250 related articles for article (PubMed ID: 20947021)
1. Hydrogen/deuterium exchange reveals distinct agonist/partial agonist receptor dynamics within vitamin D receptor/retinoid X receptor heterodimer.
Zhang J; Chalmers MJ; Stayrook KR; Burris LL; Garcia-Ordonez RD; Pascal BD; Burris TP; Dodge JA; Griffin PR
Structure; 2010 Oct; 18(10):1332-41. PubMed ID: 20947021
[TBL] [Abstract][Full Text] [Related]
2. HDX reveals the conformational dynamics of DNA sequence specific VDR co-activator interactions.
Zheng J; Chang MR; Stites RE; Wang Y; Bruning JB; Pascal BD; Novick SJ; Garcia-Ordonez RD; Stayrook KR; Chalmers MJ; Dodge JA; Griffin PR
Nat Commun; 2017 Oct; 8(1):923. PubMed ID: 29030554
[TBL] [Abstract][Full Text] [Related]
3. 25-Dehydro-1alpha-hydroxyvitamin D3-26,23S-lactone antagonizes the nuclear vitamin D receptor by mediating a unique noncovalent conformational change.
Bula CM; Bishop JE; Ishizuka S; Norman AW
Mol Endocrinol; 2000 Nov; 14(11):1788-96. PubMed ID: 11075812
[TBL] [Abstract][Full Text] [Related]
4. DNA binding alters coactivator interaction surfaces of the intact VDR-RXR complex.
Zhang J; Chalmers MJ; Stayrook KR; Burris LL; Wang Y; Busby SA; Pascal BD; Garcia-Ordonez RD; Bruning JB; Istrate MA; Kojetin DJ; Dodge JA; Burris TP; Griffin PR
Nat Struct Mol Biol; 2011 May; 18(5):556-63. PubMed ID: 21478866
[TBL] [Abstract][Full Text] [Related]
5. Critical role of helix 12 of the vitamin D(3) receptor for the partial agonism of carboxylic ester antagonists.
Väisänen S; Peräkylä M; Kärkkäinen JI; Steinmeyer A; Carlberg C
J Mol Biol; 2002 Jan; 315(2):229-38. PubMed ID: 11779241
[TBL] [Abstract][Full Text] [Related]
6. Discovery of Nuclear Receptor Ligands and Elucidation of Their Mechanisms of Action.
Yamamoto K
Chem Pharm Bull (Tokyo); 2019; 67(7):609-619. PubMed ID: 31257315
[TBL] [Abstract][Full Text] [Related]
7. Dynamic and ligand-selective interactions of vitamin D receptor with retinoid X receptor and cofactors in living cells.
Choi M; Yamada S; Makishima M
Mol Pharmacol; 2011 Dec; 80(6):1147-55. PubMed ID: 21917910
[TBL] [Abstract][Full Text] [Related]
8. 1,25-Dihydroxyvitamin D3 stimulates cyclic vitamin D receptor/retinoid X receptor DNA-binding, co-activator recruitment, and histone acetylation in intact osteoblasts.
Kim S; Shevde NK; Pike JW
J Bone Miner Res; 2005 Feb; 20(2):305-17. PubMed ID: 15647825
[TBL] [Abstract][Full Text] [Related]
9. New understanding of the molecular mechanism of receptor-mediated genomic actions of the vitamin D hormone.
Haussler MR; Jurutka PW; Hsieh JC; Thompson PD; Selznick SH; Haussler CA; Whitfield GK
Bone; 1995 Aug; 17(2 Suppl):33S-38S. PubMed ID: 8579895
[TBL] [Abstract][Full Text] [Related]
10. 22S-butyl-1alpha,24R-dihydroxyvitamin D3: recovery of vitamin D receptor agonistic activity.
Inaba Y; Nakabayashi M; Itoh T; Yoshimoto N; Ikura T; Ito N; Shimizu M; Yamamoto K
J Steroid Biochem Mol Biol; 2010 Jul; 121(1-2):146-50. PubMed ID: 20211257
[TBL] [Abstract][Full Text] [Related]
11. Agonist-triggered modulation of the activated and silent state of the vitamin D(3) receptor by interaction with co-repressors and co-activators.
Herdick M; Carlberg C
J Mol Biol; 2000 Dec; 304(5):793-801. PubMed ID: 11124027
[TBL] [Abstract][Full Text] [Related]
12. Structural Analysis of VDR Complex with ZK168281 Antagonist.
Belorusova AY; Chalhoub S; Rovito D; Rochel N
J Med Chem; 2020 Sep; 63(17):9457-9463. PubMed ID: 32787090
[TBL] [Abstract][Full Text] [Related]
13. Fine tuning of agonistic/antagonistic activity for vitamin D receptor by 22-alkyl chain length of ligands: 22S-Hexyl compound unexpectedly restored agonistic activity.
Anami Y; Sakamaki Y; Itoh T; Inaba Y; Nakabayashi M; Ikura T; Ito N; Yamamoto K
Bioorg Med Chem; 2015 Nov; 23(22):7274-81. PubMed ID: 26515040
[TBL] [Abstract][Full Text] [Related]
14. Corepressor excess shifts the two-side chain vitamin D analog Gemini from an agonist to an inverse agonist of the vitamin D receptor.
Gonzalez MM; Samenfeld P; Peräkylä M; Carlberg C
Mol Endocrinol; 2003 Oct; 17(10):2028-38. PubMed ID: 12843209
[TBL] [Abstract][Full Text] [Related]
15. The crystal structure of the nuclear receptor for vitamin D bound to its natural ligand.
Rochel N; Wurtz JM; Mitschler A; Klaholz B; Moras D
Mol Cell; 2000 Jan; 5(1):173-9. PubMed ID: 10678179
[TBL] [Abstract][Full Text] [Related]
16. Hairless modulates ligand-dependent activation of the vitamin D receptor-retinoid X receptor heterodimer.
Chuma M; Endo-Umeda K; Shimba S; Yamada S; Makishima M
Biol Pharm Bull; 2012; 35(4):582-7. PubMed ID: 22466564
[TBL] [Abstract][Full Text] [Related]
17. Carboxylic ester antagonists of 1alpha,25-dihydroxyvitamin D(3) show cell-specific actions.
Herdick M; Steinmeyer A; Carlberg C
Chem Biol; 2000 Nov; 7(11):885-94. PubMed ID: 11094341
[TBL] [Abstract][Full Text] [Related]
18. Retinoid X receptor is a nonsilent major contributor to vitamin D receptor-mediated transcriptional activation.
Bettoun DJ; Burris TP; Houck KA; Buck DW; Stayrook KR; Khalifa B; Lu J; Chin WW; Nagpal S
Mol Endocrinol; 2003 Nov; 17(11):2320-8. PubMed ID: 12893883
[TBL] [Abstract][Full Text] [Related]
19. Vitamin D receptors from patients with resistance to 1,25-dihydroxyvitamin D3: point mutations confer reduced transactivation in response to ligand and impaired interaction with the retinoid X receptor heterodimeric partner.
Whitfield GK; Selznick SH; Haussler CA; Hsieh JC; Galligan MA; Jurutka PW; Thompson PD; Lee SM; Zerwekh JE; Haussler MR
Mol Endocrinol; 1996 Dec; 10(12):1617-31. PubMed ID: 8961271
[TBL] [Abstract][Full Text] [Related]
20. Molecular basis of the selective activity of vitamin D analogues.
Carlberg C
J Cell Biochem; 2003 Feb; 88(2):274-81. PubMed ID: 12520526
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]