These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

186 related articles for article (PubMed ID: 20804196)

  • 1. Discovery of novel 5-benzylidenerhodanine and 5-benzylidenethiazolidine-2,4-dione inhibitors of MurD ligase.
    Zidar N; Tomasić T; Sink R; Rupnik V; Kovac A; Turk S; Patin D; Blanot D; Contreras Martel C; Dessen A; Müller Premru M; Zega A; Gobec S; Peterlin Masic L; Kikelj D
    J Med Chem; 2010 Sep; 53(18):6584-94. PubMed ID: 20804196
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Structure-based design of a new series of D-glutamic acid based inhibitors of bacterial UDP-N-acetylmuramoyl-L-alanine:D-glutamate ligase (MurD).
    Tomasić T; Zidar N; Sink R; Kovac A; Blanot D; Contreras-Martel C; Dessen A; Müller-Premru M; Zega A; Gobec S; Kikelj D; Masic LP
    J Med Chem; 2011 Jul; 54(13):4600-10. PubMed ID: 21591605
    [TBL] [Abstract][Full Text] [Related]  

  • 3. New 5-benzylidenethiazolidin-4-one inhibitors of bacterial MurD ligase: design, synthesis, crystal structures, and biological evaluation.
    Zidar N; Tomašić T; Šink R; Kovač A; Patin D; Blanot D; Contreras-Martel C; Dessen A; Premru MM; Zega A; Gobec S; Mašič LP; Kikelj D
    Eur J Med Chem; 2011 Nov; 46(11):5512-23. PubMed ID: 21963114
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Novel naphthalene-N-sulfonyl-D-glutamic acid derivatives as inhibitors of MurD, a key peptidoglycan biosynthesis enzyme.
    Humljan J; Kotnik M; Contreras-Martel C; Blanot D; Urleb U; Dessen A; Solmajer T; Gobec S
    J Med Chem; 2008 Dec; 51(23):7486-94. PubMed ID: 19007109
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Novel 2-thioxothiazolidin-4-one inhibitors of bacterial MurD ligase targeting D-Glu- and diphosphate-binding sites.
    Tomašić T; Kovač A; Simčič M; Blanot D; Grdadolnik SG; Gobec S; Kikelj D; Peterlin Mašič L
    Eur J Med Chem; 2011 Sep; 46(9):3964-75. PubMed ID: 21703731
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and biological evaluation of new glutamic acid-based inhibitors of MurD ligase.
    Tomasić T; Zidar N; Rupnik V; Kovac A; Blanot D; Gobec S; Kikelj D; Masic LP
    Bioorg Med Chem Lett; 2009 Jan; 19(1):153-7. PubMed ID: 19014883
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Discovery of novel benzene 1,3-dicarboxylic acid inhibitors of bacterial MurD and MurE ligases by structure-based virtual screening approach.
    Perdih A; Kovac A; Wolber G; Blanot D; Gobec S; Solmajer T
    Bioorg Med Chem Lett; 2009 May; 19(10):2668-73. PubMed ID: 19369074
    [TBL] [Abstract][Full Text] [Related]  

  • 8. 5-Benzylidenethiazolidin-4-ones as multitarget inhibitors of bacterial Mur ligases.
    Tomasić T; Zidar N; Kovac A; Turk S; Simcic M; Blanot D; Müller-Premru M; Filipic M; Grdadolnik SG; Zega A; Anderluh M; Gobec S; Kikelj D; Peterlin Masic L
    ChemMedChem; 2010 Feb; 5(2):286-95. PubMed ID: 20024979
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Green Synthesis, Biological Activity Evaluation, and Molecular Docking Studies of Aryl Alkylidene 2, 4-thiazolidinedione and Rhodanine Derivatives as Antimicrobial Agents.
    Akhavan M; Foroughifar N; Pasdar H; Bekhradnia A
    Comb Chem High Throughput Screen; 2019; 22(10):716-727. PubMed ID: 31775594
    [TBL] [Abstract][Full Text] [Related]  

