S,4R,5S)-5-methylpyrrolidine-3,4-diol derivatives that are highly selective alpha-L-fucosidase inhibitors.
Moreno-Vargas AJ; Carmona AT; Mora F; Vogel P; Robina I
Chem Commun (Camb); 2005 Oct; (39):4949-51. PubMed ID: 16205810
[TBL] [Abstract][Full Text] [Related]
4. Synthesis and evaluation of glycosidase inhibitory activity of N-butyl 1-deoxy-D-gluco-homonojirimycin and N-butyl 1-deoxy-L-ido-homonojirimycin.
Markad SD; Karanjule NS; Sharma T; Sabharwal SG; Dhavale DD
Bioorg Med Chem; 2006 Aug; 14(16):5535-9. PubMed ID: 16682208
[TBL] [Abstract][Full Text] [Related]
5. A concise synthesis of N-substituted fagomine derivatives and the systematic exploration of their α-glycosidase inhibition.
Jiang FX; Liu QZ; Zhao D; Luo CT; Guo CP; Ye WC; Luo C; Chen H
Eur J Med Chem; 2014 Apr; 77():211-22. PubMed ID: 24642564
[TBL] [Abstract][Full Text] [Related]
6. Asymmetric synthesis of the L-fuco-nojirimycin, a nanomolar alpha-L-fucosidase inhibitor.
Dubernet M; Defoin A; Tarnus C
Bioorg Med Chem Lett; 2006 Mar; 16(5):1172-4. PubMed ID: 16376079
[TBL] [Abstract][Full Text] [Related]
7. Difluoromethylenated polyhydroxylated pyrrolidines: facile synthesis, crystal structure and biological evaluation.
Wang RW; Xu J; Lopez O; Bols M; Qing FL
Future Med Chem; 2009 Aug; 1(5):991-7. PubMed ID: 21426093
[TBL] [Abstract][Full Text] [Related]
8. The 'mirror-image' postulate as a guide to the selection and evaluation of pyrrolidines as α-l-fucosidase inhibitors.
Stocker BL; Jongkees SA; Win-Mason AL; Dangerfield EM; Withers SG; Timmer MS
Carbohydr Res; 2013 Feb; 367():29-32. PubMed ID: 23295913
[TBL] [Abstract][Full Text] [Related]
9. Glycosidase-substrate interactions analysis by STD-NMR spectroscopy: study of alpha-L-fucosidase.
Berteau O; Sandström C; Bielicki J; Anson DS; Kenne L
J Am Chem Soc; 2003 Dec; 125(50):15296-7. PubMed ID: 14664566
[TBL] [Abstract][Full Text] [Related]
10. Expeditious synthesis of tri- and tetrahydroxyazepanes from D-(-)-quinic acid as potent glycosidase inhibitors.
Shih TL; Yang RY; Li ST; Chiang CF; Lin CH
J Org Chem; 2007 May; 72(11):4258-61. PubMed ID: 17480095
[TBL] [Abstract][Full Text] [Related]
11. Skeletal rearrangement of seven-membered iminosugars: synthesis of (-)-adenophorine, (-)-1-epi-adenophorine and derivatives and evaluation as glycosidase inhibitors.
Mondon M; Lecornué F; Guillard J; Nakagawa S; Kato A; Blériot Y
Bioorg Med Chem; 2013 Aug; 21(16):4803-12. PubMed ID: 23611766
[TBL] [Abstract][Full Text] [Related]
12. Spirocyclopropyl pyrrolidines as a new series of alpha-L-fucosidase inhibitors.
Laroche C; Behr JB; Szymoniak J; Bertus P; Schütz C; Vogel P; Plantier-Royon R
Bioorg Med Chem; 2006 Jun; 14(12):4047-54. PubMed ID: 16488612
[TBL] [Abstract][Full Text] [Related]
13. Discovery of different types of inhibition between the human and thermotoga maritima alpha-fucosidases by fuconojirimycin-based derivatives.
Ho CW; Lin YN; Chang CF; Li ST; Wu YT; Wu CY; Chang CF; Liu SW; Li YK; Lin CH
Biochemistry; 2006 May; 45(18):5695-702. PubMed ID: 16669613
[TBL] [Abstract][Full Text] [Related]
14. Synthesis and evaluation of N-alkylated analogues of aza-galacto-fagomine - potential pharmacological chaperones for Krabbe disease.
Viuff AH; Jensen HH
Org Biomol Chem; 2016 Sep; 14(36):8545-56. PubMed ID: 27545315
[TBL] [Abstract][Full Text] [Related]
15. The spirocyclopropyl moiety as a methyl surrogate in the structure of l-fucosidase and l-rhamnosidase inhibitors.
Pearson MS; Floquet N; Bello C; Vogel P; Plantier-Royon R; Szymoniak J; Bertus P; Behr JB
Bioorg Med Chem; 2009 Dec; 17(23):8020-6. PubMed ID: 19875298
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and evaluation of the glycosidase inhibitory activity of 5-hydroxy substituted isofagomine analogues.
Matin MM; Sharma T; Sabharwal SG; Dhavale DD
Org Biomol Chem; 2005 May; 3(9):1702-7. PubMed ID: 15858653
[TBL] [Abstract][Full Text] [Related]
17. Synthesis of branched seven-membered 1-N-iminosugars and their evaluation as glycosidase inhibitors.
Li H; Zhang Y; Favre S; Vogel P; Sollogoub M; Blériot Y
Carbohydr Res; 2012 Jul; 356():110-4. PubMed ID: 22129839
[TBL] [Abstract][Full Text] [Related]
18. Synthesis of polyhydroxylated piperidines and evaluation as glycosidase inhibitors.
Tite T; Lallemand MC; Poupon E; Kunesch N; Tillequin F; Gravier-Pelletier C; Le Merrer Y; Husson HP
Bioorg Med Chem; 2004 Oct; 12(19):5091-7. PubMed ID: 15351392
[TBL] [Abstract][Full Text] [Related]
19. Rapid diversity-oriented synthesis in microtiter plates for in situ screening: discovery of potent and selective alpha-fucosidase inhibitors.
Wu CY; Chang CF; Chen JS; Wong CH; Lin CH
Angew Chem Int Ed Engl; 2003 Oct; 42(38):4661-4. PubMed ID: 14533157
[No Abstract] [Full Text] [Related]
20. Stereoselective total synthesis of aminoiminohexitols via carbamate annulation.
Win-Mason AL; Jongkees SA; Withers SG; Tyler PC; Timmer MS; Stocker BL
J Org Chem; 2011 Dec; 76(23):9611-21. PubMed ID: 22022891
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]