BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

160 related articles for article (PubMed ID: 21055434)

  • 1. Synthesis and antinociceptive effects of endomorphin-1 analogs with C-terminal linked by oligoarginine.
    Wang CL; Guo C; Wang YQ; Zhou Y; Li Q; Ni JM; Wang R
    Peptides; 2011 Feb; 32(2):293-9. PubMed ID: 21055434
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Endomorphin-1 analogs with oligoarginine-conjugation at C-terminus produce potent antinociception with reduced opioid tolerance in paw withdrawal test.
    Yuan BY; Liu WZ; Wang XF; Zhang YZ; Yang DJ; Wang CL
    Peptides; 2018 Aug; 106():96-101. PubMed ID: 30016700
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Utilization of combined chemical modifications to enhance the blood-brain barrier permeability and pharmacological activity of endomorphin-1.
    Liu HM; Liu XF; Yao JL; Wang CL; Yu Y; Wang R
    J Pharmacol Exp Ther; 2006 Oct; 319(1):308-16. PubMed ID: 16803861
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Novel endomorphin-1 analogs with C-terminal oligoarginine-conjugation display systemic antinociceptive activity with less gastrointestinal side effects.
    Wang CL; Qiu TT; Diao YX; Zhang Y; Gu N
    Biochimie; 2015 Sep; 116():24-33. PubMed ID: 26115815
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and biological evaluation of cyclic endomorphin-2 analogs.
    Perlikowska R; do-Rego JC; Cravezic A; Fichna J; Wyrebska A; Toth G; Janecka A
    Peptides; 2010 Feb; 31(2):339-45. PubMed ID: 19995587
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Characterization of opioid activities of endomorphin analogs with C-terminal amide to hydrazide conversion.
    Wang CL; Ren YK; Xiang Q; Wang Y; Gu N; Lu C; Wang R
    Neuropeptides; 2013 Oct; 47(5):297-304. PubMed ID: 24084335
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Identification of opioid ligands possessing mixed micro agonist/delta antagonist activity among pyridomorphinans derived from naloxone, oxymorphone, and hydromorphone [correction of hydropmorphone].
    Ananthan S; Khare NK; Saini SK; Seitz LE; Bartlett JL; Davis P; Dersch CM; Porreca F; Rothman RB; Bilsky EJ
    J Med Chem; 2004 Mar; 47(6):1400-12. PubMed ID: 14998329
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Peripheral antinociceptive effects of the cyclic endomorphin-1 analog c[YpwFG] in a mouse visceral pain model.
    Bedini A; Baiula M; Gentilucci L; Tolomelli A; De Marco R; Spampinato S
    Peptides; 2010 Nov; 31(11):2135-40. PubMed ID: 20713109
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Development of potent mu-opioid receptor ligands using unique tyrosine analogues of endomorphin-2.
    Li T; Fujita Y; Tsuda Y; Miyazaki A; Ambo A; Sasaki Y; Jinsmaa Y; Bryant SD; Lazarus LH; Okada Y
    J Med Chem; 2005 Jan; 48(2):586-92. PubMed ID: 15658871
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Involvement of mu-opioid receptors in antinociception and inhibition of gastrointestinal transit induced by 7-hydroxymitragynine, isolated from Thai herbal medicine Mitragyna speciosa.
    Matsumoto K; Hatori Y; Murayama T; Tashima K; Wongseripipatana S; Misawa K; Kitajima M; Takayama H; Horie S
    Eur J Pharmacol; 2006 Nov; 549(1-3):63-70. PubMed ID: 16978601
    [TBL] [Abstract][Full Text] [Related]  

  • 11. In vitro and in vivo characterization of opioid activities of C-terminal esterified endomorphin-2 analogs.
    Wang CL; Guo C; Zhou Y; Wang R
    Peptides; 2009 Sep; 30(9):1697-704. PubMed ID: 19520129
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Endomorphin-2 analogs with C-terminal esterification produce potent systemic antinociception with reduced tolerance and gastrointestinal side effects.
    Wang CL; Qiu TT; Yang DJ; Yuan BY; Han FT; Li L; Gu N
    Neuropharmacology; 2017 Apr; 116():98-109. PubMed ID: 28042019
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Conformationally constrained deltorphin analogs with 2-aminotetralin-2-carboxylic acid in position 3.
    Tóth G; Darula Z; Péter A; Fülöp F; Tourwé D; Jaspers H; Verheyden P; Böcskey Z; Tóth Z; Borsodi A
    J Med Chem; 1997 Mar; 40(6):990-5. PubMed ID: 9083489
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Endomorphin 1[psi] and endomorphin 2[psi], endomorphins analogues containing a reduced (CH2NH) amide bond between Tyr1 and Pro2, display partial agonist potency but significant antinociception.
    Zhao QY; Chen Q; Yang DJ; Feng Y; Long Y; Wang P; Wang R
    Life Sci; 2005 Jul; 77(10):1155-65. PubMed ID: 15878600
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Enhancement of morphine antinociception by a CCKB antagonist in mice is mediated via opioid delta receptors.
    Vanderah TW; Bernstein RN; Yamamura HI; Hruby VJ; Porreca F
    J Pharmacol Exp Ther; 1996 Jul; 278(1):212-9. PubMed ID: 8764354
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Local peripheral antinociceptive effects of 14-O-methyloxymorphone derivatives in inflammatory and neuropathic pain in the rat.
    Obara I; Makuch W; Spetea M; Schütz J; Schmidhammer H; Przewlocki R; Przewlocka B
    Eur J Pharmacol; 2007 Mar; 558(1-3):60-7. PubMed ID: 17204264
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Melatonin enhances antinociceptive effects of delta-, but not mu-opioid agonist in mice.
    Li SR; Wang T; Wang R; Dai X; Chen Q; Li RD
    Brain Res; 2005 May; 1043(1-2):132-8. PubMed ID: 15862526
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Opioid receptor affinity and analgesic activity of O- and C-glycosylated opioid peptides.
    Negri L; Melchiorri P; Rocchi R; Scolaro B
    Acta Physiol Hung; 1996; 84(4):441-3. PubMed ID: 9328626
    [TBL] [Abstract][Full Text] [Related]  

  • 19. DAMGO and 6beta-glycine substituted 14-O-methyloxymorphone but not morphine show peripheral, preemptive antinociception after systemic administration in a mouse visceral pain model and high intrinsic efficacy in the isolated rat vas deferens.
    Al-Khrasani M; Spetea M; Friedmann T; Riba P; Király K; Schmidhammer H; Furst S
    Brain Res Bull; 2007 Oct; 74(5):369-75. PubMed ID: 17845912
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis and antinociceptive activity of cyclic endomorphin-2 and morphiceptin analogs.
    Janecka A; Fichna J; Kruszynski R; Sasaki Y; Ambo A; Costentin J; do-Rego JC
    Biochem Pharmacol; 2005 Dec; 71(1-2):188-95. PubMed ID: 16288997
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.