  • 10. 5-benzylidenerhodanine and 5-benzylidene-2-4-thiazolidinedione based antibacterials.
    Zvarec O; Polyak SW; Tieu W; Kuan K; Dai H; Pedersen DS; Morona R; Zhang L; Booker GW; Abell AD
    Bioorg Med Chem Lett; 2012 Apr; 22(8):2720-2. PubMed ID: 22444680
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Design, synthesis and structure-activity relationships of new phosphinate inhibitors of MurD.
    Strancar K; Blanot D; Gobec S
    Bioorg Med Chem Lett; 2006 Jan; 16(2):343-8. PubMed ID: 16271472
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis of new chalcone derivatives containing a rhodanine-3-acetic acid moiety with potential anti-bacterial activity.
    Chen ZH; Zheng CJ; Sun LP; Piao HR
    Eur J Med Chem; 2010 Dec; 45(12):5739-43. PubMed ID: 20889240
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Second-generation sulfonamide inhibitors of D-glutamic acid-adding enzyme: activity optimisation with conformationally rigid analogues of D-glutamic acid.
    Sosič I; Barreteau H; Simčič M; Sink R; Cesar J; Zega A; Grdadolnik SG; Contreras-Martel C; Dessen A; Amoroso A; Joris B; Blanot D; Gobec S
    Eur J Med Chem; 2011 Jul; 46(7):2880-94. PubMed ID: 21524830
    [TBL] [Abstract][Full Text] [Related]  

  • 14. NMR and molecular dynamics study of the binding mode of naphthalene-N-sulfonyl-D-glutamic acid derivatives: novel MurD ligase inhibitors.
    Simcic M; Hodoscek M; Humljan J; Kristan K; Urleb U; Kocjan D; Grdadolnik SG
    J Med Chem; 2009 May; 52(9):2899-908. PubMed ID: 19358612
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Structural and functional characterization of enantiomeric glutamic acid derivatives as potential transition state analogue inhibitors of MurD ligase.
    Kotnik M; Humljan J; Contreras-Martel C; Oblak M; Kristan K; Hervé M; Blanot D; Urleb U; Gobec S; Dessen A; Solmajer T
    J Mol Biol; 2007 Jun; 370(1):107-15. PubMed ID: 17507028
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis, structure and structure-activity relationship analysis of 3-tert-butoxycarbonyl-2-arylthiazolidine-4-carboxylic acid derivatives as potential antibacterial agents.
    Song ZC; Ma GY; Lv PC; Li HQ; Xiao ZP; Zhu HL
    Eur J Med Chem; 2009 Oct; 44(10):3903-8. PubMed ID: 19423200
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Benzylidene rhodanines as novel inhibitors of UDP-N-acetylmuramate/L-alanine ligase.
    Sim MM; Ng SB; Buss AD; Crasta SC; Goh KL; Lee SK
    Bioorg Med Chem Lett; 2002 Feb; 12(4):697-9. PubMed ID: 11844704
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis and biological evaluation of N-acylhydrazones as inhibitors of MurC and MurD ligases.
    Sink R; Kovac A; Tomasić T; Rupnik V; Boniface A; Bostock J; Chopra I; Blanot D; Masic LP; Gobec S; Zega A
    ChemMedChem; 2008 Sep; 3(9):1362-70. PubMed ID: 18651694
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and biological evaluation of new epalrestat analogues as aldose reductase inhibitors (ARIs).
    Reddy TN; Ravinder M; Bagul P; Ravikanti K; Bagul C; Nanubolu JB; Srinivas K; Banerjee SK; Rao VJ
    Eur J Med Chem; 2014 Jan; 71():53-66. PubMed ID: 24275248
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Discovery of new inhibitors of D-alanine:D-alanine ligase by structure-based virtual screening.
    Kovac A; Konc J; Vehar B; Bostock JM; Chopra I; Janezic D; Gobec S
    J Med Chem; 2008 Dec; 51(23):7442-8. PubMed ID: 19053785
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.