BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

125 related articles for article (PubMed ID: 20667744)

  • 1. Synthesis and biological evaluation of tetracyclic fluoroquinolones as antibacterial and anticancer agents.
    Al-Trawneh SA; Zahra JA; Kamal MR; El-Abadelah MM; Zani F; Incerti M; Cavazzoni A; Alfieri RR; Petronini PG; Vicini P
    Bioorg Med Chem; 2010 Aug; 18(16):5873-84. PubMed ID: 20667744
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and biological evaluation of tetracyclic thienopyridones as antibacterial and antitumor agents.
    Al-Trawneh SA; El-Abadelah MM; Zahra JA; Al-Taweel SA; Zani F; Incerti M; Cavazzoni A; Vicini P
    Bioorg Med Chem; 2011 Apr; 19(8):2541-8. PubMed ID: 21458275
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Hydrazones of 2-aryl-quinoline-4-carboxylic acid hydrazides: synthesis and preliminary evaluation as antimicrobial agents.
    Metwally KA; Abdel-Aziz LM; Lashine el-SM; Husseiny MI; Badawy RH
    Bioorg Med Chem; 2006 Dec; 14(24):8675-82. PubMed ID: 16949294
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Dual-targeting properties of the 3-aminopyrrolidyl quinolones, DC-159a and sitafloxacin, against DNA gyrase and topoisomerase IV: contribution to reducing in vitro emergence of quinolone-resistant Streptococcus pneumoniae.
    Okumura R; Hirata T; Onodera Y; Hoshino K; Otani T; Yamamoto T
    J Antimicrob Chemother; 2008 Jul; 62(1):98-104. PubMed ID: 18390884
    [TBL] [Abstract][Full Text] [Related]  

  • 5. New hydroxamic acid derivatives of fluoroquinolones: synthesis and evaluation of antibacterial and anticancer properties.
    Rajulu GG; Bhojya Naik HS; Viswanadhan A; Thiruvengadam J; Rajesh K; Ganesh S; Jagadheshan H; Kesavan PK
    Chem Pharm Bull (Tokyo); 2014; 62(2):168-75. PubMed ID: 24270473
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and biological evaluation of some 2,4,5-trisubstituted thiazole derivatives as potential antimicrobial and anticancer agents.
    Al-Saadi MS; Faidallah HM; Rostom SA
    Arch Pharm (Weinheim); 2008 Jul; 341(7):424-34. PubMed ID: 18574850
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis of lipophilic dimeric C-7/C-7-linked ciprofloxacin and C-6/C-6-linked levofloxacin derivatives. Versatile in vitro biological evaluations of monomeric and dimeric fluoroquinolone derivatives as potential antitumor, antibacterial or antimycobacterial agents.
    Azéma J; Guidetti B; Korolyov A; Kiss R; Roques C; Constant P; Daffé M; Malet-Martino M
    Eur J Med Chem; 2011 Dec; 46(12):6025-38. PubMed ID: 22036229
    [TBL] [Abstract][Full Text] [Related]  

  • 8. 3-aminoquinazolinediones as a new class of antibacterial agents demonstrating excellent antibacterial activity against wild-type and multidrug resistant organisms.
    Ellsworth EL; Tran TP; Showalter HD; Sanchez JP; Watson BM; Stier MA; Domagala JM; Gracheck SJ; Joannides ET; Shapiro MA; Dunham SA; Hanna DL; Huband MD; Gage JW; Bronstein JC; Liu JY; Nguyen DQ; Singh R
    J Med Chem; 2006 Nov; 49(22):6435-8. PubMed ID: 17064062
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and biological evaluation of some novel fused pyrazolopyrimidines as potential anticancer and antimicrobial agents.
    Abd El Razik HA; Wahab AE
    Arch Pharm (Weinheim); 2011 Mar; 344(3):184-96. PubMed ID: 21384418
    [TBL] [Abstract][Full Text] [Related]  

