These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
3. Participation of transmembrane proline 82 in angiotensin II AT1 receptor signal transduction. Reis RI; Santos EL; Pesquero JB; Oliveira L; Schanstra JP; Bascands JL; Pecher C; Paiva AC; Costa-Neto CM Regul Pept; 2007 Apr; 140(1-2):32-6. PubMed ID: 17239455 [TBL] [Abstract][Full Text] [Related]
4. Ghrelin receptor inverse agonists: identification of an active peptide core and its interaction epitopes on the receptor. Holst B; Lang M; Brandt E; Bach A; Howard A; Frimurer TM; Beck-Sickinger A; Schwartz TW Mol Pharmacol; 2006 Sep; 70(3):936-46. PubMed ID: 16798937 [TBL] [Abstract][Full Text] [Related]
5. Molecular basis for agonism in the BB3 receptor: an epitope located on the interface of transmembrane-III, -VI, and -VII. Gbahou F; Holst B; Schwartz TW J Pharmacol Exp Ther; 2010 Apr; 333(1):51-9. PubMed ID: 20065020 [TBL] [Abstract][Full Text] [Related]
6. Agonist-induced conformational changes in bovine rhodopsin: insight into activation of G-protein-coupled receptors. Bhattacharya S; Hall SE; Vaidehi N J Mol Biol; 2008 Oct; 382(2):539-55. PubMed ID: 18638482 [TBL] [Abstract][Full Text] [Related]
7. Recognition of privileged structures by G-protein coupled receptors. Bondensgaard K; Ankersen M; Thøgersen H; Hansen BS; Wulff BS; Bywater RP J Med Chem; 2004 Feb; 47(4):888-99. PubMed ID: 14761190 [TBL] [Abstract][Full Text] [Related]
8. The third extracellular loop of G-protein-coupled receptors: more than just a linker between two important transmembrane helices. Lawson Z; Wheatley M Biochem Soc Trans; 2004 Dec; 32(Pt 6):1048-50. PubMed ID: 15506960 [TBL] [Abstract][Full Text] [Related]
9. Structure-function relationships of the human bitter taste receptor hTAS2R1: insights from molecular modeling studies. Dai W; You Z; Zhou H; Zhang J; Hu Y J Recept Signal Transduct Res; 2011 Jun; 31(3):229-40. PubMed ID: 21619450 [TBL] [Abstract][Full Text] [Related]
10. A second disulfide bridge from the N-terminal domain to extracellular loop 2 dampens receptor activity in GPR39. Storjohann L; Holst B; Schwartz TW Biochemistry; 2008 Sep; 47(35):9198-207. PubMed ID: 18693759 [TBL] [Abstract][Full Text] [Related]
11. Photolabelling the urotensin II receptor reveals distinct agonist- and partial-agonist-binding sites. Holleran BJ; Beaulieu ME; Proulx CD; Lavigne P; Escher E; Leduc R Biochem J; 2007 Feb; 402(1):51-61. PubMed ID: 17064254 [TBL] [Abstract][Full Text] [Related]
12. Conserved water-mediated hydrogen bond network between TM-I, -II, -VI, and -VII in 7TM receptor activation. Nygaard R; Valentin-Hansen L; Mokrosinski J; Frimurer TM; Schwartz TW J Biol Chem; 2010 Jun; 285(25):19625-36. PubMed ID: 20395291 [TBL] [Abstract][Full Text] [Related]
13. Molecular mechanism of 7TM receptor activation--a global toggle switch model. Schwartz TW; Frimurer TM; Holst B; Rosenkilde MM; Elling CE Annu Rev Pharmacol Toxicol; 2006; 46():481-519. PubMed ID: 16402913 [TBL] [Abstract][Full Text] [Related]
14. Activation of the CXCR3 chemokine receptor through anchoring of a small molecule chelator ligand between TM-III, -IV, and -VI. Rosenkilde MM; Andersen MB; Nygaard R; Frimurer TM; Schwartz TW Mol Pharmacol; 2007 Mar; 71(3):930-41. PubMed ID: 17170198 [TBL] [Abstract][Full Text] [Related]
15. Extracellular loops and ligand binding to a subfamily of Family A G-protein-coupled receptors. Wheatley M; Simms J; Hawtin SR; Wesley VJ; Wootten D; Conner M; Lawson Z; Conner AC; Baker A; Cashmore Y; Kendrick R; Parslow RA Biochem Soc Trans; 2007 Aug; 35(Pt 4):717-20. PubMed ID: 17635132 [TBL] [Abstract][Full Text] [Related]
16. Allosteric agonists of 7TM receptors: expanding the pharmacological toolbox. Langmead CJ; Christopoulos A Trends Pharmacol Sci; 2006 Sep; 27(9):475-81. PubMed ID: 16889837 [TBL] [Abstract][Full Text] [Related]
17. An automated system for the analysis of G protein-coupled receptor transmembrane binding pockets: alignment, receptor-based pharmacophores, and their application. Kratochwil NA; Malherbe P; Lindemann L; Ebeling M; Hoener MC; Mühlemann A; Porter RH; Stahl M; Gerber PR J Chem Inf Model; 2005; 45(5):1324-36. PubMed ID: 16180909 [TBL] [Abstract][Full Text] [Related]
18. G protein coupled receptors as allosteric proteins and the role of allosteric modulators. Kenakin T J Recept Signal Transduct Res; 2010 Oct; 30(5):313-21. PubMed ID: 20858023 [TBL] [Abstract][Full Text] [Related]
19. The role of transmembrane segment II in 7TM receptor activation. Benned-Jensen T; Rosenkilde MM Curr Mol Pharmacol; 2009 Jun; 2(2):140-8. PubMed ID: 20021454 [TBL] [Abstract][Full Text] [Related]
20. A silent H-bond can be mutationally activated for high-affinity interaction of BMP-2 and activin type IIB receptor. Weber D; Kotzsch A; Nickel J; Harth S; Seher A; Mueller U; Sebald W; Mueller TD BMC Struct Biol; 2007 Feb; 7():6. PubMed ID: 17295905 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]