343 related articles for article (PubMed ID: 21044845)
1. Design, synthesis and in vitro antimalarial evaluation of triazole-linked chalcone and dienone hybrid compounds.
Guantai EM; Ncokazi K; Egan TJ; Gut J; Rosenthal PJ; Smith PJ; Chibale K
Bioorg Med Chem; 2010 Dec; 18(23):8243-56. PubMed ID: 21044845
[TBL] [Abstract][Full Text] [Related]
2. 7-Chloroquinolinotriazoles: synthesis by the azide-alkyne cycloaddition click chemistry, antimalarial activity, cytotoxicity and SAR studies.
Pereira GR; Brandão GC; Arantes LM; de Oliveira HA; de Paula RC; do Nascimento MF; dos Santos FM; da Rocha RK; Lopes JC; de Oliveira AB
Eur J Med Chem; 2014 Feb; 73():295-309. PubMed ID: 24469080
[TBL] [Abstract][Full Text] [Related]
3. Azide-alkyne cycloaddition en route to 1H-1,2,3-triazole-tethered 7-chloroquinoline-isatin chimeras: synthesis and antimalarial evaluation.
Raj R; Singh P; Singh P; Gut J; Rosenthal PJ; Kumar V
Eur J Med Chem; 2013 Apr; 62():590-6. PubMed ID: 23434528
[TBL] [Abstract][Full Text] [Related]
4. Synthesis and evaluation of new antimalarial phenylurenyl chalcone derivatives.
Domínguez JN; León C; Rodrigues J; Gamboa de Domínguez N; Gut J; Rosenthal PJ
J Med Chem; 2005 May; 48(10):3654-8. PubMed ID: 15887974
[TBL] [Abstract][Full Text] [Related]
5. 1H-1,2,3-Triazole-tethered isatin-7-chloroquinoline and 3-hydroxy-indole-7-chloroquinoline conjugates: synthesis and antimalarial evaluation.
Raj R; Gut J; Rosenthal PJ; Kumar V
Bioorg Med Chem Lett; 2014 Feb; 24(3):756-9. PubMed ID: 24424135
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and in vitro evaluation of new chloroquine-chalcone hybrids against chloroquine-resistant strain of Plasmodium falciparum.
Sashidhara KV; Avula SR; Palnati GR; Singh SV; Srivastava K; Puri SK; Saxena JK
Bioorg Med Chem Lett; 2012 Sep; 22(17):5455-9. PubMed ID: 22850213
[TBL] [Abstract][Full Text] [Related]
7. Comparison of the antiplasmodial and falcipain-2 inhibitory activity of beta-amino alcohol thiolactone-chalcone and isatin-chalcone hybrids.
Hans RH; Gut J; Rosenthal PJ; Chibale K
Bioorg Med Chem Lett; 2010 Apr; 20(7):2234-7. PubMed ID: 20206517
[TBL] [Abstract][Full Text] [Related]
8. In vitro efficacy of 7-benzylamino-1-isoquinolinamines against Plasmodium falciparum related to the efficacy of chalcones.
Gutteridge CE; Hoffman MM; Bhattacharjee AK; Milhous WK; Gerena L
Bioorg Med Chem Lett; 2011 Jan; 21(2):786-9. PubMed ID: 21168330
[TBL] [Abstract][Full Text] [Related]
9. Stilbene-chalcone hybrids: design, synthesis, and evaluation as a new class of antimalarial scaffolds that trigger cell death through stage specific apoptosis.
Sharma N; Mohanakrishnan D; Shard A; Sharma A; Saima ; Sinha AK; Sahal D
J Med Chem; 2012 Jan; 55(1):297-311. PubMed ID: 22098429
[TBL] [Abstract][Full Text] [Related]
10. Synthesis of 4-aminoquinoline-1,2,3-triazole and 4-aminoquinoline-1,2,3-triazole-1,3,5-triazine hybrids as potential antimalarial agents.
Manohar S; Khan SI; Rawat DS
Chem Biol Drug Des; 2011 Jul; 78(1):124-36. PubMed ID: 21457474
[TBL] [Abstract][Full Text] [Related]
11. In vitro antimalarial activity, β-haematin inhibition and structure-activity relationships in a series of quinoline triazoles.
Joshi MC; Wicht KJ; Taylor D; Hunter R; Smith PJ; Egan TJ
Eur J Med Chem; 2013 Nov; 69():338-47. PubMed ID: 24077524
[TBL] [Abstract][Full Text] [Related]
12. In vitro antiplasmodial activity of prenylated chalcone derivatives of hops (Humulus lupulus) and their interaction with haemin.
Frölich S; Schubert C; Bienzle U; Jenett-Siems K
J Antimicrob Chemother; 2005 Jun; 55(6):883-7. PubMed ID: 15824094
[TBL] [Abstract][Full Text] [Related]
13. Synthesis, antimalarial and antitubercular activity of acetylenic chalcones.
Hans RH; Guantai EM; Lategan C; Smith PJ; Wan B; Franzblau SG; Gut J; Rosenthal PJ; Chibale K
Bioorg Med Chem Lett; 2010 Feb; 20(3):942-4. PubMed ID: 20045640
[TBL] [Abstract][Full Text] [Related]
14. Piperazine-linked 4-aminoquinoline-chalcone/ferrocenyl-chalcone conjugates: Synthesis and antiplasmodial evaluation.
Singh A; Rani A; Gut J; Rosenthal PJ; Kumar V
Chem Biol Drug Des; 2017 Oct; 90(4):590-595. PubMed ID: 28332319
[TBL] [Abstract][Full Text] [Related]
15. Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline.
Delarue-Cochin S; Grellier P; Maes L; Mouray E; Sergheraert C; Melnyk P
Eur J Med Chem; 2008 Oct; 43(10):2045-55. PubMed ID: 18226428
[TBL] [Abstract][Full Text] [Related]
16. Application of multicomponent reactions to antimalarial drug discovery. Part 3: discovery of aminoxazole 4-aminoquinolines with potent antiplasmodial activity in vitro.
Musonda CC; Little S; Yardley V; Chibale K
Bioorg Med Chem Lett; 2007 Sep; 17(17):4733-6. PubMed ID: 17644333
[TBL] [Abstract][Full Text] [Related]
17. 4-Aminoquinoline-ferrocenyl-chalcone conjugates: Synthesis and anti-plasmodial evaluation.
Singh A; Gut J; Rosenthal PJ; Kumar V
Eur J Med Chem; 2017 Jan; 125():269-277. PubMed ID: 27688182
[TBL] [Abstract][Full Text] [Related]
18. Synthesis and antimalarial evaluation of novel isocryptolepine derivatives.
Whittell LR; Batty KT; Wong RP; Bolitho EM; Fox SA; Davis TM; Murray PE
Bioorg Med Chem; 2011 Dec; 19(24):7519-25. PubMed ID: 22055713
[TBL] [Abstract][Full Text] [Related]
19. Design and synthesis of new antimalarial agents from 4-aminoquinoline.
Solomon VR; Puri SK; Srivastava K; Katti SB
Bioorg Med Chem; 2005 Mar; 13(6):2157-65. PubMed ID: 15727868
[TBL] [Abstract][Full Text] [Related]
20. Bisquinolines. 2. Antimalarial N,N-bis(7-chloroquinolin-4-yl)heteroalkanediamines.
Vennerstrom JL; Ager AL; Dorn A; Andersen SL; Gerena L; Ridley RG; Milhous WK
J Med Chem; 1998 Oct; 41(22):4360-4. PubMed ID: 9784111
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