  • 10. The synthesis and biological evaluation of a novel series of C7 non-basic substituted fluoroquinolones as antibacterial agents.
    Huang X; Chen D; Wu N; Zhang A; Jia Z; Li X
    Bioorg Med Chem Lett; 2009 Aug; 19(15):4130-3. PubMed ID: 19539467
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and in vitro antibacterial activity of novel fluoroquinolone derivatives containing substituted piperidines.
    Chai Y; Liu M; Wang B; You X; Feng L; Zhang Y; Cao J; Guo H
    Bioorg Med Chem Lett; 2010 Sep; 20(17):5195-8. PubMed ID: 20667731
    [TBL] [Abstract][Full Text] [Related]  

  • 12. 4-Substituted 4-(1H-1,2,3-triazol-1-yl)piperidine: novel C7 moieties of fluoroquinolones as antibacterial agents.
    Huang X; Zhang A; Chen D; Jia Z; Li X
    Bioorg Med Chem Lett; 2010 May; 20(9):2859-63. PubMed ID: 20347299
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis and biological evaluation of some novel polysubstituted pyrimidine derivatives as potential antimicrobial and anticancer agents.
    Rostom SA; Ashour HM; Abd El Razik HA
    Arch Pharm (Weinheim); 2009 May; 342(5):299-310. PubMed ID: 19415663
    [TBL] [Abstract][Full Text] [Related]  

  • 14. [Synthesis and antibacterial activities of 7-{4-[2-[2-substituted-4-((5S)-5-acetylaminomethyl-2-oxo-oxazolidin-3-yl)}-phenyl] -ethyl]-piperazin-1-yl}-fluoroquinolones].
    Yu HJ; Zhou WC
    Yao Xue Xue Bao; 2006 Oct; 41(10):990-9. PubMed ID: 17184119
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Discovery of a novel azaindole class of antibacterial agents targeting the ATPase domains of DNA gyrase and Topoisomerase IV.
    Manchester JI; Dussault DD; Rose JA; Boriack-Sjodin PA; Uria-Nickelsen M; Ioannidis G; Bist S; Fleming P; Hull KG
    Bioorg Med Chem Lett; 2012 Aug; 22(15):5150-6. PubMed ID: 22814212
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Antimycobacterial activities of novel fluoroquinolones.
    Senthilkumar P; Dinakaran M; Yogeeswari P; China A; Nagaraja V; Sriram D
    Biomed Pharmacother; 2009 Jan; 63(1):27-35. PubMed ID: 18031974
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and in vitro antibacterial activity of 7-(4-alkoxyimino-3-amino-3-methylpiperidin-1-yl)fluoroquinolone derivatives.
    Chai Y; Wan ZL; Wang B; Guo HY; Liu ML
    Eur J Med Chem; 2009 Oct; 44(10):4063-9. PubMed ID: 19481308
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis, antimicrobial activity and molecular modeling study of substituted 5-aryl-pyrimido[5,4-c]quinoline-2,4-diones.
    Ismail MA; Al-Shihry S; Arafa RK; El-Ayaan U
    J Enzyme Inhib Med Chem; 2013 Jun; 28(3):530-8. PubMed ID: 22397395
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and antibacterial activity of novel and potent DNA gyrase inhibitors with azole ring.
    Tanitame A; Oyamada Y; Ofuji K; Fujimoto M; Suzuki K; Ueda T; Terauchi H; Kawasaki M; Nagai K; Wachi M; Yamagishi J
    Bioorg Med Chem; 2004 Nov; 12(21):5515-24. PubMed ID: 15465328
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis and antimycobacterial evaluation of newer 1-cyclopropyl-1,4-dihydro-6-fluoro-7-(substituted secondary amino)-8-methoxy-5-(sub)-4-oxoquinoline-3-carboxylic acids.
    Senthilkumar P; Dinakaran M; Banerjee D; Devakaram RV; Yogeeswari P; China A; Nagaraja V; Sriram D
    Bioorg Med Chem; 2008 Mar; 16(5):2558-69. PubMed ID: 18078756
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.