BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

129 related articles for article (PubMed ID: 21028940)

  • 1. The evaluation of novel natural products as inhibitors of human glutathione transferase P1-1.
    Mukanganyama S; Bezabih M; Robert M; Ngadjui BT; Kapche GF; Ngandeu F; Abegaz B
    J Enzyme Inhib Med Chem; 2011 Aug; 26(4):460-7. PubMed ID: 21028940
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Potent isozyme-selective inhibition of human glutathione S-transferase A1-1 by a novel glutathione S-conjugate.
    Cacciatore I; Caccuri AM; Cocco A; De Maria F; Di Stefano A; Luisi G; Pinnen F; Ricci G; Sozio P; Turella P
    Amino Acids; 2005 Nov; 29(3):255-61. PubMed ID: 16082503
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Glutathione transferase from Plasmodium falciparum--interaction with malagashanine and selected plant natural products.
    Mangoyi R; Hayeshi R; Ngadjui B; Ngandeu F; Bezabih M; Abegaz B; Razafimahefa S; Rasoanaivo P; Mukanganyama S
    J Enzyme Inhib Med Chem; 2010 Dec; 25(6):854-62. PubMed ID: 20521884
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Online biochemical detection of glutathione-S-transferase P1-specific inhibitors in complex mixtures.
    Kool J; Eggink M; van Rossum H; van Liempd SM; van Elswijk DA; Irth H; Commandeur JN; Meerman JH; Vermeulen NP
    J Biomol Screen; 2007 Apr; 12(3):396-405. PubMed ID: 17379858
    [TBL] [Abstract][Full Text] [Related]  

  • 5. The inhibition of human glutathione S-transferases activity by plant polyphenolic compounds ellagic acid and curcumin.
    Hayeshi R; Mutingwende I; Mavengere W; Masiyanise V; Mukanganyama S
    Food Chem Toxicol; 2007 Feb; 45(2):286-95. PubMed ID: 17046132
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Inhibition of human glutathione S-transferases by curcumin and analogues.
    Appiah-Opong R; Commandeur JN; Istyastono E; Bogaards JJ; Vermeulen NP
    Xenobiotica; 2009 Apr; 39(4):302-11. PubMed ID: 19350453
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Tocotrienols inhibit human glutathione S-transferase P1-1.
    van Haaften RI; Haenen GR; Evelo CT; Bast A
    IUBMB Life; 2002 Aug; 54(2):81-4. PubMed ID: 12440523
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Isoenzyme- and allozyme-specific inhibitors: 2,2'-dihydroxybenzophenones and their carbonyl N-analogues that discriminate between human glutathione transferase A1-1 and P1-1 allozymes.
    Pouliou FM; Thireou TN; Eliopoulos EE; Tsoungas PG; Labrou NE; Clonis YD
    Chem Biol Drug Des; 2015 Nov; 86(5):1055-63. PubMed ID: 25891019
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Peptide-bond modified glutathione conjugate analogs modulate GSTpi function in GSH-conjugation, drug sensitivity and JNK signaling.
    Burg D; Riepsaame J; Pont C; Mulder G; van de Water B
    Biochem Pharmacol; 2006 Jan; 71(3):268-77. PubMed ID: 16337611
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Identifying and characterizing binding sites on the irreversible inhibition of human glutathione S-transferase P1-1 by S-thiocarbamoylation.
    Quesada-Soriano I; Primavera A; Casas-Solvas JM; Téllez-Sanz R; Barón C; Vargas-Berenguel A; Lo Bello M; García-Fuentes L
    Chembiochem; 2012 Jul; 13(11):1594-604. PubMed ID: 22740430
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Characterization of bromosulphophthalein binding to human glutathione S-transferase A1-1: thermodynamics and inhibition kinetics.
    Kolobe D; Sayed Y; Dirr HW
    Biochem J; 2004 Sep; 382(Pt 2):703-9. PubMed ID: 15147239
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Concluding the trilogy: The interaction of 2,2'-dihydroxy-benzophenones and their carbonyl N-analogues with human glutathione transferase M1-1 face to face with the P1-1 and A1-1 isoenzymes involved in MDR.
    Georgakis ND; Karagiannopoulos DA; Thireou TN; Eliopoulos EE; Labrou NE; Tsoungas PG; Koutsilieris MN; Clonis YD
    Chem Biol Drug Des; 2017 Nov; 90(5):900-908. PubMed ID: 28440951
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Mechanistic studies of inactivation of glutathione S-transferase Pi isozyme by a haloenol lactone derivative.
    Zheng J; Liu G; Tozkoparan B; Wen D
    Med Chem; 2005 Mar; 1(2):191-8. PubMed ID: 16787314
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Novel oxadiazole analogues derived from ethacrynic acid: design, synthesis, and structure-activity relationships in inhibiting the activity of glutathione S-transferase P1-1 and cancer cell proliferation.
    Yang X; Liu G; Li H; Zhang Y; Song D; Li C; Wang R; Liu B; Liang W; Jing Y; Zhao G
    J Med Chem; 2010 Feb; 53(3):1015-22. PubMed ID: 20055416
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Design, synthesis, and structure-activity relationships of haloenol lactones: site-directed and isozyme-selective glutathione S-transferase inhibitors.
    Wu Z; Minhas GS; Wen D; Jiang H; Chen K; Zimniak P; Zheng J
    J Med Chem; 2004 Jun; 47(12):3282-94. PubMed ID: 15163208
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Studies of glutathione transferase P1-1 bound to a platinum(IV)-based anticancer compound reveal the molecular basis of its activation.
    Parker LJ; Italiano LC; Morton CJ; Hancock NC; Ascher DB; Aitken JB; Harris HH; Campomanes P; Rothlisberger U; De Luca A; Lo Bello M; Ang WH; Dyson PJ; Parker MW
    Chemistry; 2011 Jul; 17(28):7806-16. PubMed ID: 21681839
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Amitriptyline may have a supportive role in cancer treatment by inhibiting glutathione S-transferase pi (GST-π) and alpha (GST-α).
    Kulaksiz-Erkmen G; Dalmizrak O; Dincsoy-Tuna G; Dogan A; Ogus IH; Ozer N
    J Enzyme Inhib Med Chem; 2013 Feb; 28(1):131-6. PubMed ID: 22145766
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Purification and biochemical characterization of glutathione S-transferase from Down syndrome and normal children erythrocytes: a comparative study.
    Hamed RR; Maharem TM; Abdel-Meguid N; Sabry GM; Abdalla AM; Guneidy RA
    Res Dev Disabil; 2011; 32(5):1470-82. PubMed ID: 21377322
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Nitrobenzoxadiazole-based GSTP1-1 inhibitors containing the full peptidyl moiety of (pseudo)glutathione.
    Luisi G; Mollica A; Carradori S; Lenoci A; De Luca A; Caccuri AM
    J Enzyme Inhib Med Chem; 2016 Dec; 31(6):924-30. PubMed ID: 26329912
    [TBL] [Abstract][Full Text] [Related]  

  • 20. The synthesis of alpha,beta-unsaturated carbonyl derivatives with the ability to inhibit both glutathione S-transferase P1-1 activity and the proliferation of leukemia cells.
    Zhao G; Liu C; Wang R; Song D; Wang X; Lou H; Jing Y
    Bioorg Med Chem; 2007 Apr; 15(7):2701-7. PubMed ID: 17287120
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.