BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

96 related articles for article (PubMed ID: 20694697)

  • 1. A scintillation proximity assay for fatty acid amide hydrolase compatible with inhibitor screening.
    Wang Y; Jones P
    Methods Mol Biol; 2009; 572():247-59. PubMed ID: 20694697
    [TBL] [Abstract][Full Text] [Related]  

  • 2. A novel scintillation proximity assay for fatty acid amide hydrolase compatible with inhibitor screening.
    Wang Y; Xu J; Uveges A; Ramarao MK; Rogers KE; Jones PG
    Anal Biochem; 2006 Jul; 354(1):35-42. PubMed ID: 16707086
    [TBL] [Abstract][Full Text] [Related]  

  • 3. A fluorescence-based assay for fatty acid amide hydrolase compatible with high-throughput screening.
    Ramarao MK; Murphy EA; Shen MW; Wang Y; Bushell KN; Huang N; Pan N; Williams C; Clark JD
    Anal Biochem; 2005 Aug; 343(1):143-51. PubMed ID: 16018870
    [TBL] [Abstract][Full Text] [Related]  

  • 4. High-throughput screening for the discovery of inhibitors of fatty acid amide hydrolase using a microsome-based fluorescent assay.
    Wang Y; Ramirez F; Krishnamurthy G; Gilbert A; Kadakia N; Xu J; Kalgaonkar G; Ramarao MK; Edris W; Rogers KE; Jones PG
    J Biomol Screen; 2006 Aug; 11(5):519-27. PubMed ID: 16760367
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Use of scintillation proximity assay to measure radioligand binding to immobilized receptors without separation of bound from free ligand.
    Berry J; Price-Jones M; Killian B
    Methods Mol Biol; 2012; 897():79-94. PubMed ID: 22674161
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Biochemical characterization and in vitro activity of AZ513, a noncovalent, reversible, and noncompetitive inhibitor of fatty acid amide hydrolase.
    Scott CW; Tian G; Yu XH; Paschetto KA; Wilkins DE; Meury L; Cao CQ; Varnes J; Edwards PD
    Eur J Pharmacol; 2011 Sep; 667(1-3):74-9. PubMed ID: 21645511
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Mechanism of inhibition of fatty acid amide hydrolase by sulfonamide-containing benzothiazoles: long residence time derived from increased kinetic barrier and not exclusively from thermodynamic potency.
    Tian G; Paschetto KA; Gharahdaghi F; Gordon E; Wilkins DE; Luo X; Scott CW
    Biochemistry; 2011 Aug; 50(32):6867-78. PubMed ID: 21728345
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Identification of non-peptidic neuromedin U receptor modulators by a robust homogeneous screening assay.
    Meng T; Su HR; Binkert C; Fischli W; Zhou L; Shen JK; Wang MW
    Acta Pharmacol Sin; 2008 Apr; 29(4):517-27. PubMed ID: 18358099
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Discovery of novel spirocyclic inhibitors of fatty acid amide hydrolase (FAAH). Part 2. Discovery of 7-azaspiro[3.5]nonane urea PF-04862853, an orally efficacious inhibitor of fatty acid amide hydrolase (FAAH) for pain.
    Meyers MJ; Long SA; Pelc MJ; Wang JL; Bowen SJ; Schweitzer BA; Wilcox MV; McDonald J; Smith SE; Foltin S; Rumsey J; Yang YS; Walker MC; Kamtekar S; Beidler D; Thorarensen A
    Bioorg Med Chem Lett; 2011 Nov; 21(21):6545-53. PubMed ID: 21924613
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Development of a scintillation proximity assay for human insulin-like growth factor-binding protein 4 compatible with inhibitor high-throughput screening.
    Khawaja XZ
    Anal Biochem; 2007 Jul; 366(1):80-6. PubMed ID: 17482135
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Development of a scintillation proximity assay binding method for the human 5-hydroxytryptamine 6 receptor using intact cells.
    Carrick T; Kowal D; Nawoschik S; Zhang G; Chan K; Dunlop J
    Anal Biochem; 2008 Oct; 381(1):27-32. PubMed ID: 18601889
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Mining biologically-active molecules for inhibitors of fatty acid amide hydrolase (FAAH): identification of phenmedipham and amperozide as FAAH inhibitors.
    Vincent F; Nguyen MT; Emerling DE; Kelly MG; Duncton MA
    Bioorg Med Chem Lett; 2009 Dec; 19(23):6793-6. PubMed ID: 19850474
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Development of fragment-based n-FABS NMR screening applied to the membrane enzyme FAAH.
    Lambruschini C; Veronesi M; Romeo E; Garau G; Bandiera T; Piomelli D; Scarpelli R; Dalvit C
    Chembiochem; 2013 Sep; 14(13):1611-9. PubMed ID: 23918626
    [TBL] [Abstract][Full Text] [Related]  

