307 related articles for article (PubMed ID: 20934347)
1. Anti-leishmanial and anti-trypanosomal activities of 1,4-dihydropyridines: In vitro evaluation and structure-activity relationship study.
Reimão JQ; Scotti MT; Tempone AG
Bioorg Med Chem; 2010 Nov; 18(22):8044-53. PubMed ID: 20934347
[TBL] [Abstract][Full Text] [Related]
2. In vitro and experimental therapeutic studies of the calcium channel blocker bepridil: detection of viable Leishmania (L.) chagasi by real-time PCR.
Reimão JQ; Colombo FA; Pereira-Chioccola VL; Tempone AG
Exp Parasitol; 2011 Jun; 128(2):111-5. PubMed ID: 21354141
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and in vitro evaluation of leishmanicidal and trypanocidal activities of N-quinolin-8-yl-arylsulfonamides.
da Silva LE; Joussef AC; Pacheco LK; da Silva DG; Steindel M; Rebelo RA; Schmidt B
Bioorg Med Chem; 2007 Dec; 15(24):7553-60. PubMed ID: 17889546
[TBL] [Abstract][Full Text] [Related]
4. Phenyl substitution of furamidine markedly potentiates its anti-parasitic activity against Trypanosoma cruzi and Leishmania amazonensis.
De Souza EM; Lansiaux A; Bailly C; Wilson WD; Hu Q; Boykin DW; Batista MM; Araújo-Jorge TC; Soeiro MN
Biochem Pharmacol; 2004 Aug; 68(4):593-600. PubMed ID: 15276066
[TBL] [Abstract][Full Text] [Related]
5. In vitro antileishmanial and antitrypanosomal activities of flavanones from Baccharis retusa DC. (Asteraceae).
Grecco Sdos S; Reimão JQ; Tempone AG; Sartorelli P; Cunha RL; Romoff P; Ferreira MJ; Fávero OA; Lago JH
Exp Parasitol; 2012 Feb; 130(2):141-5. PubMed ID: 22143090
[TBL] [Abstract][Full Text] [Related]
6. SAR studies on azasterols as potential anti-trypanosomal and anti-leishmanial agents.
Gigante F; Kaiser M; Brun R; Gilbert IH
Bioorg Med Chem; 2009 Aug; 17(16):5950-61. PubMed ID: 19620005
[TBL] [Abstract][Full Text] [Related]
7. The potential effects of new synthetic drugs against Leishmania amazonensis and Trypanosoma cruzi.
Canto-Cavalheiro MM; Echevarria A; Araujo CA; Bravo MF; Santos LH; Jansen AM; Leon LL
Microbios; 1997; 90(362):51-60. PubMed ID: 9301071
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and characterization of a pyridine-2-thiol N-oxide gold(I) complex with potent antiproliferative effect against Trypanosoma cruzi and Leishmania sp. insight into its mechanism of action.
Vieites M; Smircich P; Guggeri L; Marchán E; Gómez-Barrio A; Navarro M; Garat B; Gambino D
J Inorg Biochem; 2009 Oct; 103(10):1300-6. PubMed ID: 19361864
[TBL] [Abstract][Full Text] [Related]
9. Synthesis, structural elucidation and in vitro antiparasitic activity against Trypanosoma cruzi and Leishmania chagasi parasites of novel tetrahydro-1-benzazepine derivatives.
Gómez-Ayala S; Castrillón JA; Palma A; Leal SM; Escobar P; Bahsas A
Bioorg Med Chem; 2010 Jul; 18(13):4721-39. PubMed ID: 20627590
[TBL] [Abstract][Full Text] [Related]
10. Anti-malarial, anti-trypanosomal, and anti-leishmanial activities of jacaranone isolated from Pentacalia desiderabilis (Vell.) Cuatrec. (Asteraceae).
