BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

212 related articles for article (PubMed ID: 20655754)

  • 1. Improved inhibition of the histone acetyltransferase PCAF by an anacardic acid derivative.
    Ghizzoni M; Boltjes A; Graaf Cd; Haisma HJ; Dekker FJ
    Bioorg Med Chem; 2010 Aug; 18(16):5826-34. PubMed ID: 20655754
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis of benzamides related to anacardic acid and their histone acetyltransferase (HAT) inhibitory activities.
    Souto JA; Conte M; Alvarez R; Nebbioso A; Carafa V; Altucci L; de Lera AR
    ChemMedChem; 2008 Sep; 3(9):1435-42. PubMed ID: 18537201
    [TBL] [Abstract][Full Text] [Related]  

  • 3. New anacardic acid-inspired benzamides: histone lysine acetyltransferase activators.
    Souto JA; Benedetti R; Otto K; Miceli M; Alvarez R; Altucci L; de Lera AR
    ChemMedChem; 2010 Sep; 5(9):1530-40. PubMed ID: 20683922
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Characterization of novel inhibitors of histone acetyltransferases.
    Eliseeva ED; Valkov V; Jung M; Jung MO
    Mol Cancer Ther; 2007 Sep; 6(9):2391-8. PubMed ID: 17876038
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Inhibition of PCAF by anacardic acid derivative leads to apoptosis and breaks resistance to DNA damage in BCR-ABL-expressing cells.
    Kusio-Kobialka M; Dudka-Ruszkowska W; Ghizzoni M; Dekker FJ; Piwocka K
    Anticancer Agents Med Chem; 2013 Jun; 13(5):762-7. PubMed ID: 23157591
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Inhibition of PCAF histone acetyltransferase and cytotoxic effect of N-acylanthranilic acids.
    Park WJ; Ma E
    Arch Pharm Res; 2012 Aug; 35(8):1379-86. PubMed ID: 22941480
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Enzyme kinetics and inhibition of histone acetyltransferase KAT8.
    Wapenaar H; van der Wouden PE; Groves MR; Rotili D; Mai A; Dekker FJ
    Eur J Med Chem; 2015 Nov; 105():289-96. PubMed ID: 26505788
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and biological testing of novel pyridoisothiazolones as histone acetyltransferase inhibitors.
    Furdas SD; Shekfeh S; Bissinger EM; Wagner JM; Schlimme S; Valkov V; Hendzel M; Jung M; Sippl W
    Bioorg Med Chem; 2011 Jun; 19(12):3678-89. PubMed ID: 21353783
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Histone acetyl transferases as emerging drug targets.
    Dekker FJ; Haisma HJ
    Drug Discov Today; 2009 Oct; 14(19-20):942-8. PubMed ID: 19577000
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Reactivity of isothiazolones and isothiazolone-1-oxides in the inhibition of the PCAF histone acetyltransferase.
    Ghizzoni M; Haisma HJ; Dekker FJ
    Eur J Med Chem; 2009 Dec; 44(12):4855-61. PubMed ID: 19683843
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Activation of p300 histone acetyltransferase by small molecules altering enzyme structure: probed by surface-enhanced Raman spectroscopy.
    Mantelingu K; Kishore AH; Balasubramanyam K; Kumar GV; Altaf M; Swamy SN; Selvi R; Das C; Narayana C; Rangappa KS; Kundu TK
    J Phys Chem B; 2007 May; 111(17):4527-34. PubMed ID: 17417897
    [TBL] [Abstract][Full Text] [Related]  

  • 12. 6-alkylsalicylates are selective Tip60 inhibitors and target the acetyl-CoA binding site.
    Ghizzoni M; Wu J; Gao T; Haisma HJ; Dekker FJ; George Zheng Y
    Eur J Med Chem; 2012 Jan; 47(1):337-44. PubMed ID: 22100137
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis of isothiazol-3-one derivatives as inhibitors of histone acetyltransferases (HATs).
    Gorsuch S; Bavetsias V; Rowlands MG; Aherne GW; Workman P; Jarman M; McDonald E
    Bioorg Med Chem; 2009 Jan; 17(2):467-74. PubMed ID: 19101154
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Identification of long chain alkylidenemalonates as novel small molecule modulators of histone acetyltransferases.
    Sbardella G; Castellano S; Vicidomini C; Rotili D; Nebbioso A; Miceli M; Altucci L; Mai A
    Bioorg Med Chem Lett; 2008 May; 18(9):2788-92. PubMed ID: 18434144
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Azide-alkyne cycloaddition affording enzymatically tunable bisubstrate based inhibitors of histone acetyltransferase PCAF.
    van Ameijde J; Zwiebel AP; Ruijtenbeek R; Liskamp RM
    Bioorg Med Chem Lett; 2014 Jan; 24(1):113-6. PubMed ID: 24345448
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Bisubstrate analogue structure-activity relationships for p300 histone acetyltransferase inhibitors.
    Sagar V; Zheng W; Thompson PR; Cole PA
    Bioorg Med Chem; 2004 Jun; 12(12):3383-90. PubMed ID: 15158807
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Inhibition of histone acetyltransferase activity by anacardic acid sensitizes tumor cells to ionizing radiation.
    Sun Y; Jiang X; Chen S; Price BD
    FEBS Lett; 2006 Aug; 580(18):4353-6. PubMed ID: 16844118
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Phenylephrine-induced cardiac hypertrophy is attenuated by a histone acetylase inhibitor anacardic acid in mice.
    Peng C; Luo X; Li S; Sun H
    Mol Biosyst; 2017 Mar; 13(4):714-724. PubMed ID: 28194469
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Histone Acetyltransferase (HAT) P300/CBP Inhibitors Induce Synthetic Lethality in PTEN-Deficient Colorectal Cancer Cells through Destabilizing AKT.
    Liu Y; Yang EJ; Shi C; Mou PK; Zhang B; Wu C; Lyu J; Shim JS
    Int J Biol Sci; 2020; 16(11):1774-1784. PubMed ID: 32398948
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Modulation of the activity of histone acetyltransferases by long chain alkylidenemalonates (LoCAMs).
    Milite C; Castellano S; Benedetti R; Tosco A; Ciliberti C; Vicidomini C; Boully L; Franci G; Altucci L; Mai A; Sbardella G
    Bioorg Med Chem; 2011 Jun; 19(12):3690-701. PubMed ID: 21292492
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 11.