  • 14. A scintillation proximity assay amenable for screening and characterization of DNA gyrase B subunit inhibitors.
    Gevi M; Domenici E
    Anal Biochem; 2002 Jan; 300(1):34-9. PubMed ID: 11743689
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Fatty acid amide hydrolase inhibitors display broad selectivity and inhibit multiple carboxylesterases as off-targets.
    Zhang D; Saraf A; Kolasa T; Bhatia P; Zheng GZ; Patel M; Lannoye GS; Richardson P; Stewart A; Rogers JC; Brioni JD; Surowy CS
    Neuropharmacology; 2007 Mar; 52(4):1095-105. PubMed ID: 17217969
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Discovery of novel spirocyclic inhibitors of fatty acid amide hydrolase (FAAH). Part 1: identification of 7-azaspiro[3.5]nonane and 1-oxa-8-azaspiro[4.5]decane as lead scaffolds.
    Meyers MJ; Long SA; Pelc MJ; Wang JL; Bowen SJ; Walker MC; Schweitzer BA; Madsen HM; Tenbrink RE; McDonald J; Smith SE; Foltin S; Beidler D; Thorarensen A
    Bioorg Med Chem Lett; 2011 Nov; 21(21):6538-44. PubMed ID: 21924614
    [TBL] [Abstract][Full Text] [Related]  

  • 17. A MBP-FAAH fusion protein as a tool to produce human and rat fatty acid amide hydrolase: expression and pharmacological comparison.
    Labar G; Vliet FV; Wouters J; Lambert DM
    Amino Acids; 2008 Jan; 34(1):127-33. PubMed ID: 17476568
    [TBL] [Abstract][Full Text] [Related]  

  • 18. A high throughput fluorescent assay for measuring the activity of fatty acid amide hydrolase.
    Kage KL; Richardson PL; Traphagen L; Severin J; Pereda-Lopez A; Lubben T; Davis-Taber R; Vos MH; Bartley D; Walter K; Harlan J; Solomon L; Warrior U; Holzman TF; Faltynek C; Surowy CS; Scott VE
    J Neurosci Methods; 2007 Mar; 161(1):47-54. PubMed ID: 17083980
    [TBL] [Abstract][Full Text] [Related]  

  • 19. A high-throughput, nonisotopic, competitive binding assay for kinases using nonselective inhibitor probes (ED-NSIP).
    Vainshtein I; Silveria S; Kaul P; Rouhani R; Eglen RM; Wang J
    J Biomol Screen; 2002 Dec; 7(6):507-14. PubMed ID: 14599348
    [TBL] [Abstract][Full Text] [Related]  

  • 20. High-throughput scintillation proximity assay for stearoyl-CoA desaturase-1.
    Tawa P; Falgueyret JP; Guiral S; Isabel E; Powell DA; Zuck P; Skorey K
    J Biomol Screen; 2011 Jun; 16(5):506-17. PubMed ID: 21406617
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 5.