Morais TR; Romoff P; Fávero OA; Reimão JQ; Lourenço WC; Tempone AG; Hristov AD; Di Santi SM; Lago JH; Sartorelli P; Ferreira MJ
Parasitol Res; 2012 Jan; 110(1):95-101. PubMed ID: 21614544
[TBL] [Abstract][Full Text] [Related]
11. Vanadium polypyridyl compounds as potential antiparasitic and antitumoral agents: new achievements.
Benítez J; Becco L; Correia I; Leal SM; Guiset H; Pessoa JC; Lorenzo J; Tanco S; Escobar P; Moreno V; Garat B; Gambino D
J Inorg Biochem; 2011 Feb; 105(2):303-12. PubMed ID: 21194632
[TBL] [Abstract][Full Text] [Related]
12. In vitro and in vivo antitrypanosomatid activity of 5-nitroindazoles.
Boiani L; Gerpe A; Arán VJ; Torres de Ortiz S; Serna E; Vera de Bilbao N; Sanabria L; Yaluff G; Nakayama H; Rojas de Arias A; Maya JD; Morello JA; Cerecetto H; González M
Eur J Med Chem; 2009 Mar; 44(3):1034-40. PubMed ID: 18706738
[TBL] [Abstract][Full Text] [Related]
13. Synthesis and in vitro antiprotozoal activities of water-soluble, inexpensive 3,7-bis(dialkylamino)phenoxazin-5-ium derivatives.
Ge JF; Arai C; Kaiser M; Wittlin S; Brun R; Ihara M
J Med Chem; 2008 Jun; 51(12):3654-8. PubMed ID: 18476684
[TBL] [Abstract][Full Text] [Related]
14. Leishmanicidal activity of an alkenylphenol from Piper malacophyllum is related to plasma membrane disruption.
de Oliveira A; Mesquita JT; Tempone AG; Lago JH; Guimarães EF; Kato MJ
Exp Parasitol; 2012 Nov; 132(3):383-7. PubMed ID: 22981719
[TBL] [Abstract][Full Text] [Related]
15. Triclosan-caffeic acid hybrids: Synthesis, leishmanicidal, trypanocidal and cytotoxic activities.
Otero E; García E; Palacios G; Yepes LM; Carda M; Agut R; Vélez ID; Cardona WI; Robledo SM
Eur J Med Chem; 2017 Dec; 141():73-83. PubMed ID: 29028533
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and biological evaluation of novel 2,3-disubstituted quinoxaline derivatives as antileishmanial and antitrypanosomal agents.
Cogo J; Kaplum V; Sangi DP; Ueda-Nakamura T; Corrêa AG; Nakamura CV
Eur J Med Chem; 2015 Jan; 90():107-23. PubMed ID: 25461316
[TBL] [Abstract][Full Text] [Related]
17. Trypanoside, anti-tuberculosis, leishmanicidal, and cytotoxic activities of tetrahydrobenzothienopyrimidines.
Aponte JC; Vaisberg AJ; Castillo D; Gonzalez G; Estevez Y; Arevalo J; Quiliano M; Zimic M; Verástegui M; Málaga E; Gilman RH; Bustamante JM; Tarleton RL; Wang Y; Franzblau SG; Pauli GF; Sauvain M; Hammond GB
Bioorg Med Chem; 2010 Apr; 18(8):2880-6. PubMed ID: 20356752
[TBL] [Abstract][Full Text] [Related]
18. 2H-benzimidazole 1,3-dioxide derivatives: a new family of water-soluble anti-trypanosomatid agents.
Boiani M; Boiani L; Denicola A; Torres de Ortiz S; Serna E; Vera de Bilbao N; Sanabria L; Yaluff G; Nakayama H; Rojas de Arias A; Vega C; Rolan M; Gómez-Barrio A; Cerecetto H; Gonzalez M
J Med Chem; 2006 Jun; 49(11):3215-24. PubMed ID: 16722639
[TBL] [Abstract][Full Text] [Related]
19. In vitro and in vivo antileishmanial and trypanocidal studies of new N-benzene- and N-naphthalenesulfonamide derivatives.
Galiana-Roselló C; Bilbao-Ramos P; Dea-Ayuela MA; Rolón M; Vega C; Bolás-Fernández F; García-España E; Alfonso J; Coronel C; González-Rosende ME
J Med Chem; 2013 Nov; 56(22):8984-98. PubMed ID: 24151871
[TBL] [Abstract][Full Text] [Related]
20. Structure-activity relationships for the antileishmanial and antitrypanosomal activities of 1'-substituted 9-anilinoacridines.
Gamage SA; Figgitt DP; Wojcik SJ; Ralph RK; Ransijn A; Mauel J; Yardley V; Snowdon D; Croft SL; Denny WA
J Med Chem; 1997 Aug; 40(16):2634-42. PubMed ID: 9258370
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]